GB1393993A - Agent for the regulation of plant growth - Google Patents
Agent for the regulation of plant growthInfo
- Publication number
- GB1393993A GB1393993A GB2297372A GB2297372A GB1393993A GB 1393993 A GB1393993 A GB 1393993A GB 2297372 A GB2297372 A GB 2297372A GB 2297372 A GB2297372 A GB 2297372A GB 1393993 A GB1393993 A GB 1393993A
- Authority
- GB
- United Kingdom
- Prior art keywords
- alkyl
- hnr
- novel
- optionally substituted
- stated
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/32—One oxygen, sulfur or nitrogen atom
- C07D239/42—One nitrogen atom
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
- A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/32—One oxygen, sulfur or nitrogen atom
- C07D239/38—One sulfur atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/48—Two nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/50—Three nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/60—Three or more oxygen or sulfur atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Agronomy & Crop Science (AREA)
- Pest Control & Pesticides (AREA)
- Plant Pathology (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Dentistry (AREA)
- General Health & Medical Sciences (AREA)
- Wood Science & Technology (AREA)
- Zoology (AREA)
- Environmental Sciences (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
1393993 Pyrimidines CIBA-GEIGY AG 16 May 1972 [17 May 1971] 22973/72 Heading C2C Novel 5-nitropyrimidines of Formula I wherein R 1 represents C 2-6 alkyl, C 3-5 alkenyl, C 3-5 alkinyl, C 1-4 hydroxyalkyl, C 2-5 cyanoalkyl, or alkoxyalkyl or alkylamino alkyl or trialkylammonioalkyl wherein each alkyl moiety has 1-6 C atoms, or C 3-6 cycloalkyl optionally substituted by Me or Et; R 2 and R 3 which may be identical or different each represent H or C 1-6 alkyl; R 4 represents H, C 1-6 alkyl or C 3-6 cycloalkyl optionally substituted by Me or Et; R 5 represents C 1-6 alkyl; or R 1 and R 2 taken together form a C 2-6 polymethylene group, or R 3 and R 4 taken together form a C 4-6 polymethylene group, each of which may have a methylene group replaced by O or NR<SP>1</SP> where R<SP>1</SP> represents H or C 1-6 alkyl; and acid addition salts thereof with an inorganic or organic strong acid or quaternary salts thereof, may be prepared by exchanging the halogen atoms of a dihalopyrimidine of Formula IV successively with amines of formulµ HNR 1 R 2 and HNR 3 R 4 at a temperature between -60 C. and +120 C. in the presence of a base. Certain of the intermediate pyrimidines which may be isolated after the first step of the process, i.e. those containing a single halogen atom, are stated to be novel and these and the other novel compounds I of the invention exhibit plant growth regulant properties. An alternative preparative route for the compounds I is from the 2,4,6-trihalo-5-nitropyrimidine by reaction with HNR 1 R 2 and HNR 3 R 4 to give an intermediate (some of which are stated to be novel) which may be reacted with HSR 5 or an alkali metal salt thereof.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
CH722971A CH558137A (en) | 1971-05-17 | 1971-05-17 | MEANS OF INFLUENCING PLANT GROWTH. |
Publications (1)
Publication Number | Publication Date |
