GT200600302A - Agonistas de ppara/y y procesos de preparación - Google Patents

Agonistas de ppara/y y procesos de preparación

Info

Publication number
GT200600302A
GT200600302A GT200600302A GT200600302A GT200600302A GT 200600302 A GT200600302 A GT 200600302A GT 200600302 A GT200600302 A GT 200600302A GT 200600302 A GT200600302 A GT 200600302A GT 200600302 A GT200600302 A GT 200600302A
Authority
GT
Guatemala
Prior art keywords
agonists
ppara
preparation processes
preparation
phenyl
Prior art date
Application number
GT200600302A
Other languages
English (en)
Inventor
Christine E Garrett
Guang-Pei Chen
George Tien-San Lee
Xinglong Jiang
Michael J Girgis
James Anthony Vivelo
Beata Swerydakrawiec
Dimitris Papoutsakis
Piotr Karpinski
Prasad Koteswara Kapa
Ada Skorodinsky
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of GT200600302A publication Critical patent/GT200600302A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42Oxazoles
    • A61K31/422Oxazoles not condensed and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

Abstract

LA PRESENTE INVENCIÓN PROPORCIONA UN MÉTODO PARA LA PREPARACIÓN DE COMPUESTOS QUE TIENEN LA ESTRUCTURA I, QUE SON AGONISTAS DEL RECEPTOR ACTIVADO POR LOS PROLIFERADORES DE PEROXISOMA (PPAR) ALFA Y GAMMA. DE UNA MANERA MÁS ESPECÍFICA LA INVENCIÓN SE REFIERE A UN NUEVO PROCESO PARA LA PREPARACIÓN DEL ÁCIDO (2R)-2,3-DIHIDRO-1-[[4-[5-METIL-2-[4-(TRIFLUORO-METIL)-FENIL]-4-OXAZOLIL]-METOXI]-FENIL]-SULFONIL]
GT200600302A 2005-07-13 2006-07-10 Agonistas de ppara/y y procesos de preparación GT200600302A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US69880105P 2005-07-13 2005-07-13

Publications (1)

Publication Number Publication Date
GT200600302A true GT200600302A (es) 2007-03-19

Family

ID=37637989

Family Applications (1)

Application Number Title Priority Date Filing Date
GT200600302A GT200600302A (es) 2005-07-13 2006-07-10 Agonistas de ppara/y y procesos de preparación

Country Status (21)

Country Link
US (1) US20080221336A1 (es)
EP (1) EP1912978A2 (es)
JP (1) JP2009501720A (es)
KR (1) KR20080023253A (es)
CN (1) CN101218233A (es)
AR (1) AR054829A1 (es)
AU (1) AU2006267037A1 (es)
BR (1) BRPI0613436A2 (es)
CA (1) CA2615055A1 (es)
EC (1) ECSP088091A (es)
GT (1) GT200600302A (es)
IL (1) IL188479A0 (es)
MA (1) MA29624B1 (es)
MX (1) MX2008000464A (es)
NO (1) NO20080790L (es)
PE (1) PE20070191A1 (es)
RU (1) RU2008104793A (es)
TN (1) TNSN08011A1 (es)
TW (1) TW200800973A (es)
WO (1) WO2007009080A2 (es)
ZA (1) ZA200800102B (es)

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW200303742A (en) * 2001-11-21 2003-09-16 Novartis Ag Organic compounds

Also Published As

Publication number Publication date
JP2009501720A (ja) 2009-01-22
US20080221336A1 (en) 2008-09-11
TW200800973A (en) 2008-01-01
WO2007009080A3 (en) 2007-05-31
RU2008104793A (ru) 2009-08-20
WO2007009080A2 (en) 2007-01-18
TNSN08011A1 (en) 2009-07-14
CA2615055A1 (en) 2007-01-18
KR20080023253A (ko) 2008-03-12
ZA200800102B (en) 2009-02-25
CN101218233A (zh) 2008-07-09
BRPI0613436A2 (pt) 2011-01-11
EP1912978A2 (en) 2008-04-23
PE20070191A1 (es) 2007-03-20
MA29624B1 (fr) 2008-07-01
MX2008000464A (es) 2008-03-11
AR054829A1 (es) 2007-07-18
NO20080790L (no) 2008-02-13
ECSP088091A (es) 2008-02-20
IL188479A0 (en) 2008-04-13
AU2006267037A1 (en) 2007-01-18

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