GB1393675A - Alkanolamine derivatives - Google Patents
Alkanolamine derivativesInfo
- Publication number
- GB1393675A GB1393675A GB2820571A GB2820571A GB1393675A GB 1393675 A GB1393675 A GB 1393675A GB 2820571 A GB2820571 A GB 2820571A GB 2820571 A GB2820571 A GB 2820571A GB 1393675 A GB1393675 A GB 1393675A
- Authority
- GB
- United Kingdom
- Prior art keywords
- alkyl
- alkenyl
- emulsions
- halogen
- agents
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C275/00—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups
- C07C275/28—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
- C07C275/32—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton being further substituted by singly-bound oxygen atoms
- C07C275/34—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton being further substituted by singly-bound oxygen atoms having nitrogen atoms of urea groups and singly-bound oxygen atoms bound to carbon atoms of the same non-condensed six-membered aromatic ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
- C07C323/23—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton
- C07C323/39—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton at least one of the nitrogen atoms being part of any of the groups, X being a hetero atom, Y being any atom
- C07C323/43—Y being a hetero atom
- C07C323/44—X or Y being nitrogen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Abstract
1393675 #-adrenergic blocking medicines IMPERIAL CHEMICAL INDUSTRIES Ltd 26 May 1972 [16 June 1971] 28205/71 Heading ASB [Also in Division C2] Pharmaceutical compositions, in the form of tablets, capsules, orally-acceptable solutions, suspensions or emulsions, injectable solutions, suspension or emulsions, dispersible powders, sprays or aerosols, contain novel alkanolamines or pharmaceutically acceptable acid addition salts thereof of the formula: wherein R<SP>1</SP> is C 3-5 alkyl or C 3-5 hydroxyalkyl which are branched at the alphacarbon atom or C 3-5 cycloalkyl; R<SP>2</SP> is C 1-10 alkyl or C 2-6 alkenyl; and R<SP>3</SP> is H, halogen, OH, CN, C 1-6 alkyl, C 1-6 alkoxy, C 1-6 alkylthio, C 2-6 alkenyl, C 2-6 alkonyloxy or C 7-10 aralkyl; provided that when R<SP>3</SP> is H, halogen or C 1-6 alkyl, R<SP>2</SP> is C 2-6 alkenyl, in association with pharmaceutically acceptable diluents or carriers. The compositions may also contain other active ingredients selected from sedatives, for example phonobarbitone, moprobate, chlorpromazine or a benzodiazepine, vasodilators, for example glyceryl trinitrate, pentaerythritol tetranitrate or isosorbide dinitrate, diuretics, for example chlorothiazide, hypotensive agents, for example reserpine, bethanidine or quanethidine, myocardial depressants, for example quinidine, agents used in the treatment of Parkinson's disease, for example benzhexol, cardiotonic agents, for example digitalis preparations, or sympathomimetic bronchodilators, for example isoprenaline, orciprenaline, adrenaline or ephedrine. The compounds possess #-adrenergic blocking activity.
