FR2882931B1 - Compositions pharmaceutiques contenant en association un compose antagoniste des recepteurs aux cannabinoidess et un agent antipsychotique - Google Patents

Compositions pharmaceutiques contenant en association un compose antagoniste des recepteurs aux cannabinoidess et un agent antipsychotique

Info

Publication number
FR2882931B1
FR2882931B1 FR0502508A FR0502508A FR2882931B1 FR 2882931 B1 FR2882931 B1 FR 2882931B1 FR 0502508 A FR0502508 A FR 0502508A FR 0502508 A FR0502508 A FR 0502508A FR 2882931 B1 FR2882931 B1 FR 2882931B1
Authority
FR
France
Prior art keywords
cannabinoidess
receptors
association
pharmaceutical compositions
compositions containing
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
FR0502508A
Other languages
English (en)
Other versions
FR2882931A1 (fr
Inventor
Michele Arnone
Trillou Christine Ravinet
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sanofi Aventis France
Original Assignee
Sanofi Aventis France
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority to FR0502508A priority Critical patent/FR2882931B1/fr
Application filed by Sanofi Aventis France filed Critical Sanofi Aventis France
Priority to BRPI0608438-9A priority patent/BRPI0608438A2/pt
Priority to EP06726063A priority patent/EP1863489A1/fr
Priority to MX2007011357A priority patent/MX2007011357A/es
Priority to KR1020077023434A priority patent/KR20070112266A/ko
Priority to AU2006224446A priority patent/AU2006224446A1/en
Priority to RU2007138042/15A priority patent/RU2007138042A/ru
Priority to CNA2006800081089A priority patent/CN101137373A/zh
Priority to JP2008501356A priority patent/JP2008533110A/ja
Priority to CA002600028A priority patent/CA2600028A1/fr
Priority to PCT/FR2006/000532 priority patent/WO2006097605A1/fr
Publication of FR2882931A1 publication Critical patent/FR2882931A1/fr
Application granted granted Critical
Publication of FR2882931B1 publication Critical patent/FR2882931B1/fr
Priority to IL185789A priority patent/IL185789A0/en
Priority to US11/854,032 priority patent/US20080015186A1/en
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • A61K31/4523Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/454Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/551Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/551Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
    • A61K31/55131,4-Benzodiazepines, e.g. diazepam or clozapine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Psychiatry (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
FR0502508A 2005-03-14 2005-03-14 Compositions pharmaceutiques contenant en association un compose antagoniste des recepteurs aux cannabinoidess et un agent antipsychotique Expired - Fee Related FR2882931B1 (fr)

Priority Applications (13)

Application Number Priority Date Filing Date Title
FR0502508A FR2882931B1 (fr) 2005-03-14 2005-03-14 Compositions pharmaceutiques contenant en association un compose antagoniste des recepteurs aux cannabinoidess et un agent antipsychotique
PCT/FR2006/000532 WO2006097605A1 (fr) 2005-03-14 2006-03-10 Compositions pharmaceutiques contenant en association un compose antagoniste des recepteurs aux cannabinoides et un agent antipsychotique
MX2007011357A MX2007011357A (es) 2005-03-14 2006-03-10 Composiciones farmaceuticas que contienen en asociacion un compuesto antagonista de los receptores de cannabinoides y un agente antipsicotico.
KR1020077023434A KR20070112266A (ko) 2005-03-14 2006-03-10 칸나비노이드 수용체 길항제 화합물과 항정신병제의조합물을 함유하는 제약 조성물
AU2006224446A AU2006224446A1 (en) 2005-03-14 2006-03-10 Pharmaceutical compositions containing a combination of a cannabinoid receptor antagonist compound and an antipsychotic agent
RU2007138042/15A RU2007138042A (ru) 2005-03-14 2006-03-10 Фармацевтические композиции, содержащие в сочетании соединение-антагонист рецепторов каннабиноидов и нейролептическое средство
BRPI0608438-9A BRPI0608438A2 (pt) 2005-03-14 2006-03-10 composições farmacêuticas contendo em associação um composto antagonista dos receptores aos canabinóides e um agente antipsicótico
JP2008501356A JP2008533110A (ja) 2005-03-14 2006-03-10 カンナビノイド受容体アンタゴニスト化合物および抗精神病薬剤の組合せを含有する医薬組成物
CA002600028A CA2600028A1 (fr) 2005-03-14 2006-03-10 Compositions pharmaceutiques contenant en association un compose antagoniste des recepteurs aux cannabinoides et un agent antipsychotique
EP06726063A EP1863489A1 (fr) 2005-03-14 2006-03-10 Compositions pharmaceutiques contenant en association un compose antagoniste des recepteurs aux cannabinoides et un agent antipsychotique
CNA2006800081089A CN101137373A (zh) 2005-03-14 2006-03-10 含有大麻素受体拮抗化合物与防治精神病剂组合的药物组合物
IL185789A IL185789A0 (en) 2005-03-14 2007-09-06 Pharmaceutical compositions containing a combination of a cannabinoid receptor antagonist compound and an antipsychotic agent
US11/854,032 US20080015186A1 (en) 2005-03-14 2007-09-12 Pharmaceutical compositions containing in combination a cannabinoid receptor antagonist and an antipsychotic

