FI914556A0 - 4- ELLER 5-SUBSTITUERADE PYRIDINER-2-KARBOXYLSYROR, FOERFARANDE FOER DERAS FRAMSTAELLNING OCH DERAS ANVAENDNING SOM LAEKEMEDEL. - Google Patents
4- ELLER 5-SUBSTITUERADE PYRIDINER-2-KARBOXYLSYROR, FOERFARANDE FOER DERAS FRAMSTAELLNING OCH DERAS ANVAENDNING SOM LAEKEMEDEL.Info
- Publication number
- FI914556A0 FI914556A0 FI914556A FI914556A FI914556A0 FI 914556 A0 FI914556 A0 FI 914556A0 FI 914556 A FI914556 A FI 914556A FI 914556 A FI914556 A FI 914556A FI 914556 A0 FI914556 A0 FI 914556A0
- Authority
- FI
- Finland
- Prior art keywords
- deras
- karboxylsyror
- pyridiner
- substituerade
- eller
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/62—Oxygen or sulfur atoms
- C07D213/63—One oxygen atom
- C07D213/64—One oxygen atom attached in position 2 or 6
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D213/81—Amides; Imides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D213/81—Amides; Imides
- C07D213/82—Amides; Imides in position 3
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Immunology (AREA)
- Transplantation (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Pyridine Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE4031000A DE4031000A1 (en) | 1990-10-01 | 1990-10-01 | 4- OR 5-SUBSTITUTED PYRIDINE-2-CARBONIC ACIDS, METHOD FOR THE PRODUCTION THEREOF AND THEIR USE AS A MEDICINAL PRODUCT |
Publications (2)
Publication Number | Publication Date |
---|---|
FI914556A0 true FI914556A0 (en) | 1991-09-27 |
FI914556A FI914556A (en) | 1992-04-02 |
Family
ID=6415345
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FI914556A FI914556A (en) | 1990-10-01 | 1991-09-27 | 4- ELLER 5-SUBSTITUERADE PYRIDINER-2-KARBOXYLSYROR, FOERFARANDE FOER DERAS FRAMSTAELLNING OCH DERAS ANVAENDNING SOM LAEKEMEDEL. |
Country Status (20)
Country | Link |
---|---|
EP (1) | EP0479177A3 (en) |
JP (1) | JPH04247070A (en) |
KR (1) | KR920007999A (en) |
CN (1) | CN1060655A (en) |
AU (1) | AU8485291A (en) |
BG (1) | BG95162A (en) |
BR (1) | BR9104205A (en) |
CA (1) | CA2052510A1 (en) |
CS (1) | CS299191A3 (en) |
DE (1) | DE4031000A1 (en) |
FI (1) | FI914556A (en) |
HU (1) | HUT59103A (en) |
IE (1) | IE913435A1 (en) |
IL (1) | IL99605A0 (en) |
MA (1) | MA22313A1 (en) |
MX (1) | MX9101347A (en) |
NO (1) | NO913834L (en) |
PL (1) | PL291881A1 (en) |
PT (1) | PT99132A (en) |
ZA (1) | ZA917805B (en) |
Families Citing this family (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0617020A1 (en) * | 1992-04-02 | 1994-09-28 | Shudo, Koichi, Prof. Dr. | Carboxylic acid derivatives having retinoic acid-like activity |
DE4233124A1 (en) * | 1992-10-02 | 1994-04-07 | Hoechst Ag | Acylsulfonamido and sulfonamidopyridine-2-carboxylic acid esters and their pyridine N-oxides, processes for their preparation and their use as medicaments |
EP1814551A2 (en) | 2004-09-20 | 2007-08-08 | Xenon Pharmaceuticals Inc. | Pyridazine derivatives for inhibiting human stearoyl-coa-desaturase |
TW200626139A (en) | 2004-09-20 | 2006-08-01 | Xenon Pharmaceuticals Inc | Heterocyclic derivatives and their use as therapeutic agents |
BRPI0515488A (en) | 2004-09-20 | 2008-07-29 | Xenon Pharmaceuticals Inc | heterocyclic derivatives and their use as therapeutic agents |
TW200626572A (en) | 2004-09-20 | 2006-08-01 | Xenon Pharmaceuticals Inc | Heterocyclic derivatives and their use as therapeutic agents |