Priority Applications (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB2820571A GB1393675A (en) | 1971-06-16 | 1971-06-16 | Alkanolamine derivatives |
DE19722229241 DE2229241A1 (en) | 1971-06-16 | 1972-06-15 | Alkanolamide derivatives |
FR7221650A FR2141978B1 (en) | 1971-06-16 | 1972-06-15 | |
CH901172A CH570358A5 (en) | 1971-06-16 | 1972-06-16 |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB2820571A GB1393675A (en) | 1971-06-16 | 1971-06-16 | Alkanolamine derivatives |
Publications (1)
Publication Number | Publication Date |
---|---|
GB1393675A true GB1393675A (en) | 1975-05-07 |
Family
ID=10271980
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
GB2820571A Expired GB1393675A (en) | 1971-06-16 | 1971-06-16 | Alkanolamine derivatives |
Country Status (4)
Country | Link |
---|---|
CH (1) | CH570358A5 (en) |
DE (1) | DE2229241A1 (en) |
FR (1) | FR2141978B1 (en) |
GB (1) | GB1393675A (en) |
Cited By (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4038313A (en) | 1970-01-08 | 1977-07-26 | Ciba-Geigy Corporation | Cycloalkylureido phenoxy propanolamines |
US4145363A (en) * | 1975-02-05 | 1979-03-20 | Yamanouchi Pharmaceutical Co., Ltd. | 4-Carbamoylamino-α-aminomethylbenzyl alcohol derivatives |
-
1971
- 1971-06-16 GB GB2820571A patent/GB1393675A/en not_active Expired
-
1972
- 1972-06-15 DE DE19722229241 patent/DE2229241A1/en active Pending
- 1972-06-15 FR FR7221650A patent/FR2141978B1/fr not_active Expired
- 1972-06-16 CH CH901172A patent/CH570358A5/xx not_active IP Right Cessation
Cited By (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4038313A (en) | 1970-01-08 | 1977-07-26 | Ciba-Geigy Corporation | Cycloalkylureido phenoxy propanolamines |
US4145363A (en) * | 1975-02-05 | 1979-03-20 | Yamanouchi Pharmaceutical Co., Ltd. | 4-Carbamoylamino-α-aminomethylbenzyl alcohol derivatives |
Also Published As
Publication number | Publication date |
---|---|
CH570358A5 (en) | 1975-12-15 |
DE2229241A1 (en) | 1972-12-21 |
FR2141978B1 (en) | 1976-04-16 |
FR2141978A1 (en) | 1973-01-26 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
GB1199037A (en) | Alkanolamine Derivatives | |
GB1455116A (en) | Pharmaceutical compositions | |
IE39306B1 (en) | Ethanolamine derivatives | |
US3671625A (en) | Compositions for treating asthma comprising bis-chromonyl compounds and method of employing same | |
GB1285038A (en) | Alkanolamine derivatives | |
GB1199632A (en) | Alkanolamine Derivatives | |
GB1269775A (en) | Alkanolamine derivatives | |
HUT60507A (en) | Process for producing trifluoromethyl ketone derivatives and pharmaceutical compositions comprising same as active ingredient | |
ATE48001T1 (en) | CEPHEM COMPOUNDS, PROCESSES FOR THEIR PRODUCTION AND THEIR PHARMACEUTICAL PREPARATIONS. | |
ES8203382A1 (en) | Indolobenzoxazines, processes for preparing and pharmaceutical compositions containing the same. | |
ES8605760A1 (en) | (Omega-(diethylamino)-alkoxy)-alpha-(ethyl)-benzhydrol derivatives, their acid addition salts and quaternary salts, process for their preparation and medicines containing these compounds. | |
GB1393675A (en) | Alkanolamine derivatives | |
IE852823L (en) | Medicaments containing spergualin | |
GB1460071A (en) | Tetrahydronaphthyloxy-amines and related compounds | |
GB1396322A (en) | Alkanolamine derivatives | |
GB1387630A (en) | Phenoxyalkanolamine derivatives | |
GB1269781A (en) | Alkanolamine derivatives | |
GB1415505A (en) | Alkanolamine derivatives | |
GB1312555A (en) | Alkanolamine derivatives | |
MY106235A (en) | New 2 - carbonyl substituted n, n'' -di (trimethoxybenzoyl) piperazines, process for preparing the same and therapeutical compounds containing them. | |
GB1312055A (en) | Alkanolamine derivatives | |
GB1392610A (en) | Alkanolamine derivatives | |
GB1414781A (en) | Alkanolamine derivatives | |
GB1481948A (en) | 2-(disubstituted-amino)-4-phenyl-imidazolines and their use in pharmaceutical compositions | |
KR890009919A (en) | 4-heteroaryl-1,3-benzodiazepine and 2-substituted-α- (heteroaryl) benzeneethanamine, methods of preparation and use thereof as medicaments |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
PS | Patent sealed |