FR2664271B1 - NEW SULFUR DERIVATIVES OF IMIDAZOLE, THEIR PREPARATION PROCESS, THE NEW INTERMEDIATES OBTAINED, THEIR APPLICATION AS MEDICAMENTS AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING THEM. - Google Patents

NEW SULFUR DERIVATIVES OF IMIDAZOLE, THEIR PREPARATION PROCESS, THE NEW INTERMEDIATES OBTAINED, THEIR APPLICATION AS MEDICAMENTS AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING THEM.

Info

Publication number
FR2664271B1
FR2664271B1 FR9008538A FR9008538A FR2664271B1 FR 2664271 B1 FR2664271 B1 FR 2664271B1 FR 9008538 A FR9008538 A FR 9008538A FR 9008538 A FR9008538 A FR 9008538A FR 2664271 B1 FR2664271 B1 FR 2664271B1
Authority
FR
France
Prior art keywords
new
medicaments
imidazole
application
pharmaceutical compositions
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
FR9008538A
Other languages
French (fr)
Other versions
FR2664271A1 (en
Inventor
Jean-Claude Caille
Alain Corbier
Michel Fortin
Gilles Hamon
Simone Jouquey
Jean-Paul Vevert
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sanofi Aventis France
Original Assignee
Roussel Uclaf SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Roussel Uclaf SA filed Critical Roussel Uclaf SA
Priority to FR9008538A priority Critical patent/FR2664271B1/en
Priority to IL98319A priority patent/IL98319A/en
Priority to MA22476A priority patent/MA22203A1/en
Priority to HU265/91A priority patent/HU217444B/en
Priority to US07/838,289 priority patent/US5412101A/en
Priority to DK91401857T priority patent/DK0465368T3/en
Priority to AT91401857T priority patent/ATE166344T1/en
Priority to FI913250A priority patent/FI111542B/en
Priority to UA5001537A priority patent/UA26130A/en
Priority to IE233591A priority patent/IE912335A1/en
Priority to SU915001537A priority patent/RU2086542C1/en
Priority to PCT/FR1991/000543 priority patent/WO2004074258A1/en
Priority to CA002046265A priority patent/CA2046265C/en
Priority to EP91401857A priority patent/EP0465368B1/en
Priority to AU80163/91A priority patent/AU653160B2/en
Priority to DE69129428T priority patent/DE69129428T2/en
Priority to ES91401857T priority patent/ES2117001T3/en
Priority to KR1019910011310A priority patent/KR100216006B1/en
Priority to OA60035A priority patent/OA09506A/en
Priority to JP19114491A priority patent/JP3192171B2/en
Priority to MX9100092A priority patent/MX9100092A/en
Priority to ZA915225A priority patent/ZA915225B/en
Priority to CN91105292A priority patent/CN1045769C/en
Publication of FR2664271A1 publication Critical patent/FR2664271A1/en
Application granted granted Critical
Publication of FR2664271B1 publication Critical patent/FR2664271B1/en
Priority to US08/369,909 priority patent/US5599830A/en
Priority to US08/723,471 priority patent/US5684028A/en
Priority to JP2000317651A priority patent/JP3261403B2/en
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/10—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/84—Sulfur atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/90—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
FR9008538A 1990-07-05 1990-07-05 NEW SULFUR DERIVATIVES OF IMIDAZOLE, THEIR PREPARATION PROCESS, THE NEW INTERMEDIATES OBTAINED, THEIR APPLICATION AS MEDICAMENTS AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING THEM. Expired - Fee Related FR2664271B1 (en)

Priority Applications (26)