BRPI0515483A (en) | 2004-09-20 | 2008-07-22 | Xenon Pharmaceuticals Inc | heterocyclic derivatives for the treatment of stearoyl coa desaturase mediated diseases |
WO2006034440A2 (en) | 2004-09-20 | 2006-03-30 | Xenon Pharmaceuticals Inc. | Heterocyclic derivatives and their use as stearoyl-coa desaturase inhibitors |
MX2007003332A (en) | 2004-09-20 | 2007-06-05 | Xenon Pharmaceuticals Inc | Heterocyclic derivatives and their use as stearoyl-coa desaturase inhibitors. |
EP2540296A1 (en) | 2005-06-03 | 2013-01-02 | Xenon Pharmaceuticals Inc. | Arminothiazole derivatives as human stearoyl-coa desaturase inhibitors |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE3703959A1 (en) * | 1987-02-10 | 1988-08-18 | Hoechst Ag | PYRIDINE-2,4- AND 2,5-DICARBONIC ACID AMIDES, METHOD FOR THE PRODUCTION THEREOF, USE OF THE SAME AND MEDICINAL PRODUCTS BASED ON THESE COMPOUNDS |
DE3703962A1 (en) * | 1987-02-10 | 1988-08-18 | Hoechst Ag | PYRIDINE-2,4- AND 2,5-DICARBONIC ACID DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF, USE OF THE SAME AND MEDICINAL PRODUCTS BASED ON THESE COMPOUNDS |
ATE113036T1 (en) * | 1988-08-04 | 1994-11-15 | Hoechst Ag | IMPROVED PROCESS FOR THE PRODUCTION OF N,N-BIS(ALKOXYALKYL)-PYRIDINE-2,4-DICARBONIC DIAMIDES. |
-
1990
- 1990-10-01 DE DE4031000A patent/DE4031000A1/en not_active Withdrawn
-
1991
- 1991-09-24 BG BG095162A patent/BG95162A/en unknown
- 1991-09-27 IL IL99605A patent/IL99605A0/en unknown
- 1991-09-27 FI FI914556A patent/FI914556A/en unknown
- 1991-09-30 KR KR1019910017066A patent/KR920007999A/en not_active Application Discontinuation
- 1991-09-30 IE IE343591A patent/IE913435A1/en not_active Application Discontinuation
- 1991-09-30 ZA ZA917805A patent/ZA917805B/en unknown
- 1991-09-30 NO NO91913834A patent/NO913834L/en unknown
- 1991-09-30 PL PL29188191A patent/PL291881A1/en unknown
- 1991-09-30 EP EP19910116632 patent/EP0479177A3/en not_active Withdrawn
- 1991-09-30 BR BR919104205A patent/BR9104205A/en unknown
- 1991-09-30 MX MX9101347A patent/MX9101347A/en unknown
- 1991-09-30 JP JP3250719A patent/JPH04247070A/en active Pending
- 1991-09-30 HU HU913119A patent/HUT59103A/en unknown
- 1991-09-30 CA CA002052510A patent/CA2052510A1/en not_active Abandoned
- 1991-09-30 CN CN91109400A patent/CN1060655A/en active Pending
- 1991-09-30 CS CS912991A patent/CS299191A3/en unknown
- 1991-09-30 AU AU84852/91A patent/AU8485291A/en not_active Abandoned
- 1991-10-01 PT PT99132A patent/PT99132A/en not_active Application Discontinuation
- 1991-10-01 MA MA22593A patent/MA22313A1/en unknown
Also Published As
Publication number | Publication date |
---|---|
BG95162A (en) | 1993-12-24 |
MX9101347A (en) | 1992-06-05 |
HUT59103A (en) | 1992-04-28 |
DE4031000A1 (en) | 1992-04-09 |
HU913119D0 (en) | 1992-01-28 |
ZA917805B (en) | 1992-05-27 |
AU8485291A (en) | 1992-04-02 |
PL291881A1 (en) | 1992-06-15 |
CS299191A3 (en) | 1992-06-17 |
NO913834L (en) | 1992-04-02 |
CN1060655A (en) | 1992-04-29 |
EP0479177A3 (en) | 1992-10-28 |
NO913834D0 (en) | 1991-09-30 |
IE913435A1 (en) | 1992-04-08 |
PT99132A (en) | 1992-09-30 |
EP0479177A2 (en) | 1992-04-08 |
MA22313A1 (en) | 1992-07-01 |
JPH04247070A (en) | 1992-09-03 |
CA2052510A1 (en) | 1992-04-02 |
FI914556A (en) | 1992-04-02 |
KR920007999A (en) | 1992-05-27 |
BR9104205A (en) | 1992-06-02 |
IL99605A0 (en) | 1992-08-18 |
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