FR1545694A - Préparation de composés de la série des benzodiazépines - Google Patents

Préparation de composés de la série des benzodiazépines

Info

Publication number
FR1545694A
FR1545694A FR117190A FR117190A FR1545694A FR 1545694 A FR1545694 A FR 1545694A FR 117190 A FR117190 A FR 117190A FR 117190 A FR117190 A FR 117190A FR 1545694 A FR1545694 A FR 1545694A
Authority
FR
France
Prior art keywords
compounds
preparation
benzodiazepine series
benzodiazepine
series
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
FR117190A
Other languages
English (en)
Inventor
Josef Schmitt
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Clin Byla SA
Original Assignee
Clin Byla SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Clin Byla SA filed Critical Clin Byla SA
Priority to FR117190A priority Critical patent/FR1545694A/fr
Priority to IE917/68A priority patent/IE32395B1/xx
Priority to IE680/71A priority patent/IE32396B1/xx
Priority to IL30470A priority patent/IL30470A0/xx
Priority to DE19681795053 priority patent/DE1795053A1/de
Priority to CH1176568A priority patent/CH488711A/fr
Priority to SE10550/68A priority patent/SE351430B/xx
Priority to CH255070A priority patent/CH491939A/fr
Priority to SE12794/71A priority patent/SE366316B/xx
Priority to GB37560/68A priority patent/GB1223032A/en
Priority to GB32016/70A priority patent/GB1224720A/en
Priority to NL6811210A priority patent/NL6811210A/xx
Priority to BE719199D priority patent/BE719199A/xx
Priority to DK380568AA priority patent/DK117426B/da
Priority to ES357055A priority patent/ES357055A1/es
Priority to US773368A priority patent/US3551412A/en
Application granted granted Critical
Publication of FR1545694A publication Critical patent/FR1545694A/fr
Priority to DK21070AA priority patent/DK126943B/da
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D243/00Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/141,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/161,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • C07D243/181,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
    • C07D243/24Oxygen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D243/00Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/141,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
FR117190A 1967-08-08 1967-08-08 Préparation de composés de la série des benzodiazépines Expired FR1545694A (fr)

Priority Applications (17)

Application Number Priority Date Filing Date Title
FR117190A FR1545694A (fr) 1967-08-08 1967-08-08 Préparation de composés de la série des benzodiazépines
IE917/68A IE32395B1 (en) 1967-08-08 1968-07-30 Benzodiazepine derivatives
IE680/71A IE32396B1 (en) 1967-08-08 1968-07-30 Production of benzodiazepines
IL30470A IL30470A0 (en) 1967-08-08 1968-07-31 Preparation of 5-substituted benzodiazepines
DE19681795053 DE1795053A1 (de) 1967-08-08 1968-08-02 Verfahren zur Herstellung von Verbindungen der Benzodiazepinreihe
SE12794/71A SE366316B (fr) 1967-08-08 1968-08-05
SE10550/68A SE351430B (fr) 1967-08-08 1968-08-05
CH255070A CH491939A (fr) 1967-08-08 1968-08-05 Procédé de préparation d'un composé de la série des benzodiazépines
CH1176568A CH488711A (fr) 1967-08-08 1968-08-05 Procédé de préparation de composés de la série des benzodiazépines
GB37560/68A GB1223032A (en) 1967-08-08 1968-08-06 Benzodiazepine derivatives
GB32016/70A GB1224720A (en) 1967-08-08 1968-08-06 Production of benzodiazepines
BE719199D BE719199A (fr) 1967-08-08 1968-08-07
DK380568AA DK117426B (da) 1967-08-08 1968-08-07 Fremgangsmåde til fremstilling af en 5-(1-cylohexenyl)-2-oxo-2,3-dihyro-1H-1,4-benzodiazepin.
NL6811210A NL6811210A (fr) 1967-08-08 1968-08-07
ES357055A ES357055A1 (es) 1967-08-08 1968-08-08 Procedimiento de obtencion de derivados en benzodiazepina halogenados.
US773368A US3551412A (en) 1967-08-08 1968-10-29 5-substituted benzodiazepines
DK21070AA DK126943B (da) 1967-08-08 1970-01-19 1-Alkylsubstituerede 1,4-benzodiazepiner til anvendelse ved fremstillingen af 1,4-benzodiazepiner med nyttige fysiologiske virkninger og fremgangsmåde til fremstilling deraf.

