HK1197229A1 - 製備蛋白酶抑制劑的方法 - Google Patents

製備蛋白酶抑制劑的方法

Info

Publication number
HK1197229A1
HK1197229A1 HK14110522A HK14110522A HK1197229A1 HK 1197229 A1 HK1197229 A1 HK 1197229A1 HK 14110522 A HK14110522 A HK 14110522A HK 14110522 A HK14110522 A HK 14110522A HK 1197229 A1 HK1197229 A1 HK 1197229A1
Authority
HK
Hong Kong
Prior art keywords
preparation
protease inhibitors
protease
inhibitors
Prior art date
Application number
HK14110522A
Other languages
English (en)
Inventor
Gerald J Tanoury
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of HK1197229A1 publication Critical patent/HK1197229A1/zh

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B53/00—Asymmetric syntheses
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/52—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring condensed with a ring other than six-membered

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
HK14110522A 2011-05-13 2014-10-22 製備蛋白酶抑制劑的方法 HK1197229A1 (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201161486150P 2011-05-13 2011-05-13
PCT/US2012/037515 WO2012158515A1 (en) 2011-05-13 2012-05-11 Process for the preparation of protease inhibitors

Publications (1)

Publication Number Publication Date
HK1197229A1 true HK1197229A1 (zh) 2015-01-09

Family

ID=46147756

Family Applications (1)

Application Number Title Priority Date Filing Date
HK14110522A HK1197229A1 (zh) 2011-05-13 2014-10-22 製備蛋白酶抑制劑的方法

Country Status (5)

Country Link
EP (1) EP2707346A1 (zh)
CN (1) CN103748059A (zh)
HK (1) HK1197229A1 (zh)
IL (1) IL229427A0 (zh)
WO (1) WO2012158515A1 (zh)

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HN2002000136A (es) * 2001-06-11 2003-07-31 Basf Ag Inhibidores de la proteasa del virus hiv, compuestos que contienen a los mismos, sus usos farmaceuticos y los materiales para su sintesis
JP2007525512A (ja) * 2004-02-27 2007-09-06 シェーリング　コーポレイション Ｃ型肝炎ウイルスｎｓ３セリンプロテアーゼのインヒビターとしての３，４−（シクロペンチル）−縮合プロリン化合物
WO2007022459A2 (en) * 2005-08-19 2007-02-22 Vertex Pharmaceuticals Incorporated Processes and intermediates
CN101611001B (zh) * 2006-12-20 2015-11-25 默沙东公司 利用亚硫酸氢盐中间体制备6,6-二甲基-3-氮杂双环-[3.1.0]-己烷化合物的方法
CN103108865A (zh) * 2010-06-03 2013-05-15 弗特克斯药品有限公司 方法和中间体

Also Published As

Publication number Publication date
WO2012158515A1 (en) 2012-11-22
IL229427A0 (en) 2014-01-30
CN103748059A (zh) 2014-04-23
EP2707346A1 (en) 2014-03-19

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