GB1510073A - 1,3,5-triazapenta-1,4-dienes and their use as acaricides - Google Patents

1,3,5-triazapenta-1,4-dienes and their use as acaricides

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Publication number
GB1510073A
GB1510073A GB15812/76A GB1581276A GB1510073A GB 1510073 A GB1510073 A GB 1510073A GB 15812/76 A GB15812/76 A GB 15812/76A GB 1581276 A GB1581276 A GB 1581276A GB 1510073 A GB1510073 A GB 1510073A
Authority
GB
United Kingdom
Prior art keywords
formula
alkyl
triazapenta
dienes
april
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
GB15812/76A
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Ltd
Original Assignee
Pfizer Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Ltd filed Critical Pfizer Ltd
Priority to GB15812/76A priority Critical patent/GB1510073A/en
Priority to ZA00771561A priority patent/ZA771561B/en
Priority to US05/787,084 priority patent/US4128652A/en
Priority to NZ183875A priority patent/NZ183875A/en
Priority to ES457914A priority patent/ES457914A1/en
Priority to BE176816A priority patent/BE853713A/en
Priority to GR53231A priority patent/GR66426B/el
Priority to NLAANVRAGE7704190,A priority patent/NL170732C/en
Priority to FI771222A priority patent/FI771222A/fi
Priority to IT22627/77A priority patent/IT1074856B/en
Priority to DK172177A priority patent/DK172177A/en
Priority to DE2717280A priority patent/DE2717280C3/en
Priority to IE797/77A priority patent/IE45652B1/en
Priority to BR7702457A priority patent/BR7702457A/en
Priority to CH482477A priority patent/CH604512A5/xx
Priority to LU77155A priority patent/LU77155A1/xx
Priority to FR7711725A priority patent/FR2348920A1/en
Priority to JP4561777A priority patent/JPS52128375A/en
Priority to PL19750677A priority patent/PL197506A1/en
Publication of GB1510073A publication Critical patent/GB1510073A/en
Priority to US05/943,665 priority patent/US4186264A/en
Expired legal-status Critical Current

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
    • C07D333/54—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
    • A—HUMAN NECESSITIES
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    • A01N37/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom having three bonds to hetero atoms with at the most two bonds to halogen, e.g. carboxylic acids
    • A01N37/52—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom having three bonds to hetero atoms with at the most two bonds to halogen, e.g. carboxylic acids containing groups, e.g. carboxylic acid amidines
    • A—HUMAN NECESSITIES
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    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/02—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms
    • A01N43/04—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms with one hetero atom
    • A01N43/06—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms with one hetero atom five-membered rings
    • A01N43/12—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms with one hetero atom five-membered rings condensed with a carbocyclic ring
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    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/34—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom
    • A01N43/40—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
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    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/34—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom
    • A01N43/40—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings
    • A01N43/42—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings condensed with carbocyclic rings
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    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
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    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
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    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/64—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with three nitrogen atoms as the only ring hetero atoms
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    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/74—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,3
    • A01N43/76—1,3-Oxazoles; Hydrogenated 1,3-oxazoles
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/74—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,3
    • A01N43/78—1,3-Thiazoles; Hydrogenated 1,3-thiazoles
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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72—Nitrogen atoms
    • C07D213/74—Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals
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    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32—One oxygen, sulfur or nitrogen atom
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    • C07D277/82—Nitrogen atoms

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  • Chemical & Material Sciences (AREA)
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Abstract

1510073 1,3,5 - triazapenta - 1,4 - dienes PFIZER Ltd 19 April 1977 [20 April 1976 18 Aug 1976] 15812/76 and 34319/76 Heading C2C Novel 1,3,5 - triazapenta - 1,4 - dienes of the general formula wherein R<SP>1</SP> is (C 1 -C 4 ) alkyl; R<SP>2</SP> is hydrogen, halogen, or (C 1 -C 4 ) alkyl; R<SP>3</SP> is an optionally substituted mono- or bicyclic heteroaryl group attached to the nitrogen atom by a carbon atom of said group, and R<SP>4</SP> is hydrogen or (C 1 -C 4 ) alkyl, together with the acid-addition salts thereof are prepared by several methods but preferably either by reacting an amidine of the formula (IV) with an isonitrile of the formula or by reacting formamidine of the the formula with an imidate of the formula wherein R<SP>6</SP> is (C 1 -C 4 ) alkyl. The novel compounds possess acaricidal properties.
GB15812/76A 1976-04-20 1976-04-20 1,3,5-triazapenta-1,4-dienes and their use as acaricides Expired GB1510073A (en)

