FR2554816B1 - NEW NORORIPAVIN DERIVATIVE HAVING BOTH AGONIST AND ANTAGONIST ACTIVITY OF MORPHINIC RECEPTORS - Google Patents

NEW NORORIPAVIN DERIVATIVE HAVING BOTH AGONIST AND ANTAGONIST ACTIVITY OF MORPHINIC RECEPTORS

Info

Publication number
FR2554816B1
FR2554816B1 FR8318230A FR8318230A FR2554816B1 FR 2554816 B1 FR2554816 B1 FR 2554816B1 FR 8318230 A FR8318230 A FR 8318230A FR 8318230 A FR8318230 A FR 8318230A FR 2554816 B1 FR2554816 B1 FR 2554816B1
Authority
FR
France
Prior art keywords
nororipavin
agonist
derivative
new
antagonist activity
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
FR8318230A
Other languages
French (fr)
Other versions
FR2554816A1 (en
Inventor
Claude Moulineau
Robert Boigegrain
Michel Morre
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sanofi SA
Original Assignee
Sanofi SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi SA filed Critical Sanofi SA
Priority to FR8318230A priority Critical patent/FR2554816B1/en
Publication of FR2554816A1 publication Critical patent/FR2554816A1/en
Application granted granted Critical
Publication of FR2554816B1 publication Critical patent/FR2554816B1/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D489/00—Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula:
    • C07D489/09—Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula: containing 4aH-8, 9 c-Iminoethano- phenanthro [4, 5-b, c, d] furan ring systems condensed with carbocyclic rings or ring systems
    • C07D489/10—Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula: containing 4aH-8, 9 c-Iminoethano- phenanthro [4, 5-b, c, d] furan ring systems condensed with carbocyclic rings or ring systems with a bridge between positions 6 and 14
    • C07D489/12—Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula: containing 4aH-8, 9 c-Iminoethano- phenanthro [4, 5-b, c, d] furan ring systems condensed with carbocyclic rings or ring systems with a bridge between positions 6 and 14 the bridge containing only two carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
FR8318230A 1983-11-16 1983-11-16 NEW NORORIPAVIN DERIVATIVE HAVING BOTH AGONIST AND ANTAGONIST ACTIVITY OF MORPHINIC RECEPTORS Expired FR2554816B1 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
FR8318230A FR2554816B1 (en) 1983-11-16 1983-11-16 NEW NORORIPAVIN DERIVATIVE HAVING BOTH AGONIST AND ANTAGONIST ACTIVITY OF MORPHINIC RECEPTORS

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR8318230A FR2554816B1 (en) 1983-11-16 1983-11-16 NEW NORORIPAVIN DERIVATIVE HAVING BOTH AGONIST AND ANTAGONIST ACTIVITY OF MORPHINIC RECEPTORS

Publications (2)

Publication Number Publication Date
FR2554816A1 FR2554816A1 (en) 1985-05-17
FR2554816B1 true FR2554816B1 (en) 1986-09-26

Family

ID=9294184

Family Applications (1)

Application Number Title Priority Date Filing Date
FR8318230A Expired FR2554816B1 (en) 1983-11-16 1983-11-16 NEW NORORIPAVIN DERIVATIVE HAVING BOTH AGONIST AND ANTAGONIST ACTIVITY OF MORPHINIC RECEPTORS

Country Status (1)

Country Link
FR (1) FR2554816B1 (en)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2388369B (en) 2002-05-10 2004-05-05 Reckitt Benckiser Healthcare Demethylation of thebaine derivative
EP3321269B1 (en) 2011-10-03 2020-04-29 Johnson Matthey Public Limited Company Process for preparing buprenorphine intermediates

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1136214A (en) * 1965-06-15 1968-12-11 Reckitt & Sons Ltd Thebaine and oripavine derivatives
FR1481859A (en) * 1965-06-03 1967-05-19 Reckitt And Sons Ltd Process for the preparation of thebaine compounds

Also Published As

Publication number Publication date
FR2554816A1 (en) 1985-05-17

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Legal Events

Date Code Title Description
ST Notification of lapse