GT200700040A - MODIFICATION DIRECTED TO THE FVIII SITE - Google Patents

MODIFICATION DIRECTED TO THE FVIII SITE

Info

Publication number
GT200700040A
GT200700040A GT200700040A GT200700040A GT200700040A GT 200700040 A GT200700040 A GT 200700040A GT 200700040 A GT200700040 A GT 200700040A GT 200700040 A GT200700040 A GT 200700040A GT 200700040 A GT200700040 A GT 200700040A
Authority
GT
Guatemala
Prior art keywords
fviii
site
modification directed
modification
directed
Prior art date
Application number
GT200700040A
Other languages
Spanish (es)
Inventor
Clark Q Pan
John E Murphy
Baisong Mei
Jonathan S Strauss
Hendri Tjandra
Jianmin Chen
Thomas Barnett
Liang Tang
Deqian Wang
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Priority to GT200700040A priority Critical patent/GT200700040A/en
Publication of GT200700040A publication Critical patent/GT200700040A/en

Links

Abstract

LA INVENCIÓN SE RELACIONA CON MUTEÍNAS DEL FACTOR VIII QUE ESTÁN LIGADAS COVALENTEMENTE, EN UN SITIO PREDEFINIDO QUE NO ES UNA AMINA DE TERMINAL N, A UNO O MÁS POLÍMEROS BIOCOMPATIBLES TALES COMO POLIETILENGLICOL. LOS CONJUGADOS DE LA MUTEÍNA RETIENEN LA ACTIVIDAD PROCOAGULANTE DEL FVIII Y TIENEN PROPIEDADES FARMACOCINÉTICAS MEJORADAS. T2007THE INVENTION IS RELATED TO MUTEINS OF FACTOR VIII THAT ARE COVALENTLY LINKED, IN A PRE-DEFINED SITE THAT IS NOT A TERMINAL AMINE N, TO ONE OR MORE BIOCOMPATIBLE POLYMERS SUCH AS POLYETHYLENE. THE MUTEINE CONJUGATES WITHDRAW THE PROVIAGULANT ACTIVITY OF FVIII AND HAVE IMPROVED PHARMACOCINETIC PROPERTIES. T2007

GT200700040A 2007-05-11 2007-05-11 MODIFICATION DIRECTED TO THE FVIII SITE GT200700040A (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
GT200700040A GT200700040A (en) 2007-05-11 2007-05-11 MODIFICATION DIRECTED TO THE FVIII SITE

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GT200700040A GT200700040A (en) 2007-05-11 2007-05-11 MODIFICATION DIRECTED TO THE FVIII SITE

Publications (1)

Publication Number Publication Date
GT200700040A true GT200700040A (en) 2008-12-18

Family

ID=47044086

Family Applications (1)

Application Number Title Priority Date Filing Date
GT200700040A GT200700040A (en) 2007-05-11 2007-05-11 MODIFICATION DIRECTED TO THE FVIII SITE

Country Status (1)

Country Link
GT (1) GT200700040A (en)

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