Priority Applications (20)

Application Number Priority Date Filing Date Title
GB15812/76A GB1510073A (en) 1976-04-20 1976-04-20 1,3,5-triazapenta-1,4-dienes and their use as acaricides
ZA00771561A ZA771561B (en) 1976-04-20 1977-03-15 Acaricidal compounds
US05/787,084 US4128652A (en) 1976-04-20 1977-04-13 Triazapentadienes as acaricides
NZ183875A NZ183875A (en) 1976-04-20 1977-04-15 -(2-alkylphenyl)-3-methyl-5-heter-oaryl-1,3,5-triazapenta-1,4-dienes
ES457914A ES457914A1 (en) 1976-04-20 1977-04-18 Triazapentadienes as acaricides
BE176816A BE853713A (en) 1976-04-20 1977-04-18 NEW TRIAZAPENTADIENES, THEIR PREPARATION PROCESS AND THEIR APPLICATION AS ACARICIDES
GR53231A GR66426B (en) 1976-04-20 1977-04-18
NLAANVRAGE7704190,A NL170732C (en) 1976-04-20 1977-04-18 METHODS FOR PREPARING ACARICIDE COMPOUNDS AND FOR PREPARING PREPARATIONS CONTAINING THEM.
FI771222A FI771222A (en) 1976-04-20 1977-04-18
IT22627/77A IT1074856B (en) 1976-04-20 1977-04-19 TRIAZAPENTADIENI EQUIPPED WITH ACARICIDE PROPERTY
DK172177A DK172177A (en) 1976-04-20 1977-04-19 TRIAZAPENTADIENES PROCEDURE FOR THEIR PREPARATION AND ACARICIDE COMPOSITIONS
DE2717280A DE2717280C3 (en) 1976-04-20 1977-04-19 Triazapentadienes, process for their preparation and their use as anti-mite agents
IE797/77A IE45652B1 (en) 1976-04-20 1977-04-19 1,3,5-triazapenta-1,4-dienes and their use as acaricides
BR7702457A BR7702457A (en) 1976-04-20 1977-04-19 PROCESS FOR THE PREPARATION OF TRI-AZA-PENTA-DIENOS; AND PROCESS FOR THE PROTECTION OF IRRATIONAL ANIMALS, ESPECIALLY CATTLE, AGAINST ACARIDEOS, ESPECIALLY CATTLE TICKS
CH482477A CH604512A5 (en) 1976-04-20 1977-04-19
LU77155A LU77155A1 (en) 1976-04-20 1977-04-19
FR7711725A FR2348920A1 (en) 1976-04-20 1977-04-19 NEW TRIAZAPENTADIENES, THEIR PREPARATION PROCESS AND THEIR APPLICATION AS ACARICIDES
JP4561777A JPS52128375A (en) 1976-04-20 1977-04-20 Acaricidal compound and preparation thereof
PL19750677A PL197506A1 (en) 1976-04-20 1977-04-20 METHOD OF MAKING HETEROARYL TRIAZAPENTADIENES
US05/943,665 US4186264A (en) 1976-04-20 1978-09-18 Triazapentadienes as acaricides

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB15812/76A GB1510073A (en) 1976-04-20 1976-04-20 1,3,5-triazapenta-1,4-dienes and their use as acaricides

Publications (1)

Publication Number Publication Date
GB1510073A true GB1510073A (en) 1978-05-10

Family

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Family Applications (1)

Application Number Title Priority Date Filing Date
GB15812/76A Expired GB1510073A (en) 1976-04-20 1976-04-20 1,3,5-triazapenta-1,4-dienes and their use as acaricides

Country Status (3)

Country Link
BE (1) BE853713A (en)
GB (1) GB1510073A (en)
ZA (1) ZA771561B (en)

Also Published As

Publication number Publication date
BE853713A (en) 1977-10-18
ZA771561B (en) 1978-01-25

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