FR1423609A - Dérivés de la benzimidazole et leur procédé de fabrication - Google Patents
Dérivés de la benzimidazole et leur procédé de fabricationInfo
- Publication number
- FR1423609A FR1423609A FR849060A FR849060A FR1423609A FR 1423609 A FR1423609 A FR 1423609A FR 849060 A FR849060 A FR 849060A FR 849060 A FR849060 A FR 849060A FR 1423609 A FR1423609 A FR 1423609A
- Authority
- FR
- France
- Prior art keywords
- manufacturing process
- benzimidazole derivatives
- benzimidazole
- derivatives
- manufacturing
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR877469A FR1879M (fr) | 1961-01-06 | 1961-10-30 | Dérivés du benzimidazole comme médicaments noveaux pour le traitement des affections helminthiques. |
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US2856A US3017415A (en) | 1960-01-18 | 1960-01-18 | Certain benzimidazoles carrying thiazolyl, thiadiazolyl and isothiazolyl substituents in the 2 position |
| US15518A US3055907A (en) | 1960-01-18 | 1960-03-17 | Acyl benzimidazoles and method of preparing same |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| FR1423609A true FR1423609A (fr) | 1966-01-07 |
Family
ID=26670973
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| FR849060A Expired FR1423609A (fr) | 1960-01-18 | 1961-01-06 | Dérivés de la benzimidazole et leur procédé de fabrication |
Country Status (12)
| Country | Link |
|---|---|
| US (2) | US3017415A (cg-RX-API-DMAC7.html) |
| BE (1) | BE599143A (cg-RX-API-DMAC7.html) |
| CH (5) | CH423791A (cg-RX-API-DMAC7.html) |
| CY (1) | CY309A (cg-RX-API-DMAC7.html) |
| DE (1) | DE1235321B (cg-RX-API-DMAC7.html) |
| DK (1) | DK107167C (cg-RX-API-DMAC7.html) |
| ES (1) | ES263822A1 (cg-RX-API-DMAC7.html) |
| FR (1) | FR1423609A (cg-RX-API-DMAC7.html) |
| GB (1) | GB948635A (cg-RX-API-DMAC7.html) |
| MY (1) | MY6500075A (cg-RX-API-DMAC7.html) |
| OA (1) | OA00999A (cg-RX-API-DMAC7.html) |
| SE (2) | SE310883B (cg-RX-API-DMAC7.html) |
Cited By (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0387941A1 (en) * | 1989-03-15 | 1990-09-19 | Janssen Pharmaceutica N.V. | [5(6)-(benzisoxa-, benzisothia- or indazol-3-yl)-1H-benzimidazol-2-yl] carbamates |
| WO1990010630A1 (en) * | 1989-03-15 | 1990-09-20 | Janssen Pharmaceutica N.V. | [5(6)-(benzisoxa-, benzisothia- or indazol-3-yl)-1h-benzimidazol-2-yl] carbamates |
| WO1994025457A1 (en) * | 1993-04-30 | 1994-11-10 | E.I. Du Pont De Nemours And Company | Process for preparing thiabendazole |
Families Citing this family (57)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3239532A (en) * | 1960-04-07 | 1966-03-08 | Geigy Ag J R | Certain diazolylmethyl esters of thiophosphoric and dithiophosphoric acids |
| NL133760C (cg-RX-API-DMAC7.html) * | 1961-02-23 | |||
| NL295012A (cg-RX-API-DMAC7.html) * | 1962-07-05 | |||
| US3324102A (en) * | 1963-01-31 | 1967-06-06 | Merck & Co Inc | Water-soluble benzimidazole-containing coordination compounds and methods relating thereto |
| NL134354C (cg-RX-API-DMAC7.html) * | 1963-05-23 | |||
