FI922903A0 - 4-ACETOXIPIPERIDINE DERIVATIVES, DERAS FRAMSTAELLNINGSFOERFARANDE OCH ANVAENDNING SOM ANTAGONIST FOER MUSKARINA M-3 RECEPTORER. - Google Patents
4-ACETOXIPIPERIDINE DERIVATIVES, DERAS FRAMSTAELLNINGSFOERFARANDE OCH ANVAENDNING SOM ANTAGONIST FOER MUSKARINA M-3 RECEPTORER.Info
- Publication number
- FI922903A0 FI922903A0 FI922903A FI922903A FI922903A0 FI 922903 A0 FI922903 A0 FI 922903A0 FI 922903 A FI922903 A FI 922903A FI 922903 A FI922903 A FI 922903A FI 922903 A0 FI922903 A0 FI 922903A0
- Authority
- FI
- Finland
- Prior art keywords
- receptorer
- muskarina
- acetoxipiperidine
- foer
- antagonist
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/08—Bronchodilators
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D211/40—Oxygen atoms
- C07D211/44—Oxygen atoms attached in position 4
- C07D211/46—Oxygen atoms attached in position 4 having a hydrogen atom as the second substituent in position 4
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB909023023A GB9023023D0 (en) | 1990-10-23 | 1990-10-23 | Pharmaceutical compositions |
PCT/GB1991/001810 WO1992006958A1 (en) | 1990-10-23 | 1991-10-17 | 4-acetoxy-piperidine derivatives, process for their preparation and use as a muscarinic m3-receptor antagonist |
Publications (2)
Publication Number | Publication Date |
---|---|
FI922903A0 true FI922903A0 (en) | 1992-06-22 |
FI922903A FI922903A (en) | 1992-06-22 |
Family
ID=10684199
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FI922903A FI922903A (en) | 1990-10-23 | 1992-06-22 | 4-ACETOXIPIPERIDINE DERIVATIVES, DERAS FRAMSTAELLNINGSFOERFARANDE OCH ANVAENDNING SOM ANTAGONIST FOER MUSKARINA M-3 RECEPTORER. |
Country Status (9)
Country | Link |
---|---|
EP (1) | EP0506903A1 (en) |
JP (1) | JPH05504578A (en) |
AU (1) | AU8714991A (en) |
CA (1) | CA2072598A1 (en) |
FI (1) | FI922903A (en) |
GB (2) | GB9023023D0 (en) |
PT (1) | PT99299A (en) |
WO (1) | WO1992006958A1 (en) |
ZA (1) | ZA918381B (en) |
Families Citing this family (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AU7545894A (en) * | 1993-09-02 | 1995-03-22 | Yamanouchi Pharmaceutical Co., Ltd. | Carbamate derivative and medicine containing the same |
NO2005012I1 (en) * | 1994-12-28 | 2005-06-06 | Debio Rech Pharma Sa | Triptorelin and pharmaceutically acceptable salts thereof |
CA2179574A1 (en) * | 1995-06-26 | 1996-12-27 | Tomomi Okada | Substituted piperidine derivative and medicine comprising the same |
PE92198A1 (en) * | 1996-08-01 | 1999-01-09 | Banyu Pharma Co Ltd | DERIVATIVES OF FLUORINE-CONTAINED 1,4-PIPERIDINE |
PE20050231A1 (en) * | 2003-06-24 | 2005-05-20 | Novartis Ag | DERIVATIVES OF PIPERIDINIUM AND PYRROLIDINIUM AS ANTAGONISTS OF THE MUSCARINIC M3 RECEPTOR |
GB0428418D0 (en) | 2004-12-24 | 2005-02-02 | Novartis Ag | Organic compounds |
EP3233799B1 (en) * | 2014-12-19 | 2021-05-19 | The Broad Institute, Inc. | Dopamine d2 receptor ligands |
WO2016100940A1 (en) | 2014-12-19 | 2016-06-23 | The Broad Institute, Inc. | Dopamine d2 receptor ligands |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
BE792043A (en) * | 1971-11-30 | 1973-05-29 | Ciba Geigy | PIPERIDINE DERIVATIVES USED TO STABILIZE ORGANIC MATERIALS |
IT1231238B (en) * | 1987-09-21 | 1991-11-26 | Angeli Inst Spa | AMIDIDIC DERIVATIVES |
-
1990
- 1990-10-23 GB GB909023023A patent/GB9023023D0/en active Pending
-
1991
- 1991-10-17 JP JP3516505A patent/JPH05504578A/en active Pending
- 1991-10-17 GB GB9122083A patent/GB2249093A/en not_active Withdrawn
- 1991-10-17 WO PCT/GB1991/001810 patent/WO1992006958A1/en not_active Application Discontinuation
- 1991-10-17 CA CA002072598A patent/CA2072598A1/en not_active Abandoned
- 1991-10-17 AU AU87149/91A patent/AU8714991A/en not_active Abandoned
- 1991-10-17 EP EP91917741A patent/EP0506903A1/en not_active Withdrawn
- 1991-10-21 ZA ZA918381A patent/ZA918381B/en unknown
- 1991-10-22 PT PT99299A patent/PT99299A/en not_active Application Discontinuation
-
1992
- 1992-06-22 FI FI922903A patent/FI922903A/en not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
WO1992006958A1 (en) | 1992-04-30 |
CA2072598A1 (en) | 1992-04-24 |
GB9023023D0 (en) | 1990-12-05 |
ZA918381B (en) | 1993-04-21 |
AU8714991A (en) | 1992-05-20 |
GB9122083D0 (en) | 1991-11-27 |
PT99299A (en) | 1992-08-31 |
EP0506903A1 (en) | 1992-10-07 |
FI922903A (en) | 1992-06-22 |
GB2249093A (en) | 1992-04-29 |
JPH05504578A (en) | 1993-07-15 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FD | Application lapsed |