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR117190A FR1545694A (fr) 1967-08-08 1967-08-08 Préparation de composés de la série des benzodiazépines

Publications (1)

Publication Number Publication Date
FR1545694A true FR1545694A (fr) 1968-11-15

Family

ID=8636550

Family Applications (1)

Application Number Title Priority Date Filing Date
FR117190A Expired FR1545694A (fr) 1967-08-08 1967-08-08 Préparation de composés de la série des benzodiazépines

Country Status (12)

Country Link
US (1) US3551412A (fr)
BE (1) BE719199A (fr)
CH (1) CH488711A (fr)
DE (1) DE1795053A1 (fr)
DK (2) DK117426B (fr)
ES (1) ES357055A1 (fr)
FR (1) FR1545694A (fr)
GB (2) GB1224720A (fr)
IE (1) IE32395B1 (fr)
IL (1) IL30470A0 (fr)
NL (1) NL6811210A (fr)
SE (2) SE351430B (fr)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4368157A (en) * 1978-05-15 1983-01-11 Hoffmann-La Roche Inc. Intermediates to produce imidazodiazepines
US4368159A (en) * 1978-05-15 1983-01-11 Hoffmann-La Roche Inc. Intermediates to produce imidazodiazepines
US4401597A (en) * 1978-05-15 1983-08-30 Hoffmann-La Roche Inc. Imidazodiazepines and processes therefor

Also Published As

Publication number Publication date
US3551412A (en) 1970-12-29
GB1223032A (en) 1971-02-17
IL30470A0 (en) 1968-09-26
SE351430B (fr) 1972-11-27
CH488711A (fr) 1970-04-15
NL6811210A (fr) 1969-02-11
IE32395L (en) 1969-02-08
BE719199A (fr) 1969-01-16
DK126943B (da) 1973-09-03
ES357055A1 (es) 1970-02-16
SE366316B (fr) 1974-04-22
DK117426B (da) 1970-04-27
DE1795053A1 (de) 1972-01-05
GB1224720A (en) 1971-03-10
IE32395B1 (en) 1973-07-25

Similar Documents

Publication Publication Date Title
CH486427A (fr) Procédé de préparation d'amidines aromatiques N. substituées
OA03388A (fr) Nouveaux composés bicycliques et leur préparation.
FI791055A (fi) Foerfarande foer framstaellning av 5-fenyl-1h-1,5-bensodiazepin-2,4-dioner
FR1455581A (fr) Azurants de la série stilbénique et leur préparation
FR1541746A (fr) Préparation de la canthaxanthine
CH508653A (fr) Procédé de préparation de benzothiazin-4-ones substituées
FR1503630A (fr) Préparation de composés fluoroaromatiques
FR1545694A (fr) Préparation de composés de la série des benzodiazépines
FR1462206A (fr) Composés gem-bithiényliques et leur préparation
FI48090C (fi) Menetelmä 1-syaaniaminoalkyyli-2H-1,4-bentsodiatsepiini-2-oni-johdanna isten valmistamiseksi
CH497407A (de) Procédé de préparation de 2,2-diméthyl stéroides insaturés
FI48087C (fi) Menetelmä 5-fenyyli-1,3,4,5-tetrahydro-2H-1,4-bentsodiatsepiini-2-onie n valmistamiseksi
FR1543469A (fr) Composés de la classe des beta-hydroxyphosphonates et leur obtention
FR1438608A (fr) Composés de la série de la vitamine alpha et leur préparation
FR1455048A (fr) Composés de la série des benzodiazépines et leur préparation
FR1528292A (fr) Préparation de copolymères de lactame-lactone
FR1527707A (fr) Préparation de la 5-5-diméthyl-2-pipéridone
FR1475374A (fr) Préparation de composés de 5-cyano-uraciles
OA02877A (fr) Procédé de préparation de benzène-sulfonyl-urées.
OA02250A (fr) Préparation de benzène-sulfonyl-urées.
FR1506734A (fr) Composés dibenzo-azépiniques et leur préparation
FR1449298A (fr) Préparation de composés diorgano-zinciques
FR1501589A (fr) Préparation de formylméthylène-4-oxazolidinones-2
CH495929A (fr) Préparation de composés biallyliques
FR1501498A (fr) Composés azépiniques et leur prépartion