| GB1069937A (en) * | 1963-06-24 | 1967-05-24 | Merck & Co Inc | N-(halopyruvoyl)-nitroanilides |
| US3471508A (en) * | 1963-11-06 | 1969-10-07 | Merck & Co Inc | 5-aryl (or heteroaromatic) benzazoles |
| IL22369A (en) * | 1963-11-19 | 1968-10-24 | Merck & Co Inc | 2-heteroaryl-5 and/or 6-substituted benzazoles |
| GB1082354A (en) * | 1963-11-29 | 1967-09-06 | Merck & Co Inc | Trifluoroacetoxy-haloalkyl benzimidazoles |
| US3350211A (en) * | 1964-12-31 | 1967-10-31 | Merck & Co Inc | Compositions useful in controlling marine fouling and methods for their use |
| BR6575771D0 (pt) * | 1964-12-31 | 1973-12-26 | Merck & Co Inc | Processo para preparar 1-oxido de benzimidazol |
| US3429890A (en) * | 1964-12-31 | 1969-02-25 | Merck & Co Inc | Certain 2-thiazolylbenzimidazole-1-oxy derivatives |
| US3484519A (en) * | 1965-12-02 | 1969-12-16 | Merck & Co Inc | Anthelmintic 2-substituted benzimidazole-metal arsenate compositions and method |
| US3475444A (en) * | 1966-02-18 | 1969-10-28 | Merck & Co Inc | Complexes of 2-substituted benzimidazoles and bis-halogenated phenols |
| US3546341A (en) * | 1966-02-18 | 1970-12-08 | Merck & Co Inc | Complexes of 2-substituted benzimidazoles and bis-halogenated phenols in anthelmintic compositions and methods |
| US3506678A (en) * | 1967-02-21 | 1970-04-14 | Merck & Co Inc | Certain 2-substituted thieno(2,3-d) imidazoles |
| US3535331A (en) * | 1967-07-26 | 1970-10-20 | Merck & Co Inc | Water-soluble 2-substituted benzimidazole hypophosphite salts |
| US3538108A (en) * | 1967-08-17 | 1970-11-03 | Merck & Co Inc | Water - soluble 2 - substituted benzimidazole methanesulfonic acid salts |
| GB1221596A (en) * | 1967-12-06 | 1971-02-03 | Merck & Co Inc | Benzimidazole derivatives |
| US3625954A (en) * | 1968-03-20 | 1971-12-07 | Pfizer | 1-aroylbenzimidazoles |
| US3711608A (en) * | 1971-04-13 | 1973-01-16 | Merck & Co Inc | The treatment of pain, fever and inflammation with benzimidazoles |
| US3864351A (en) * | 1971-10-04 | 1975-02-04 | Pfizer | 1-({60 -Carboxymethoxybenzoyl-2-(2{40 -pyridyl)benzimidazoles |
| US3899503A (en) * | 1974-01-25 | 1975-08-12 | Morton Norwich Products Inc | Process for preparing 2-(2{40 )-furyl-, 2-(2{40 )-thienyl- 2-(4{40 )-thiazolyl- or 2-(2{40 )-pyrryl-5 (or 6) nitrobenzimidazole |
| US3998785A (en) * | 1974-06-13 | 1976-12-21 | International Business Machines Corporation | Anti-fungal and/or anti-bacterial hardware for ink printing apparatus |
| US4006259A (en) * | 1975-04-01 | 1977-02-01 | Fmc Corporation | Preservative coating for fruits and vegetables |
| US4017503A (en) * | 1975-06-12 | 1977-04-12 | Merck & Co., Inc. | Antifungal 1-substituted benzimidazoles |
| US4017504A (en) * | 1975-06-12 | 1977-04-12 | Merck & Co., Inc. | Antifungal 1-substituted benzimidazoles |
| JPS54127960A (en) * | 1978-03-29 | 1979-10-04 | Toray Silicone Co Ltd | Organopolysiloxane composition |
| GB2176106A (en) * | 1985-06-05 | 1986-12-17 | Uniroyal Ltd | Fungicides comprising carboxamidothiazoles |
| EP0236689A3 (de) * | 1986-01-27 | 1988-04-27 | Shell Internationale Researchmaatschappij B.V. | Fungizide Mittel |
