FR2943674B1 - AZACARBOLINE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC USE - Google Patents

AZACARBOLINE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC USE

Info

Publication number
FR2943674B1
FR2943674B1 FR0901368A FR0901368A FR2943674B1 FR 2943674 B1 FR2943674 B1 FR 2943674B1 FR 0901368 A FR0901368 A FR 0901368A FR 0901368 A FR0901368 A FR 0901368A FR 2943674 B1 FR2943674 B1 FR 2943674B1
Authority
FR
France
Prior art keywords
preparation
therapeutic use
azacarboline
derivatives
azacarboline derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
FR0901368A
Other languages
French (fr)
Other versions
FR2943674A1 (en
Inventor
Didier Babin
Olivier Bedel
Thierry Gouyon
Serge Mignani
David Papin
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sanofi Aventis France
Original Assignee
Sanofi Aventis France
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority to FR0901368A priority Critical patent/FR2943674B1/en
Application filed by Sanofi Aventis France filed Critical Sanofi Aventis France
Priority to TW098140843A priority patent/TW201035097A/en
Priority to BRPI0924844A priority patent/BRPI0924844A2/en
Priority to PCT/FR2009/052330 priority patent/WO2010109084A2/en
Priority to UY0001032275A priority patent/UY32275A/en
Priority to CA2756152A priority patent/CA2756152A1/en
Priority to EP09797115A priority patent/EP2411389A2/en
Priority to CN2009801583033A priority patent/CN102365282A/en
Priority to US13/258,924 priority patent/US20120208809A1/en
Priority to RU2011142791/04A priority patent/RU2011142791A/en
Priority to AU2009342734A priority patent/AU2009342734A1/en
Priority to JP2012501334A priority patent/JP2012521394A/en
Priority to ARP090104599A priority patent/AR073431A1/en
Priority to KR1020117024857A priority patent/KR20110130504A/en
Priority to SG2011068889A priority patent/SG174903A1/en
Priority to MX2011010062A priority patent/MX2011010062A/en
Publication of FR2943674A1 publication Critical patent/FR2943674A1/en
Priority to IL215286A priority patent/IL215286A0/en
Application granted granted Critical
Publication of FR2943674B1 publication Critical patent/FR2943674B1/en
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/14—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
FR0901368A 2009-03-24 2009-03-24 AZACARBOLINE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC USE Expired - Fee Related FR2943674B1 (en)

Priority Applications (17)

Application Number Priority Date Filing Date Title
FR0901368A FR2943674B1 (en) 2009-03-24 2009-03-24 AZACARBOLINE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC USE
ARP090104599A AR073431A1 (en) 2009-03-24 2009-11-30 DERIVATIVES OF AZACARBOLINAS 9H- PIRROLO (2,3-B: 5,4-C) DIPIRIDINE, ITS PREPARATION AND IF THERAPEUTIC USE
PCT/FR2009/052330 WO2010109084A2 (en) 2009-03-24 2009-11-30 9h-pyrrolo[2,3-b: 5,4-c'] dipyridine azacarboline derivatives, preparation thereof, and therapeutic use thereof
UY0001032275A UY32275A (en) 2009-03-24 2009-11-30 DERIVATIVES OF AZACARBOLINAS 9H-PIRROLO [2,3-b: 5,4-c '] DIPIRIDINE, ITS PREPARATION AND ITS THERAPEUTIC USE.
CA2756152A CA2756152A1 (en) 2009-03-24 2009-11-30 9h-pyrrolo[2,3-b: 5,4-c'] dipyridine azacarboline derivatives, preparation thereof, and therapeutic use thereof
EP09797115A EP2411389A2 (en) 2009-03-24 2009-11-30 9h-pyrrolo[2,3-b: 5,4-c']dipyridine azacarboline derivatives, preparation thereof, and therapeutic use thereof
CN2009801583033A CN102365282A (en) 2009-03-24 2009-11-30 9H-pyrrolo[2,3-B: 5,4-C'] dipyridine azacarboline derivatives, preparation thereof, and therapeutic use thereof
US13/258,924 US20120208809A1 (en) 2009-03-24 2009-11-30 9h-pyrrolo[2,3-b: 5,4-c'] dipyridine azacarboline derivatives, preparation thereof, and therapeutic use thereof
TW098140843A TW201035097A (en) 2009-03-24 2009-11-30 9H-pyrrolo[2,3-b:5,4-c']dipyridine azacarboline derivatives, preparation and therapeutic use thereof
AU2009342734A AU2009342734A1 (en) 2009-03-24 2009-11-30 9H-pyrrolo[2,3-b: 5,4-c'] dipyridine azacarboline derivatives, preparation thereof, and therapeutic use thereof
JP2012501334A JP2012521394A (en) 2009-03-24 2009-11-30 9H-pyrrolo [2,3-B: 5,4-C '] dipyridine azacarboline derivative, its preparation and its therapeutic use
BRPI0924844A BRPI0924844A2 (en) 2009-03-24 2009-11-30 azacarbolines derivatives 9h-pyrrol [2,3-b: 5,4-c '] dipyridine, their preparation and their therapeutic use.
KR1020117024857A KR20110130504A (en) 2009-03-24 2009-11-30 9h-pyrrolo[2,3-b:5,4-c']dipyridine azacarboline derivatives, preparation thereof, and therapeutic use thereof
SG2011068889A SG174903A1 (en) 2009-03-24 2009-11-30 9h-pyrrolo[2,3-b: 5,4-c'] dipyridine azacarboline derivatives, preparation thereof, and therapeutic use thereof
MX2011010062A MX2011010062A (en) 2009-03-24 2009-11-30 9h-pyrrolo[2,3-b: 5,4-c'] dipyridine azacarboline derivatives, preparation thereof, and therapeutic use thereof.
RU2011142791/04A RU2011142791A (en) 2009-03-24 2009-11-30 9H-PYRROLO DERIVATIVES [2,3-B: 5,4-C ′] DIPYRIDINE-AZACARBOLINES, METHOD FOR PRODUCING THEM AND USE IN THERAPY
IL215286A IL215286A0 (en) 2009-03-24 2011-09-21 9h-pyrrolo[2,3-b:5,4-c]dipridine azacarboline derivatives, preparation thereof, and therapeutic use thereof

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0901368A FR2943674B1 (en) 2009-03-24 2009-03-24 AZACARBOLINE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC USE

Publications (2)

Publication Number Publication Date
FR2943674A1 FR2943674A1 (en) 2010-10-01
FR2943674B1 true FR2943674B1 (en) 2013-02-22

Family

ID=41087376

Family Applications (1)

Application Number Title Priority Date Filing Date
FR0901368A Expired - Fee Related FR2943674B1 (en) 2009-03-24 2009-03-24 AZACARBOLINE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC USE

Country Status (1)

Country Link
FR (1) FR2943674B1 (en)

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1209158A1 (en) * 2000-11-18 2002-05-29 Aventis Pharma Deutschland GmbH Substituted beta-carbolines
EP1134221A1 (en) * 2000-03-15 2001-09-19 Aventis Pharma Deutschland GmbH Substituted beta-carbolines as lkB kinase inhibitors
WO2006131552A1 (en) * 2005-06-09 2006-12-14 Boehringer Ingelheim International Gmbh Alpha-carbolines as cdk-1 inhibitors
US8119655B2 (en) * 2005-10-07 2012-02-21 Takeda Pharmaceutical Company Limited Kinase inhibitors

Also Published As

Publication number Publication date
FR2943674A1 (en) 2010-10-01

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Legal Events

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Effective date: 20141128