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0502508A FR2882931B1 (fr) 2005-03-14 2005-03-14 Compositions pharmaceutiques contenant en association un compose antagoniste des recepteurs aux cannabinoidess et un agent antipsychotique

Publications (2)

Publication Number Publication Date
FR2882931A1 FR2882931A1 (fr) 2006-09-15
FR2882931B1 true FR2882931B1 (fr) 2007-05-18

Family

ID=34955355

Family Applications (1)

Application Number Title Priority Date Filing Date
FR0502508A Expired - Fee Related FR2882931B1 (fr) 2005-03-14 2005-03-14 Compositions pharmaceutiques contenant en association un compose antagoniste des recepteurs aux cannabinoidess et un agent antipsychotique

Country Status (13)

Country Link
US (1) US20080015186A1 (fr)
EP (1) EP1863489A1 (fr)
JP (1) JP2008533110A (fr)
KR (1) KR20070112266A (fr)
CN (1) CN101137373A (fr)
AU (1) AU2006224446A1 (fr)
BR (1) BRPI0608438A2 (fr)
CA (1) CA2600028A1 (fr)
FR (1) FR2882931B1 (fr)
IL (1) IL185789A0 (fr)
MX (1) MX2007011357A (fr)
RU (1) RU2007138042A (fr)
WO (1) WO2006097605A1 (fr)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PE20071092A1 (es) * 2005-12-08 2007-12-10 Aventis Pharma Inc Composicion farmaceutica que comprende un antagonista de cb1 y un agente antisicotico
ES2330071B1 (es) * 2007-01-15 2010-07-05 Laboratorios Del Dr. Esteve, S.A. Combinacion de sustancias activas.
EP1946777A1 (fr) * 2007-01-16 2008-07-23 Laboratorios del Dr. Esteve S.A. Composés de pyrazoline substituée pour éviter la prise de poids
GB2456183A (en) 2008-01-04 2009-07-08 Gw Pharma Ltd Anti-psychotic composition comprising cannabinoids and anti-psychotic medicament
US8566459B2 (en) 2009-05-29 2013-10-22 Red Hat, Inc. Systems and methods for integrated console management interface

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2692575B1 (fr) * 1992-06-23 1995-06-30 Sanofi Elf Nouveaux derives du pyrazole, procede pour leur preparation et compositions pharmaceutiques les contenant.
FR2789079B3 (fr) * 1999-02-01 2001-03-02 Sanofi Synthelabo Derive d'acide pyrazolecarboxylique, sa preparation, les compositions pharmaceutiques en contenant
CA2537535A1 (fr) * 2003-09-02 2005-03-10 Solvay Pharmaceuticals Gmbh Nouvelles utilisations medicales d'antagonistes selectifs du recepteur cb<sb>1</sb>

Also Published As

Publication number Publication date
FR2882931A1 (fr) 2006-09-15
CN101137373A (zh) 2008-03-05
BRPI0608438A2 (pt) 2009-12-29
EP1863489A1 (fr) 2007-12-12
RU2007138042A (ru) 2009-04-20
WO2006097605A1 (fr) 2006-09-21
AU2006224446A1 (en) 2006-09-21
MX2007011357A (es) 2007-11-12
IL185789A0 (en) 2008-02-09
US20080015186A1 (en) 2008-01-17
KR20070112266A (ko) 2007-11-22
JP2008533110A (ja) 2008-08-21
CA2600028A1 (fr) 2006-09-21

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Effective date: 20111130