| US5013746A (en) * | 1988-04-08 | 1991-05-07 | Janssen Pharmaceutica N.V. | Imazalil containing synergistic compositions |
| PL219699B1 (pl) * | 2002-03-21 | 2015-06-30 | Basf Ag | Mieszanina grzybobójcza zawierająca protiokonazol i prochloraz, sposób zwalczania szkodliwych grzybów i środek grzybobójczy |
| AU2003297597A1 (en) * | 2002-11-26 | 2004-06-18 | Isis Pharmaceuticals, Inc. | Benzimidazoles and analogs thereof as antibacterials |
| WO2004050035A2 (en) * | 2002-12-03 | 2004-06-17 | Isis Pharmaceuticals, Inc. | Benzimidazoles and analogs thereof as antivirals |
| US20100041682A1 (en) | 2006-09-18 | 2010-02-18 | Langewald Juergen | Ternary Pesticidal Mixtures |
| EP2258177A3 (en) | 2006-12-15 | 2011-11-09 | Rohm and Haas Company | Mixtures comprising 1-methylcyclopropene |
| WO2008095924A2 (de) | 2007-02-06 | 2008-08-14 | Basf Se | Insektizide als safener für fungizide mit phytotoxischer wirkung |
| CL2008001181A1 (es) | 2007-04-23 | 2009-10-23 | Basf Se | Metodo para mejorar la salud de la planta y/o controlar plagas en plantas con al menos una modificacion transgenica relacionada con el aumento del rendimiento que consiste en la aplicacion de una composicion quimica que comprende al menos un ingrediente activo seleccionado de insecticidas, fungicidas o herbicidas. |
| JP2010540495A (ja) | 2007-09-26 | 2010-12-24 | ビーエーエスエフ ソシエタス・ヨーロピア | ボスカリド及びクロロタロニルを含む三成分殺菌組成物 |
| US20090191138A1 (en) * | 2008-01-30 | 2009-07-30 | Mediquest Therapeutics, Inc. | Novel topical formulations for improving the appearance of nails |
| EP2251010A1 (en) | 2009-05-08 | 2010-11-17 | Sygnis Bioscience GmbH & Co. KG | Use of thiabendazole and derivatives thereof for the therapy of neurological conditions |
| WO2011026796A1 (en) | 2009-09-01 | 2011-03-10 | Basf Se | Synergistic fungicidal mixtures comprising lactylates and method for combating phytopathogenic fungi |
| KR20130132942A (ko) | 2010-12-20 | 2013-12-05 | 바스프 에스이 | 피라졸 화합물을 포함하는 살충 활성 혼합물 |
| EP2481284A3 (en) | 2011-01-27 | 2012-10-17 | Basf Se | Pesticidal mixtures |
| WO2012127009A1 (en) | 2011-03-23 | 2012-09-27 | Basf Se | Compositions containing polymeric, ionic compounds comprising imidazolium groups |
| US20140200136A1 (en) | 2011-09-02 | 2014-07-17 | Basf Se | Agricultural mixtures comprising arylquinazolinone compounds |
| CN102388909A (zh) * | 2011-10-13 | 2012-03-28 | 光华化学股份有限公司 | 一种含喹啉铜和噻菌灵的复配农药组合物 |
| ES2660132T3 (es) | 2012-06-20 | 2018-03-20 | Basf Se | Compuestos de pirazol plaguicidas |
| US20150257383A1 (en) | 2012-10-12 | 2015-09-17 | Basf Se | Method for combating phytopathogenic harmful microbes on cultivated plants or plant propagation material |
| JP6576829B2 (ja) | 2012-12-20 | 2019-09-18 | ビーエーエスエフ アグロ ベー.ブイ. | トリアゾール化合物を含む組成物 |
| EP2783569A1 (en) | 2013-03-28 | 2014-10-01 | Basf Se | Compositions comprising a triazole compound |
| EP2835052A1 (en) | 2013-08-07 | 2015-02-11 | Basf Se | Fungicidal mixtures comprising pyrimidine fungicides |
