HK1131787A1 - Oxa-steroids derivatives as selective progesterone receptor modulators - Google Patents

Oxa-steroids derivatives as selective progesterone receptor modulators

Info

Publication number
HK1131787A1
HK1131787A1 HK09109803.9A HK09109803A HK1131787A1 HK 1131787 A1 HK1131787 A1 HK 1131787A1 HK 09109803 A HK09109803 A HK 09109803A HK 1131787 A1 HK1131787 A1 HK 1131787A1
Authority
HK
Hong Kong
Prior art keywords
oxa
receptor modulators
progesterone receptor
selective progesterone
steroids
Prior art date
Application number
HK09109803.9A
Other languages
English (en)
Inventor
Fu-An Kang
Nareshkumar F Jain
Zhihua Sui
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of HK1131787A1 publication Critical patent/HK1131787A1/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J73/00—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms
    • C07J73/001—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms by one hetero atom
    • C07J73/003—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms by one hetero atom by oxygen as hetero atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/18—Feminine contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/36—Antigestagens
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/38—Drugs for disorders of the endocrine system of the suprarenal hormones
    • A61P5/46—Drugs for disorders of the endocrine system of the suprarenal hormones for decreasing, blocking or antagonising the activity of glucocorticosteroids

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Gynecology & Obstetrics (AREA)
  • Emergency Medicine (AREA)
  • Pregnancy & Childbirth (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
HK09109803.9A 2006-02-17 2009-10-22 Oxa-steroids derivatives as selective progesterone receptor modulators HK1131787A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US77504206P 2006-02-17 2006-02-17
PCT/US2007/062289 WO2007098388A2 (en) 2006-02-17 2007-02-16 Oxa-steroids derivatives as selective progesterone receptor modulators

Publications (1)

Publication Number Publication Date
HK1131787A1 true HK1131787A1 (en) 2010-02-05

Family

ID=38438064

Family Applications (2)

Application Number Title Priority Date Filing Date
HK09104474.8A HK1125946A1 (en) 2006-02-17 2009-05-15 Oxa-steroids derivatives as selective progesterone receptor modulators
HK09109803.9A HK1131787A1 (en) 2006-02-17 2009-10-22 Oxa-steroids derivatives as selective progesterone receptor modulators

Family Applications Before (1)

Application Number Title Priority Date Filing Date
HK09104474.8A HK1125946A1 (en) 2006-02-17 2009-05-15 Oxa-steroids derivatives as selective progesterone receptor modulators

Country Status (14)

Country Link
US (1) US7763648B2 (xx)
EP (1) EP1991559B1 (xx)
JP (1) JP2009527494A (xx)
CN (1) CN101426806B (xx)
AU (1) AU2007217101A1 (xx)
CA (1) CA2642834C (xx)
CY (1) CY1113127T1 (xx)
DK (1) DK1991559T3 (xx)
ES (1) ES2389113T3 (xx)
HK (2) HK1125946A1 (xx)
PL (1) PL1991559T3 (xx)
PT (1) PT1991559E (xx)
SI (1) SI1991559T1 (xx)
WO (1) WO2007098388A2 (xx)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2680119A1 (en) 2007-03-07 2008-09-12 Janssen Pharmaceutica N.V. Steroids derivatives as selective progesterone receptor modulators

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3962275A (en) * 1972-06-05 1976-06-08 Hoffmann-La Roche Inc. 7-oxa steroids
ZA8231B (en) * 1981-01-09 1982-11-24 Roussel Uclaf New 11 -substituted steroid derivatives, their preparation, their use as medicaments, the compositions containing them and the new intermediates thus obtained

Also Published As

Publication number Publication date
EP1991559A2 (en) 2008-11-19
JP2009527494A (ja) 2009-07-30
WO2007098388A3 (en) 2007-12-06
AU2007217101A1 (en) 2007-08-30
US20070197635A1 (en) 2007-08-23
EP1991559B1 (en) 2012-06-27
HK1125946A1 (en) 2009-08-21
CA2642834C (en) 2014-04-15
CN101426806A (zh) 2009-05-06
CN101426806B (zh) 2012-02-01
ES2389113T3 (es) 2012-10-23
WO2007098388A2 (en) 2007-08-30
DK1991559T3 (da) 2012-10-08
US7763648B2 (en) 2010-07-27
CA2642834A1 (en) 2007-08-30
PT1991559E (pt) 2012-09-06
SI1991559T1 (sl) 2012-09-28
PL1991559T3 (pl) 2012-11-30
CY1113127T1 (el) 2016-04-13

Similar Documents

Publication Publication Date Title
IL196533A0 (en) Selective androgen receptor modulators, analogs and derivatives thereof and uses thereof
ZA200807551B (en) Selective androgen receptor modulators
HK1136302A1 (en) Progesterone receptor antagonists
HRP20130374T1 (xx) Derivati pirolidin-2-ona kao modulatori androgenih receptora
ZA200902187B (en) 8-Ethinylxanthine derivatives as selective A2A receptor antagonists
HK1131396A1 (en) 11-phosphorous steroid derivatives useful as progesterone receptor modulators
GB0701992D0 (en) Grehlin Receptor Modulators
ZA200800689B (en) Benzofuranone derivatives as nonsteroidal progesterone receptor modulators
EP2265273A4 (en) HEXAHYDROCYCLOPENTYL [F] INDAZOL-SULFONAMIDES AND THEIR DERIVATIVES AS SELECTIVE GLUCOCORTICOID RECEPTOR MODULATORS
HK1144287A1 (en) Steroids derivatives as selective progesterone receptor modulators
ZA200800690B (en) Non-steroidal progesterone receptor modulators
EP2049104A4 (en) PYRROLIDINONE ANILINES AS MODULATORS OF THE PROGESTERONE RECEPTOR
ZA200806237B (en) Cannibinoid receptor modulators
ATE478078T1 (de) Pyridooxazepin-progesteronrezeptor-modulatoren
HK1131787A1 (en) Oxa-steroids derivatives as selective progesterone receptor modulators
ZA200907546B (en) New progesterone receptor modulators
HK1096405A1 (en) Progesterone receptor modulators
GB0604684D0 (en) Receptor
GB0608516D0 (en) Receptor
GB0623399D0 (en) Receptor
GB0623853D0 (en) Receptor

Legal Events

Date Code Title Description
PC Patent ceased (i.e. patent has lapsed due to the failure to pay the renewal fee)

Effective date: 20160216