GB2058062A - Spectinomycin analogues and their preparation - Google Patents

Spectinomycin analogues and their preparation Download PDF

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Publication number
GB2058062A
GB2058062A GB8027621A GB8027621A GB2058062A GB 2058062 A GB2058062 A GB 2058062A GB 8027621 A GB8027621 A GB 8027621A GB 8027621 A GB8027621 A GB 8027621A GB 2058062 A GB2058062 A GB 2058062A
Authority
GB
United Kingdom
Prior art keywords
compound
formula
alkyl
group
hydrogen
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
GB8027621A
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pharmacia and Upjohn Co
Original Assignee
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Upjohn Co filed Critical Upjohn Co
Publication of GB2058062A publication Critical patent/GB2058062A/en
Withdrawn legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20—Carbocyclic rings
    • C07H15/22—Cyclohexane rings, substituted by nitrogen atoms
    • C07H15/222—Cyclohexane rings substituted by at least two nitrogen atoms
    • C07H15/224—Cyclohexane rings substituted by at least two nitrogen atoms with only one saccharide radical directly attached to the cyclohexyl radical, e.g. destomycin, fortimicin, neamine

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Health & Medical Sciences (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
GB8027621A 1979-08-23 1980-08-26 Spectinomycin analogues and their preparation Withdrawn GB2058062A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/068,926 US4282152A (en) 1979-08-23 1979-08-23 Intermediates for preparing spectinomycin and analogs thereof

Publications (1)

Publication Number Publication Date
GB2058062A true GB2058062A (en) 1981-04-08

Family

ID=22085589

Family Applications (2)

Application Number Title Priority Date Filing Date
GB8027621A Withdrawn GB2058062A (en) 1979-08-23 1980-08-26 Spectinomycin analogues and their preparation
GB8130015A Expired GB2083039B (en) 1979-08-23 1980-08-26 Spectinomycin analogues and their preparation

Family Applications After (1)

Application Number Title Priority Date Filing Date
GB8130015A Expired GB2083039B (en) 1979-08-23 1980-08-26 Spectinomycin analogues and their preparation

Country Status (8)

Country Link
US (1) US4282152A (enExample)
JP (1) JPS5634682A (enExample)
BE (1) BE884889A (enExample)
DE (1) DE3028339A1 (enExample)
FR (2) FR2463772A1 (enExample)
GB (2) GB2058062A (enExample)
IT (1) IT1133042B (enExample)
NL (1) NL8004338A (enExample)

Cited By (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2117757A (en) * 1982-03-19 1983-10-19 Upjohn Co Alkylspectinomycins and their preparation
US4603212A (en) * 1983-10-18 1986-07-29 The Upjohn Company Analogs of the antibiotic spectinomycin
US4698436A (en) * 1982-05-24 1987-10-06 The Upjohn Company Processes for the preparation of spectinomycin analogs, novel products and intermediates therein

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4380652A (en) * 1981-07-20 1983-04-19 The Upjohn Company Enamines of 6'-methylspectinomycin and process for preparing the same
US4380651A (en) * 1981-07-20 1983-04-19 The Upjohn Company Process for preparing 6'-methylspectinomycin and analogs thereof
US4465848A (en) * 1981-10-23 1984-08-14 The Upjohn Company Spectinomycin compounds
JPH0720967B2 (ja) * 1982-03-19 1995-03-08 ザ・アツプジヨン・カンパニ− スペクチノマイシンの６′−アルキル類似体およびその製造方法
US4542227A (en) * 1982-05-24 1985-09-17 The Upjohn Company Processes for the preparation of spectinomycin analogs, novel products and intermediates therein

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3165533A (en) * 1962-01-22 1965-01-12 Upjohn Co Dihydroactinospectacin, amides and esters thereof
US3147277A (en) * 1962-02-09 1964-09-01 Upjohn Co Nu, nu'-bis (alpha-sulfoalkyl) actinospectacins and process for their production
DE2756914A1 (de) * 1977-12-21 1979-07-05 Thomae Gmbh Dr K 4-spectinomycylamin und seine physiologisch vertraegliche salze, verfahren zur herstellung und diese stoffe enthaltende arzneimittel

Cited By (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2117757A (en) * 1982-03-19 1983-10-19 Upjohn Co Alkylspectinomycins and their preparation
US4698436A (en) * 1982-05-24 1987-10-06 The Upjohn Company Processes for the preparation of spectinomycin analogs, novel products and intermediates therein
US4603212A (en) * 1983-10-18 1986-07-29 The Upjohn Company Analogs of the antibiotic spectinomycin

Also Published As

Publication number Publication date
IT8049516A0 (it) 1980-08-18
GB2083039B (en) 1983-06-08
US4282152A (en) 1981-08-04
JPS5634682A (en) 1981-04-06
BE884889A (fr) 1981-02-23
GB2083039A (en) 1982-03-17
DE3028339A1 (de) 1981-04-16
FR2474503A1 (fr) 1981-07-31
FR2463772A1 (fr) 1981-02-27
NL8004338A (nl) 1981-02-25
IT1133042B (it) 1986-07-09
FR2474503B1 (enExample) 1983-12-23
FR2463772B1 (enExample) 1983-12-09

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Legal Events

Date Code Title Description
WAP Application withdrawn, taken to be withdrawn or refused ** after publication under section 16(1)