GEP20196952B - Substituted quinolizine derivatives useful as hiv integrase inhibitors - Google Patents

Substituted quinolizine derivatives useful as hiv integrase inhibitors

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Publication number
GEP20196952B
GEP20196952B GEAP201414124A GEAP2014014124A GEP20196952B GE P20196952 B GEP20196952 B GE P20196952B GE AP201414124 A GEAP201414124 A GE AP201414124A GE AP2014014124 A GEAP2014014124 A GE AP2014014124A GE P20196952 B GEP20196952 B GE P20196952B
Authority
GE
Georgia
Prior art keywords
derivatives useful
hiv integrase
integrase inhibitors
quinolizine derivatives
substituted quinolizine
Prior art date
Application number
GEAP201414124A
Inventor
Sharp & Dohme Corp Merck
Original Assignee
Merck Sharp & Dohme
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Sharp & Dohme filed Critical Merck Sharp & Dohme
Priority to GEAP201414124A priority Critical patent/GEP20196952B/en
Publication of GEP20196952B publication Critical patent/GEP20196952B/en

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Abstract

Compound of formula (I), (I) wherein values of substitutes R1, R2, R3, R4, R5, R9, R10, X, Y are provided in the claims or their pharmaceutically acceptable salt, pharmaceutical composition on a basis thereof, and their usage for prevention or treatment of HIV-infection or AIDS. s Table: 6
GEAP201414124A 2013-09-27 2014-09-26 Substituted quinolizine derivatives useful as hiv integrase inhibitors GEP20196952B (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
GEAP201414124A GEP20196952B (en) 2013-09-27 2014-09-26 Substituted quinolizine derivatives useful as hiv integrase inhibitors

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201361883463P 2013-09-27 2013-09-27
GEAP201414124A GEP20196952B (en) 2013-09-27 2014-09-26 Substituted quinolizine derivatives useful as hiv integrase inhibitors

Publications (1)

Publication Number Publication Date
GEP20196952B true GEP20196952B (en) 2019-03-11

Family

ID=65899479

Family Applications (1)

Application Number Title Priority Date Filing Date
GEAP201414124A GEP20196952B (en) 2013-09-27 2014-09-26 Substituted quinolizine derivatives useful as hiv integrase inhibitors

Country Status (1)

Country Link
GE (1) GEP20196952B (en)

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