Application Number Priority Date Filing Date Title
FR9008538A FR2664271B1 (en) 1990-07-05 1990-07-05 NEW SULFUR DERIVATIVES OF IMIDAZOLE, THEIR PREPARATION PROCESS, THE NEW INTERMEDIATES OBTAINED, THEIR APPLICATION AS MEDICAMENTS AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING THEM.
IL98319A IL98319A (en) 1990-07-05 1991-05-31 Sulphurous derivatives of imidazole, their preparation process, and pharmaceutical compositions containing them
MA22476A MA22203A1 (en) 1990-07-05 1991-07-03 NEW SULFUR DERIVATIVES OF IMIDAZOLE, THEIR PREPARATION PROCESS, THE NEW INTERMEDIARIES OBTAINED, THEIR APPLICATION AS MEDICINAL PRODUCTS AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
ES91401857T ES2117001T3 (en) 1990-07-05 1991-07-04 NEW SULFURATED DERIVATIVES OF IMIDAZOLE, ITS PREPARATION PROCEDURE, NEW INTERMEDIATE COMPOUNDS OBTAINED, ITS APPLICATION AS A DRUG AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING THEM.
DK91401857T DK0465368T3 (en) 1990-07-05 1991-07-04 New sulfur compounds derived from imidazole, process for their preparation, newly obtained intermediate compounds, their use
AT91401857T ATE166344T1 (en) 1990-07-05 1991-07-04 SULFUR DERIVATIVES OF IMIDAZOLE, METHOD FOR THE PRODUCTION THEREOF, INTERMEDIATE PRODUCTS, THEIR USE AS MEDICINAL PRODUCTS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
FI913250A FI111542B (en) 1990-07-05 1991-07-04 A process for the preparation of therapeutically useful sulfur derivatives of imidazole
UA5001537A UA26130A (en) 1990-07-05 1991-07-04 SULFUR-CONTAINING IMIDAZOLE DERIVATIVES WITH HYPOTHESIVE ACTIVITY, METHOD OF OBTAINING THEM, INTERMEDIATE COMPOUNDS AND PHARMACEUTICAL COMPOSITION
IE233591A IE912335A1 (en) 1990-07-05 1991-07-04 New sulphurous derivatives of imidazole, their preparation¹process, the new intermediates obtained, their use as¹medicaments and the pharmaceutical compositions containing¹them
SU915001537A RU2086542C1 (en) 1990-07-05 1991-07-04 Sulfur-containing imidazole derivatives, method of their synthesis, new intermediate compounds and pharmaceutical composition
PCT/FR1991/000543 WO2004074258A1 (en) 1990-07-05 1991-07-04 Novel sulphated imidazole derivatives, method for production thereof, novel intermediates obtained, application thereof as medicaments and pharmaceutical compositions comprising the above
CA002046265A CA2046265C (en) 1990-07-05 1991-07-04 Sulphured imadazole derivatives, their preparation process, the new intermediates obtained, their application as drugs and the pharmaceutical preparations containing them
EP91401857A EP0465368B1 (en) 1990-07-05 1991-07-04 Sulfur derivatives of imidazole, process for their preparation, intermediates, their use as medicaments, and pharmaceutical compositions containing them
AU80163/91A AU653160B2 (en) 1990-07-05 1991-07-04 New sulphurous derivatives of imidazole, their preparation process, the new intermediates obtained, their use as medicaments and the pharmaceutical compositions containing them
HU265/91A HU217444B (en) 1990-07-05 1991-07-04 Process for producing new sulfur-containing imidazol derivatives and pharmaceutical compositions containing them
US07/838,289 US5412101A (en) 1990-07-05 1991-07-04 Sulphorous derivatives of imidazole, and their use as medicaments and the pharmaceutical compositions containing them
KR1019910011310A KR100216006B1 (en) 1990-07-05 1991-07-04 Sulfur derivatives of imidazole process for their preparation intermediates their use as medicaments, and pharmaceutical compositions containing them
DE69129428T DE69129428T2 (en) 1990-07-05 1991-07-04 Sulfur derivatives of imidazole, processes for their preparation, intermediates, their use as medicines and pharmaceutical compositions containing them
JP19114491A JP3192171B2 (en) 1990-07-05 1991-07-05 Novel sulfur derivative of imidazole, process for its production, novel intermediate obtained, its use as a drug, and pharmaceutical composition containing it
MX9100092A MX9100092A (en) 1990-07-05 1991-07-05 NEW SULFURATED DERIVATIVES OF IMIDAZOLE, PROCEDURE FOR ITS PREPARATION, NEW INTERMEDIATE COMPOUNDS OBTAINED AND PHARMACEUTICAL COMPOSITIONS THAT CONTAIN THEM
ZA915225A ZA915225B (en) 1990-07-05 1991-07-05 Sulphurous derivatives of imidazole,their preparation process,the intermediate obtained,their use as medicaments and the pharmaceutical compositions containing them
CN91105292A CN1045769C (en) 1990-07-05 1991-07-05 Sulphurous derivatives of imidazole, their preparation process, intermediates obtained, their use as medicaments and pharmaceutical compositions containing them
OA60035A OA09506A (en) 1990-07-05 1991-07-05 New sulfur derivatives of imidazole their preparation process the new intermediates obtained their application as medicaments and the pharmaceutical compositions containing them
US08/369,909 US5599830A (en) 1990-07-05 1995-01-09 Sulphorous derivatives of imidazole and their use as medicaments
US08/723,471 US5684028A (en) 1990-07-05 1996-10-09 Sulphorous derivatives of imidazole, their preparation process, the new intermediates obtained, their use as medicaments and the pharmaceutical compositions
JP2000317651A JP3261403B2 (en) 1990-07-05 2000-10-18 Process for producing novel sulfur derivatives of imidazole

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9008538A FR2664271B1 (en) 1990-07-05 1990-07-05 NEW SULFUR DERIVATIVES OF IMIDAZOLE, THEIR PREPARATION PROCESS, THE NEW INTERMEDIATES OBTAINED, THEIR APPLICATION AS MEDICAMENTS AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING THEM.

Publications (2)

Publication Number Publication Date
FR2664271A1 FR2664271A1 (en) 1992-01-10
FR2664271B1 true FR2664271B1 (en) 1994-02-18

Family

ID=9398388

Family Applications (1)

Application Number Title Priority Date Filing Date
FR9008538A Expired - Fee Related FR2664271B1 (en) 1990-07-05 1990-07-05 NEW SULFUR DERIVATIVES OF IMIDAZOLE, THEIR PREPARATION PROCESS, THE NEW INTERMEDIATES OBTAINED, THEIR APPLICATION AS MEDICAMENTS AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING THEM.

Country Status (2)

Country Link
FR (1) FR2664271B1 (en)
ZA (1) ZA915225B (en)

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4179512A (en) * 1977-03-01 1979-12-18 Merck & Co., Inc. 4-Substituted-2-arylimidazoles
PT78388B (en) * 1983-04-12 1986-09-15 Smithkline Beckman Corp Dopamine-beta-hydroxylase inhibitors
CA1334092C (en) * 1986-07-11 1995-01-24 David John Carini Angiotensin ii receptor blocking imidazoles
US4882348A (en) * 1987-12-29 1989-11-21 Smithkline Beckman Corporation 2-(aminoalkylthio)imidazoles as dopamine-β-hydroxylase inhibitors
CA1338238C (en) * 1988-01-07 1996-04-09 David John Carini Angiotensin ii receptor blocking imidazoles and combinations thereof with diuretics and nsaids

Also Published As

Publication number Publication date
ZA915225B (en) 1992-09-30
FR2664271A1 (en) 1992-01-10

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TP Transmission of property
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