FR2406631A1 - NEW A-HALOGENOMETHYL HISTAMINE DERIVATIVES USEFUL IN PARTICULAR AS ANTIHISTAMINICS AND THEIR PROCESS FOR PREPARATION - Google Patents
NEW A-HALOGENOMETHYL HISTAMINE DERIVATIVES USEFUL IN PARTICULAR AS ANTIHISTAMINICS AND THEIR PROCESS FOR PREPARATIONInfo
- Publication number
- FR2406631A1 FR2406631A1 FR7829697A FR7829697A FR2406631A1 FR 2406631 A1 FR2406631 A1 FR 2406631A1 FR 7829697 A FR7829697 A FR 7829697A FR 7829697 A FR7829697 A FR 7829697A FR 2406631 A1 FR2406631 A1 FR 2406631A1
- Authority
- FR
- France
- Prior art keywords
- antihistaminics
- halogenomethyl
- preparation
- new
- derivatives useful
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/64—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
L'invention concerne de nouveaux dérivés alpha -halogénométhylés d'histamine répondant à la formule générale :The invention relates to novel alpha-halogenomethylated histamine derivatives corresponding to the general formula:
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US84365977A | 1977-10-19 | 1977-10-19 |
Publications (2)
Publication Number | Publication Date |
---|---|
FR2406631A1 true FR2406631A1 (en) | 1979-05-18 |
FR2406631B1 FR2406631B1 (en) | 1980-09-19 |
Family
ID=25290634
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FR7829697A Granted FR2406631A1 (en) | 1977-10-19 | 1978-10-18 | NEW A-HALOGENOMETHYL HISTAMINE DERIVATIVES USEFUL IN PARTICULAR AS ANTIHISTAMINICS AND THEIR PROCESS FOR PREPARATION |
Country Status (13)
Country | Link |
---|---|
JP (1) | JPS5466676A (en) |
AU (1) | AU522245B2 (en) |
BE (1) | BE871356A (en) |
CA (1) | CA1111432A (en) |
CH (1) | CH637384A5 (en) |
DE (1) | DE2844104A1 (en) |
ES (1) | ES474321A1 (en) |
FR (1) | FR2406631A1 (en) |
GB (1) | GB2007231B (en) |
IT (1) | IT1106448B (en) |
NL (1) | NL7810173A (en) |
NZ (1) | NZ188498A (en) |
ZA (1) | ZA785435B (en) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CA1302919C (en) * | 1985-07-03 | 1992-06-09 | Robert T. Buckler | Histamine derivatives, immunogen conjugates and antibodies raised thereto |
JP2009184686A (en) * | 2008-02-04 | 2009-08-20 | Mitsubishi Heavy Industries Food & Packaging Machinery Co Ltd | Rotary filling machine and filling method of rotary filling machine |
Citations (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR1457259A (en) * | 1961-08-18 | 1966-01-24 | Merck & Co Inc | Production of alpha-alkyl-histidine amino acids |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE920250C (en) * | 1951-09-19 | 1954-11-18 | Hoffmann La Roche | Process for the preparation of 4-(ª-amino-ª-bromopropyl)imidazole salts |
DE1161903B (en) * | 1960-08-19 | 1964-01-30 | Merck & Co Inc | Process for the production of ª ‡ -Methyl-dl-histidine with antihistamine activity |
IE46910B1 (en) * | 1977-06-01 | 1983-11-02 | Merck & Co Inc | Fluorinated alkylamines and process for preparing same |
-
1978
- 1978-09-25 NZ NZ188498A patent/NZ188498A/en unknown
- 1978-09-25 ZA ZA00785435A patent/ZA785435B/en unknown
- 1978-09-26 CA CA312,083A patent/CA1111432A/en not_active Expired
- 1978-10-10 DE DE19782844104 patent/DE2844104A1/en not_active Withdrawn
- 1978-10-10 NL NL7810173A patent/NL7810173A/en not_active Application Discontinuation
- 1978-10-13 CH CH1066078A patent/CH637384A5/en not_active IP Right Cessation
- 1978-10-13 AU AU40706/78A patent/AU522245B2/en not_active Expired
- 1978-10-16 GB GB7840731A patent/GB2007231B/en not_active Expired
- 1978-10-17 IT IT51542/78A patent/IT1106448B/en active
- 1978-10-18 BE BE191193A patent/BE871356A/en not_active IP Right Cessation
- 1978-10-18 JP JP12746678A patent/JPS5466676A/en active Granted
- 1978-10-18 ES ES474321A patent/ES474321A1/en not_active Expired
- 1978-10-18 FR FR7829697A patent/FR2406631A1/en active Granted
Patent Citations (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR1457259A (en) * | 1961-08-18 | 1966-01-24 | Merck & Co Inc | Production of alpha-alkyl-histidine amino acids |
Also Published As
Publication number | Publication date |
---|---|
CH637384A5 (en) | 1983-07-29 |
ZA785435B (en) | 1979-09-26 |
AU522245B2 (en) | 1982-05-27 |
BE871356A (en) | 1979-02-15 |
DE2844104A1 (en) | 1979-04-26 |
JPS6223753B2 (en) | 1987-05-25 |
ES474321A1 (en) | 1980-01-16 |
AU4070678A (en) | 1980-04-17 |
GB2007231B (en) | 1982-03-24 |
GB2007231A (en) | 1979-05-16 |
IT1106448B (en) | 1985-11-11 |
CA1111432A (en) | 1981-10-27 |
NZ188498A (en) | 1980-08-26 |
FR2406631B1 (en) | 1980-09-19 |
NL7810173A (en) | 1979-04-23 |
IT7851542A0 (en) | 1978-10-17 |
JPS5466676A (en) | 1979-05-29 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
ST | Notification of lapse |