FR2362141A1 - N- (6- (R3R4N) -4 (OR 5) -R5-3-PYRIDAZINYL) THERAPEUTIC ALKYLIDENYL AMINOMETHYLENEMALONATES - Google Patents

N- (6- (R3R4N) -4 (OR 5) -R5-3-PYRIDAZINYL) THERAPEUTIC ALKYLIDENYL AMINOMETHYLENEMALONATES

Info

Publication number
FR2362141A1
FR2362141A1 FR7725414A FR7725414A FR2362141A1 FR 2362141 A1 FR2362141 A1 FR 2362141A1 FR 7725414 A FR7725414 A FR 7725414A FR 7725414 A FR7725414 A FR 7725414A FR 2362141 A1 FR2362141 A1 FR 2362141A1
Authority
FR
France
Prior art keywords
aminomethylenemalonates
alkylidenyl
r3r4n
pyridazinyl
therapeutic
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
FR7725414A
Other languages
French (fr)
Other versions
FR2362141B1 (en
Inventor
Y Lesher
Chester J Opalka Jr
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
STWB Inc
Original Assignee
Sterling Drug Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US05/805,419 external-priority patent/US4104385A/en
Application filed by Sterling Drug Inc filed Critical Sterling Drug Inc
Publication of FR2362141A1 publication Critical patent/FR2362141A1/en
Application granted granted Critical
Publication of FR2362141B1 publication Critical patent/FR2362141B1/fr
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D237/00—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
    • C07D237/02—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings
    • C07D237/06—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
    • C07D237/10—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D237/20—Nitrogen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Nouveaux composés à activité chimiothérapeutique. N-16-(R3 R4 N)-4 (ou 5)-R5 -3-pyfidazinylõ aminométhylènemalonates d'alkylidényle cyclique de formule :New compounds with chemotherapeutic activity. Cyclic alkylidenyl N-16- (R3 R4 N) -4 (or 5) -R5 -3-pyfidazinylõ aminomethylenemalonates of the formula:

FR7725414A 1976-08-19 1977-08-19 N- (6- (R3R4N) -4 (OR 5) -R5-3-PYRIDAZINYL) THERAPEUTIC ALKYLIDENYL AMINOMETHYLENEMALONATES Granted FR2362141A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US71569976A 1976-08-19 1976-08-19
US05/805,419 US4104385A (en) 1976-08-19 1977-06-10 Cyclic alkylidenyl N-[6-(amino)-3-pyridazinyl]aminomethylenemalonates

Publications (2)

Publication Number Publication Date
FR2362141A1 true FR2362141A1 (en) 1978-03-17
FR2362141B1 FR2362141B1 (en) 1981-07-17

Family

ID=27109402

Family Applications (1)

Application Number Title Priority Date Filing Date
FR7725414A Granted FR2362141A1 (en) 1976-08-19 1977-08-19 N- (6- (R3R4N) -4 (OR 5) -R5-3-PYRIDAZINYL) THERAPEUTIC ALKYLIDENYL AMINOMETHYLENEMALONATES

Country Status (14)

Country Link
JP (1) JPS5334782A (en)
AR (1) AR221687A1 (en)
AU (1) AU515629B2 (en)
DE (1) DE2737542A1 (en)
DK (1) DK368177A (en)
EG (1) EG12733A (en)
FR (1) FR2362141A1 (en)
GB (1) GB1542030A (en)
IL (1) IL52681A (en)
LU (1) LU77976A1 (en)
NL (1) NL7709162A (en)
NZ (1) NZ184875A (en)
PH (1) PH12796A (en)
PT (1) PT66928B (en)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH03133573A (en) * 1989-07-26 1991-06-06 Sanso Aaku Kogyo Kk Melt-cutting electrode
WO1999021834A1 (en) * 1997-10-27 1999-05-06 Neurosearch A/S Heteroaryl diazacycloalkanes as cholinergic ligands at nicotinic acetylcholine receptors

Also Published As

Publication number Publication date
AU515629B2 (en) 1981-04-16
EG12733A (en) 1979-09-30
IL52681A (en) 1981-06-29
AU2770477A (en) 1979-02-15
FR2362141B1 (en) 1981-07-17
AR221687A1 (en) 1981-03-13
IL52681A0 (en) 1977-10-31
PT66928B (en) 1979-02-05
DK368177A (en) 1978-02-20
GB1542030A (en) 1979-03-14
NZ184875A (en) 1979-03-28
DE2737542A1 (en) 1978-02-23
PH12796A (en) 1979-08-17
NL7709162A (en) 1978-02-21
PT66928A (en) 1977-09-01
LU77976A1 (en) 1978-04-27
JPS5334782A (en) 1978-03-31

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Legal Events

Date Code Title Description
ST Notification of lapse