---|---|
GB1393993A true GB1393993A (en) | 1975-05-14 |
Family
ID=4321885
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
GB2297372A Expired GB1393993A (en) | 1971-05-17 | 1972-05-16 | Agent for the regulation of plant growth |
Country Status (18)
Country | Link |
---|---|
JP (1) | JPS5654283B1 (en) |
BG (1) | BG19073A3 (en) |
BR (1) | BR7203098D0 (en) |
CA (1) | CA994773A (en) |
CH (1) | CH558137A (en) |
CS (1) | CS177082B2 (en) |
DE (1) | DE2223644A1 (en) |
EG (1) | EG10574A (en) |
ES (1) | ES402755A1 (en) |
FR (1) | FR2137933B1 (en) |
GB (1) | GB1393993A (en) |
HU (1) | HU164885B (en) |
IL (1) | IL39417A (en) |
IT (1) | IT955556B (en) |
NL (1) | NL7206602A (en) |
SU (1) | SU578825A3 (en) |
TR (1) | TR17050A (en) |
ZA (1) | ZA723325B (en) |
Cited By (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO1991001310A1 (en) * | 1989-07-21 | 1991-02-07 | Beecham Group Plc | Process for preparing 2,5-diamino-4,6-dichloropyrimidine |
US7812159B2 (en) | 2005-01-10 | 2010-10-12 | Arena Pharamaceuticals, Inc. | Processes for preparing aromatic ethers |
US7838525B2 (en) | 2003-07-11 | 2010-11-23 | Arena Pharmaceuticals, Inc. | Trisubstituted aryl and heteroaryl derivatives as modulators of metabolism and the prophylaxis and treatment of disorders related thereto |
US8933083B2 (en) | 2003-01-14 | 2015-01-13 | Arena Pharmaceuticals, Inc. | 1,2,3-trisubstituted aryl and heteroaryl derivatives as modulators of metabolism and the prophylaxis and treatment of disorders related thereto such as diabetes and hyperglycemia |
US10894787B2 (en) | 2010-09-22 | 2021-01-19 | Arena Pharmaceuticals, Inc. | Modulators of the GPR119 receptor and the treatment of disorders related thereto |
US11007175B2 (en) | 2015-01-06 | 2021-05-18 | Arena Pharmaceuticals, Inc. | Methods of treating conditions related to the S1P1 receptor |
US11884626B2 (en) | 2015-06-22 | 2024-01-30 | Arena Pharmaceuticals, Inc. | Crystalline L-arginine salt of (R)-2-(7-(4-cyclopentyl-3-(trifluoromethyl)benzyloxy)-1,2,3,4-tetrahydrocyclo-penta [b]indol-3-yl)acetic acid(Compound1) for use in S1P1 receptor-associated disorders |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CH595061A5 (en) * | 1974-05-10 | 1978-01-31 | Ciba Geigy Ag | |
TWI229674B (en) | 1998-12-04 | 2005-03-21 | Astra Pharma Prod | Novel triazolo[4,5-d]pyrimidine compounds, pharmaceutical composition containing the same, their process for preparation and uses |
MY148521A (en) | 2005-01-10 | 2013-04-30 | Arena Pharm Inc | Substituted pyridinyl and pyrimidinyl derivatives as modulators of metabolism and the treatment of disorders related thereto |
GB0512844D0 (en) * | 2005-06-23 | 2005-08-03 | Novartis Ag | Organic compounds |
CN110520124A (en) | 2017-02-16 | 2019-11-29 | 艾尼纳制药公司 | For treating the Compounds and methods for of primary biliary cholangitis |
-
1971
- 1971-05-17 CH CH722971A patent/CH558137A/en not_active IP Right Cessation
-
1972
- 1972-05-11 IL IL39417A patent/IL39417A/en unknown
- 1972-05-13 EG EG200/72*UA patent/EG10574A/en active
- 1972-05-15 DE DE19722223644 patent/DE2223644A1/en not_active Ceased
- 1972-05-16 NL NL7206602A patent/NL7206602A/xx not_active Application Discontinuation
- 1972-05-16 ZA ZA723325A patent/ZA723325B/en unknown
