FR2422645A1 - BENZIMIDAZOLES DERIVATIVES WITH ANTHELMINTIC ACTIVITY - Google Patents

BENZIMIDAZOLES DERIVATIVES WITH ANTHELMINTIC ACTIVITY

Info

Publication number
FR2422645A1
FR2422645A1 FR7836791A FR7836791A FR2422645A1 FR 2422645 A1 FR2422645 A1 FR 2422645A1 FR 7836791 A FR7836791 A FR 7836791A FR 7836791 A FR7836791 A FR 7836791A FR 2422645 A1 FR2422645 A1 FR 2422645A1
Authority
FR
France
Prior art keywords
anthelmintic activity
benzimidazoles derivatives
benzimidazoles
derivatives
anthelmintic
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
FR7836791A
Other languages
French (fr)
Inventor
Rudiger D Haugwitz
Barbara V Maurer
Peter C Wade
Larry R Cruthers
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
ER Squibb and Sons LLC
Original Assignee
ER Squibb and Sons LLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US05/868,148 external-priority patent/US4156006A/en
Priority claimed from US05/870,391 external-priority patent/US4136174A/en
Priority claimed from US05/885,717 external-priority patent/US4138493A/en
Application filed by ER Squibb and Sons LLC filed Critical ER Squibb and Sons LLC
Publication of FR2422645A1 publication Critical patent/FR2422645A1/en
Withdrawn legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C17/00—Preparation of halogenated hydrocarbons
    • C07C17/26—Preparation of halogenated hydrocarbons by reactions involving an increase in the number of carbon atoms in the skeleton
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/24—Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • C07D235/30—Nitrogen atoms not forming part of a nitro radical
    • C07D235/32—Benzimidazole-2-carbamic acids, unsubstituted or substituted; Esters thereof; Thio-analogues thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic System
    • C07F7/02—Silicon compounds
    • C07F7/08—Compounds having one or more C—Si linkages
    • C07F7/0803—Compounds with Si-C or Si-Si linkages
    • C07F7/081—Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te
    • C07F7/0812—Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te comprising a heterocyclic ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic System
    • C07F7/02—Silicon compounds
    • C07F7/08—Compounds having one or more C—Si linkages
    • C07F7/18—Compounds having one or more C—Si linkages as well as one or more C—O—Si linkages
    • C07F7/1804—Compounds having Si-O-C linkages

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

L'invention concerne des benzimidazoles de formule :The invention relates to benzimidazoles of the formula:

FR7836791A 1978-01-09 1978-12-28 BENZIMIDAZOLES DERIVATIVES WITH ANTHELMINTIC ACTIVITY Withdrawn FR2422645A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US05/868,148 US4156006A (en) 1978-01-09 1978-01-09 Vinyl sulfide derivatives of benzimidazoles
US05/870,391 US4136174A (en) 1978-01-18 1978-01-18 Benzimidazolecarbamates and method
US05/885,717 US4138493A (en) 1978-03-13 1978-03-13 2,2-Dihalo-1(3)-lower alkyl-cyclopropylalkylthio benzimidazole derivatives, compositions thereof and method of use in treating tapeworms and whipworms

Publications (1)

Publication Number Publication Date
FR2422645A1 true FR2422645A1 (en) 1979-11-09

Family

ID=27420450

Family Applications (1)

Application Number Title Priority Date Filing Date
FR7836791A Withdrawn FR2422645A1 (en) 1978-01-09 1978-12-28 BENZIMIDAZOLES DERIVATIVES WITH ANTHELMINTIC ACTIVITY

Country Status (8)

Country Link
JP (1) JPS54100374A (en)
AU (1) AU4185678A (en)
CA (1) CA1117538A (en)
DE (1) DE2856796A1 (en)
FR (1) FR2422645A1 (en)
GB (1) GB2011896A (en)
IE (1) IE47530B1 (en)
IT (1) IT1102784B (en)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2443461A1 (en) * 1978-12-06 1980-07-04 Montedison Spa BENZIMIDAZOLE-CARBAMATES AND ITS APPLICATION IN VETERINARY MEDICINE

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2443461A1 (en) * 1978-12-06 1980-07-04 Montedison Spa BENZIMIDAZOLE-CARBAMATES AND ITS APPLICATION IN VETERINARY MEDICINE

Also Published As

Publication number Publication date
IT1102784B (en) 1985-10-07
IE782412L (en) 1979-07-09
IT7831383A0 (en) 1978-12-28
DE2856796A1 (en) 1979-07-12
AU4185678A (en) 1979-07-19
JPS54100374A (en) 1979-08-08
IE47530B1 (en) 1984-04-18
GB2011896A (en) 1979-07-18
CA1117538A (en) 1982-02-02

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Legal Events

Date Code Title Description
ST Notification of lapse