FR2326928A1 - ANTIBACTERIAL PHOSPHONOPENAM DERIVATIVES AND PRODUCTION PROCESS - Google Patents

ANTIBACTERIAL PHOSPHONOPENAM DERIVATIVES AND PRODUCTION PROCESS

Info

Publication number
FR2326928A1
FR2326928A1 FR7629606A FR7629606A FR2326928A1 FR 2326928 A1 FR2326928 A1 FR 2326928A1 FR 7629606 A FR7629606 A FR 7629606A FR 7629606 A FR7629606 A FR 7629606A FR 2326928 A1 FR2326928 A1 FR 2326928A1
Authority
FR
France
Prior art keywords
phosphonopenam
antibacterial
derivatives
production process
production
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
FR7629606A
Other languages
French (fr)
Other versions
FR2326928B1 (en
Inventor
Wayne Ernest Barth
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Inc
Original Assignee
Pfizer Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Inc filed Critical Pfizer Inc
Publication of FR2326928A1 publication Critical patent/FR2326928A1/en
Application granted granted Critical
Publication of FR2326928B1 publication Critical patent/FR2326928B1/fr
Granted legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D499/00Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • AHUMAN NECESSITIES
    • A23FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
    • A23KFODDER
    • A23K20/00Accessory food factors for animal feeding-stuffs
    • A23K20/10Organic substances
    • A23K20/116Heterocyclic compounds
    • AHUMAN NECESSITIES
    • A23FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
    • A23KFODDER
    • A23K20/00Accessory food factors for animal feeding-stuffs
    • A23K20/10Organic substances
    • A23K20/116Heterocyclic compounds
    • A23K20/137Heterocyclic compounds containing two hetero atoms, of which at least one is nitrogen
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/08Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D277/10Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic System
    • C07F9/02Phosphorus compounds
    • C07F9/547Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6561Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing systems of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring or ring system, with or without other non-condensed hetero rings
    • C07F9/65611Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing systems of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring or ring system, with or without other non-condensed hetero rings containing the ring system (X = CH2, O, S, NH) optionally with an additional double bond and/or substituents, e.g. penicillins and analogs
FR7629606A 1975-10-06 1976-10-01 ANTIBACTERIAL PHOSPHONOPENAM DERIVATIVES AND PRODUCTION PROCESS Granted FR2326928A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US61963475A 1975-10-06 1975-10-06
US05/680,423 US4031077A (en) 1975-10-06 1976-04-26 Antibacterial 3-phosphono penams

Publications (2)

Publication Number Publication Date
FR2326928A1 true FR2326928A1 (en) 1977-05-06
FR2326928B1 FR2326928B1 (en) 1980-12-26

Family

ID=27088560

Family Applications (2)

Application Number Title Priority Date Filing Date
FR7629606A Granted FR2326928A1 (en) 1975-10-06 1976-10-01 ANTIBACTERIAL PHOSPHONOPENAM DERIVATIVES AND PRODUCTION PROCESS
FR7712772A Granted FR2337728A1 (en) 1975-10-06 1977-04-27 NEW INTERMEDIARIES FOR THE PREPARATION OF PENAM DERIVATIVES

Family Applications After (1)

Application Number Title Priority Date Filing Date
FR7712772A Granted FR2337728A1 (en) 1975-10-06 1977-04-27 NEW INTERMEDIARIES FOR THE PREPARATION OF PENAM DERIVATIVES

Country Status (13)

Country Link
US (1) US4031077A (en)
JP (1) JPS5921878B2 (en)
AR (2) AR212638A1 (en)
CA (1) CA1094548A (en)
DE (1) DE2643577A1 (en)
DK (1) DK145060C (en)
ES (1) ES451982A1 (en)
FR (2) FR2326928A1 (en)
GB (2) GB1526150A (en)
IE (1) IE43398B1 (en)
LU (1) LU75919A1 (en)
NL (1) NL7610821A (en)
SE (2) SE7610632L (en)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4136096A (en) * 1977-02-25 1979-01-23 Pfizer Inc. 6-amino-2,2-dimethyl-3-(5-tetrazolyl)penam process and intermediates therefor
JPS614584U (en) * 1984-06-15 1986-01-11 宏 田口 Fishing bait container and fish collector
US5067945A (en) * 1988-03-01 1991-11-26 Ryan Medical, Inc. Safety needled medical devices capable of one-handed manipulation

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3870713A (en) * 1970-12-07 1975-03-11 Pfizer Phosphono substituted alkylcephalosporins
US3875152A (en) * 1971-11-09 1975-04-01 American Home Prod Intermediates for producing semi-synthetic cephalosporins and methods of production
US4032521A (en) * 1972-12-29 1977-06-28 Merck & Co., Inc. Cephalosporin phosphonic acid, sulfonic acid and sulfonamide compounds

Also Published As

Publication number Publication date
FR2326928B1 (en) 1980-12-26
CA1094548A (en) 1981-01-27
DE2643577A1 (en) 1977-05-12
LU75919A1 (en) 1977-05-25
ES451982A1 (en) 1977-10-01
GB1526149A (en) 1978-09-27
FR2337728A1 (en) 1977-08-05
JPS5265290A (en) 1977-05-30
SE7610632L (en) 1977-04-07
AR211565A1 (en) 1978-01-30
AR212638A1 (en) 1978-08-31
DK145060C (en) 1983-01-17
IE43398L (en) 1977-04-06
IE43398B1 (en) 1981-02-11
DK440476A (en) 1977-04-07
US4031077A (en) 1977-06-21
NL7610821A (en) 1977-04-12
DK145060B (en) 1982-08-16
JPS5921878B2 (en) 1984-05-22
SE8104682L (en) 1981-08-04
GB1526150A (en) 1978-09-27
FR2337728B1 (en) 1980-10-17

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Legal Events

Date Code Title Description
ST Notification of lapse