- 1972-05-16 CS CS3315A patent/CS177082B2/cs unknown
- 1972-05-16 BG BG020491A patent/BG19073A3/en unknown
- 1972-05-16 BR BR3098/72A patent/BR7203098D0/en unknown
- 1972-05-16 IT IT24402/72A patent/IT955556B/en active
- 1972-05-16 GB GB2297372A patent/GB1393993A/en not_active Expired
- 1972-05-16 ES ES402755A patent/ES402755A1/en not_active Expired
- 1972-05-16 SU SU7201785752A patent/SU578825A3/en active
- 1972-05-16 FR FR727217420A patent/FR2137933B1/fr not_active Expired
- 1972-05-16 TR TR17050A patent/TR17050A/en unknown
- 1972-05-16 HU HUCI1238A patent/HU164885B/hu unknown
- 1972-05-17 CA CA142,388A patent/CA994773A/en not_active Expired
- 1972-05-17 JP JP4949172A patent/JPS5654283B1/ja active Pending
Cited By (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO1991001310A1 (en) * | 1989-07-21 | 1991-02-07 | Beecham Group Plc | Process for preparing 2,5-diamino-4,6-dichloropyrimidine |
AU634564B2 (en) * | 1989-07-21 | 1993-02-25 | Beecham Group Plc | Process for preparing 2,5-diamino-4,6-dichloropyrimidine |
US8933083B2 (en) | 2003-01-14 | 2015-01-13 | Arena Pharmaceuticals, Inc. | 1,2,3-trisubstituted aryl and heteroaryl derivatives as modulators of metabolism and the prophylaxis and treatment of disorders related thereto such as diabetes and hyperglycemia |
US7838525B2 (en) | 2003-07-11 | 2010-11-23 | Arena Pharmaceuticals, Inc. | Trisubstituted aryl and heteroaryl derivatives as modulators of metabolism and the prophylaxis and treatment of disorders related thereto |
US8546429B2 (en) | 2003-07-11 | 2013-10-01 | Arena Pharmaceuticals, Inc. | 1,2,3-trisubstituted aryl and heteroaryl derivatives as modulators of metabolism and the prophylaxis and treatment of disorders related thereto |
US7812159B2 (en) | 2005-01-10 | 2010-10-12 | Arena Pharamaceuticals, Inc. | Processes for preparing aromatic ethers |
US10894787B2 (en) | 2010-09-22 | 2021-01-19 | Arena Pharmaceuticals, Inc. | Modulators of the GPR119 receptor and the treatment of disorders related thereto |
US11007175B2 (en) | 2015-01-06 | 2021-05-18 | Arena Pharmaceuticals, Inc. | Methods of treating conditions related to the S1P1 receptor |
US11884626B2 (en) | 2015-06-22 | 2024-01-30 | Arena Pharmaceuticals, Inc. | Crystalline L-arginine salt of (R)-2-(7-(4-cyclopentyl-3-(trifluoromethyl)benzyloxy)-1,2,3,4-tetrahydrocyclo-penta [b]indol-3-yl)acetic acid(Compound1) for use in S1P1 receptor-associated disorders |
Also Published As
Publication number | Publication date |
---|---|
BR7203098D0 (en) | 1973-05-31 |
FR2137933B1 (en) | 1973-07-13 |
IT955556B (en) | 1973-09-29 |
IL39417A (en) | 1975-07-28 |
SU578825A3 (en) | 1977-10-30 |
FR2137933A1 (en) | 1972-12-29 |
ZA723325B (en) | 1973-02-28 |
CS177082B2 (en) | 1977-07-29 |
NL7206602A (en) | 1972-11-21 |
TR17050A (en) | 1974-04-25 |
HU164885B (en) | 1974-05-28 |
JPS5654283B1 (en) | 1981-12-24 |
BG19073A3 (en) | 1975-04-30 |
EG10574A (en) | 1976-01-31 |
DE2223644A1 (en) | 1972-11-30 |
ES402755A1 (en) | 1975-04-01 |
IL39417A0 (en) | 1972-07-26 |
CA994773A (en) | 1976-08-10 |
CH558137A (en) | 1975-01-31 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
PS | Patent sealed [section 19, patents act 1949] | ||
PCNP | Patent ceased through non-payment of renewal fee |