| WO2015036059A1 (en) | 2013-09-16 | 2015-03-19 | Basf Se | Fungicidal pyrimidine compounds |
| CN105722833A (zh) | 2013-09-16 | 2016-06-29 | 巴斯夫欧洲公司 | 杀真菌的嘧啶化合物 |
| EP2979549A1 (en) | 2014-07-31 | 2016-02-03 | Basf Se | Method for improving the health of a plant |
| CN107075712A (zh) | 2014-10-24 | 2017-08-18 | 巴斯夫欧洲公司 | 改变固体颗粒的表面电荷的非两性、可季化和水溶性聚合物 |
| US20180184654A1 (en) | 2015-07-02 | 2018-07-05 | BASF Agro B.V. | Pesticidal Compositions Comprising a Triazole Compound |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US2483392A (en) * | 1949-10-04 | Substituted ethylenes and process | ||
| US2985661A (en) * | 1956-02-06 | 1961-05-23 | American Cyanamid Co | Preparation of 2(omicron-aminophenyl)-benzimidazole |
-
0
- BE BE599143D patent/BE599143A/xx unknown
-
1960
- 1960-01-18 US US2856A patent/US3017415A/en not_active Expired - Lifetime
- 1960-03-17 US US15518A patent/US3055907A/en not_active Expired - Lifetime
- 1960-06-01 DE DEM45481A patent/DE1235321B/de active Pending
- 1960-06-09 GB GB20378/60A patent/GB948635A/en not_active Expired
-
1961
- 1961-01-04 ES ES0263822A patent/ES263822A1/es not_active Expired
- 1961-01-06 FR FR849060A patent/FR1423609A/fr not_active Expired
- 1961-01-17 DK DK19761AA patent/DK107167C/da active
- 1961-01-17 SE SE436/61A patent/SE310883B/xx unknown
- 1961-01-17 CH CH1531665A patent/CH423791A/de unknown
- 1961-01-17 CH CH1531565A patent/CH423790A/de unknown
- 1961-01-17 CH CH1531765A patent/CH423792A/de unknown
- 1961-01-17 CH CH1531865A patent/CH423793A/de unknown
- 1961-01-17 CH CH49061A patent/CH423789A/de unknown
-
1964
- 1964-12-29 OA OA51102A patent/OA00999A/xx unknown
-
1965
- 1965-02-18 CY CY30965A patent/CY309A/xx unknown
- 1965-12-31 MY MY196575A patent/MY6500075A/xx unknown
-
1967
- 1967-08-23 SE SE11797/67A patent/SE320977B/xx unknown
Cited By (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0387941A1 (en) * | 1989-03-15 | 1990-09-19 | Janssen Pharmaceutica N.V. | [5(6)-(benzisoxa-, benzisothia- or indazol-3-yl)-1H-benzimidazol-2-yl] carbamates |
| WO1990010630A1 (en) * | 1989-03-15 | 1990-09-20 | Janssen Pharmaceutica N.V. | [5(6)-(benzisoxa-, benzisothia- or indazol-3-yl)-1h-benzimidazol-2-yl] carbamates |
| WO1994025457A1 (en) * | 1993-04-30 | 1994-11-10 | E.I. Du Pont De Nemours And Company | Process for preparing thiabendazole |
Also Published As
| Publication number | Publication date |
|---|---|
| DK107167C (da) | 1967-05-01 |
| BE599143A (cg-RX-API-DMAC7.html) | |
| US3055907A (en) | 1962-09-25 |
| CH423789A (de) | 1966-11-15 |
| US3017415A (en) | 1962-01-16 |
| CH423792A (de) | 1966-11-15 |
| CY309A (en) | 1965-02-18 |
| CH423790A (de) | 1966-11-15 |
| GB948635A (en) | 1964-02-05 |
| ES263822A1 (es) | 1961-05-16 |
| DE1235321B (de) | 1967-03-02 |
| MY6500075A (en) | 1965-12-31 |
| SE320977B (cg-RX-API-DMAC7.html) | 1970-02-23 |
| CH423791A (de) | 1966-11-15 |
| SE310883B (cg-RX-API-DMAC7.html) | 1969-05-19 |
| OA00999A (fr) | 1968-08-07 |
| CH423793A (de) | 1966-11-15 |
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