HK1217195A1 - Propane i sulfonic acid 3 [5 (4 chloro phenyl) 1h pyrrolo [2, 3 b pyridine 3 carbonyl] 2, 4 difluoro phenyl amide compositions and uses thereof 1 3 [5 (4 ) 1h [23 b] 3 ] 24 - Google Patents

Propane i sulfonic acid 3 [5 (4 chloro phenyl) 1h pyrrolo [2, 3 b pyridine 3 carbonyl] 2, 4 difluoro phenyl amide compositions and uses thereof 1 3 [5 (4 ) 1h [23 b] 3 ] 24

Info

Publication number
HK1217195A1
HK1217195A1 HK16105154.3A HK16105154A HK1217195A1 HK 1217195 A1 HK1217195 A1 HK 1217195A1 HK 16105154 A HK16105154 A HK 16105154A HK 1217195 A1 HK1217195 A1 HK 1217195A1
Authority
HK
Hong Kong
Prior art keywords
pyrrolo
propane
carbonyl
pyridine
phenyl
Prior art date
Application number
HK16105154.3A
Other languages
Chinese (zh)
Inventor
Dipen Desai
Ralph Diodone
Zenaida Go
Prabha N Ibrahim
Raman Mahadevan Iyer
Hans-Juergen Mair
Harpreet K Sandhu
Navnit Hargovindas Shah
Gary Conard Visor
Nicole Wyttenbach
Stephan Lauper
Johannes Pudewell
Frank Wierschem
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of HK1217195A1 publication Critical patent/HK1217195A1/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0014—Skin, i.e. galenical aspects of topical compositions
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/10—Dispersions; Emulsions
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605—Excipients; Inactive ingredients
    • A61K9/1629—Organic macromolecular compounds
    • A61K9/1635—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605—Excipients; Inactive ingredients
    • A61K9/1629—Organic macromolecular compounds
    • A61K9/1652—Polysaccharides, e.g. alginate, cellulose derivatives; Cyclodextrin
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13—Crystalline forms, e.g. polymorphs

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Organic Chemistry (AREA)
  • Dermatology (AREA)
  • Dispersion Chemistry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
HK16105154.3A 2009-04-03 2016-05-05 Propane i sulfonic acid 3 [5 (4 chloro phenyl) 1h pyrrolo [2, 3 b pyridine 3 carbonyl] 2, 4 difluoro phenyl amide compositions and uses thereof 1 3 [5 (4 ) 1h [23 b] 3 ] 24 HK1217195A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US16667709P 2009-04-03 2009-04-03
US17605109P 2009-05-06 2009-05-06
EP09175665 2009-11-11

Publications (1)

Publication Number Publication Date
HK1217195A1 true HK1217195A1 (en) 2016-12-30

Family

ID=54978682

Family Applications (2)

Application Number Title Priority Date Filing Date
HK12107426.5A HK1168590A1 (en) 2009-04-03 2012-07-30 Propane- i-sulfonic acid 3- [5- (4 -chloro-phenyl) -1h-pyrrolo [2, 3-b] pyridine-3-carbonyl] -2, 4-difluoro-phenyl -amide compositions and uses thereof -1-3-[5-(4--)-1h-[23-b]-3-]-24---
HK16105154.3A HK1217195A1 (en) 2009-04-03 2016-05-05 Propane i sulfonic acid 3 [5 (4 chloro phenyl) 1h pyrrolo [2, 3 b pyridine 3 carbonyl] 2, 4 difluoro phenyl amide compositions and uses thereof 1 3 [5 (4 ) 1h [23 b] 3 ] 24

Family Applications Before (1)

Application Number Title Priority Date Filing Date
HK12107426.5A HK1168590A1 (en) 2009-04-03 2012-07-30 Propane- i-sulfonic acid 3- [5- (4 -chloro-phenyl) -1h-pyrrolo [2, 3-b] pyridine-3-carbonyl] -2, 4-difluoro-phenyl -amide compositions and uses thereof -1-3-[5-(4--)-1h-[23-b]-3-]-24---

Country Status (4)

Country Link
HK (2) HK1168590A1 (en)
HR (1) HRP20151156T1 (en)
IL (1) IL251336B (en)
JO (1) JO3056B1 (en)

Also Published As

Publication number Publication date
HK1168590A1 (en) 2013-01-04
HRP20151156T1 (en) 2016-01-01
JO3056B1 (en) 2017-03-15
IL251336A0 (en) 2017-05-29
IL251336B (en) 2020-04-30

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