FI894139A0 - Antibiotiska sulfonylaminokarbonyl aktiverade b-laktamer. - Google Patents

Antibiotiska sulfonylaminokarbonyl aktiverade b-laktamer.

Info

Publication number
FI894139A0
FI894139A0 FI894139A FI894139A FI894139A0 FI 894139 A0 FI894139 A0 FI 894139A0 FI 894139 A FI894139 A FI 894139A FI 894139 A FI894139 A FI 894139A FI 894139 A0 FI894139 A0 FI 894139A0
Authority
FI
Finland
Prior art keywords
sulphonylaminocarbonyl
activatory
antibiotic
lactose
sulphonylaminocarbonyl activatory
Prior art date
Application number
FI894139A
Other languages
English (en)
Other versions
FI894139A (fi
Inventor
Michael R Barbachyn
Steven J Brickner
Richard C Thomas
Original Assignee
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Upjohn Co filed Critical Upjohn Co
Publication of FI894139A0 publication Critical patent/FI894139A0/fi
Publication of FI894139A publication Critical patent/FI894139A/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Cephalosporin Compounds (AREA)
FI894139A 1987-03-03 1989-09-01 Antibiotiska sulfonylaminokarbonyl aktiverade b-laktamer. FI894139A (fi)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
US2109487A 1987-03-03 1987-03-03
US2340387A 1987-03-09 1987-03-09
US2494887A 1987-03-12 1987-03-12
US2692587A 1987-03-17 1987-03-17
US6543187A 1987-06-23 1987-06-23
PCT/US1988/000404 WO1988006588A1 (en) 1987-03-03 1988-02-19 ANTIBIOTIC SULFONYLAMINOCARBONYL ACTIVATED beta-LACTAMS

Publications (2)

Publication Number Publication Date
FI894139A0 true FI894139A0 (fi) 1989-09-01
FI894139A FI894139A (fi) 1989-09-01

Family

ID=27533899

Family Applications (1)

Application Number Title Priority Date Filing Date
FI894139A FI894139A (fi) 1987-03-03 1989-09-01 Antibiotiska sulfonylaminokarbonyl aktiverade b-laktamer.

Country Status (8)

Country Link
US (1) US4975538A (fi)
EP (2) EP0281289A1 (fi)
JP (1) JPH02502281A (fi)
KR (1) KR890700589A (fi)
AU (1) AU599766B2 (fi)
CA (1) CA1317298C (fi)
FI (1) FI894139A (fi)
WO (1) WO1988006588A1 (fi)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1988006156A1 (en) * 1987-02-11 1988-08-25 The Upjohn Company NOVEL N-1 SUBSTITUTED beta-LACTAMS AS ANTIBIOTICS
EP1049682A1 (en) 1998-01-23 2000-11-08 Versicor, Inc. Oxazolidinone combinatorial libraries, compositions and methods of preparation
US7002020B1 (en) 1998-01-23 2006-02-21 Pharmacia & Upjohn Company Oxazolidinone combinatorial libraries, compositions and methods of preparation
US6562844B2 (en) 1998-01-23 2003-05-13 Pharmacia & Upjohn Company Oxazolidinone combinatorial libraries, compositions and methods of preparation
JP2002174928A (ja) * 2000-09-26 2002-06-21 Ricoh Co Ltd 画像形成装置及び画像形成方法
TW200510425A (en) 2003-08-13 2005-03-16 Japan Tobacco Inc Nitrogen-containing fused ring compound and use thereof as HIV integrase inhibitor
US7511159B2 (en) * 2003-12-25 2009-03-31 Ono Pharmaceutical Co., Ltd. Azetidine ring compounds and drugs comprising the same
CA2488034C (en) * 2004-11-19 2009-10-06 Apotex Inc. Process for the manufacture of 3-hydroxy-n-alkyl-1-cycloalkyl-6-alkyl-4-oxo-1,4-dihydropyridine-2-carboxamide and its related analogues
EP2320909B8 (en) * 2008-07-25 2016-03-30 VIIV Healthcare Company Chemical compounds
EP2379546A1 (en) * 2008-12-19 2011-10-26 Pfizer Inc. Monocarbams
CA2872376A1 (en) 2012-05-03 2013-11-07 Bayer Cropscience Ag 6-pyridone-2-carbamoyl-azoles and their use as herbicides
BR112020004036A2 (pt) 2017-08-31 2020-09-01 Hokko Chemical Industry Co., Ltd derivado de 1-(n,n-carbamoíla dissubstituída) 4-(sulfonila substituída) triazolin-5-ona, derivado de 4-(n,n-carbamoíla dissubstituída) 1-(sulfonila substituída) triazolin-5-ona e herbicida contendo os mesmos como ingrediente ativo
WO2020132820A1 (zh) * 2018-12-24 2020-07-02 广东莱佛士制药技术有限公司 一种3-(苄氧基)-4-氧代-4h-吡喃-2-羧酸的合成方法
CN109438405B (zh) * 2018-12-24 2023-04-07 广东莱佛士制药技术有限公司 一种3-(苄氧基)-4-氧代-4h-吡喃-2-羧酸的合成方法

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE96297C (fi) *
WO1982001873A1 (en) * 1980-12-05 1982-06-10 Takeda Chemical Industries Ltd 1-sulfo-2-oxoazetidine derivatives and process for their preparation
MX7096E (es) * 1980-12-05 1987-06-19 Takeda Chemical Industries Ltd Metodo para preparacion de derivados de 2-oxoazetidina
US4587047A (en) * 1981-04-09 1986-05-06 E. R. Squibb & Sons, Inc. 2-oxo-1-[[(substituted sulfonyl)amino]-carbonyl]azetidines
NZ199981A (en) * 1981-04-09 1985-08-16 Squibb & Sons Inc 2-oxo-1-(((substituted sulphonyl)amino)carbonyl)azetidines
EP0076758B1 (en) * 1981-10-05 1987-01-07 E.R. Squibb & Sons, Inc. 4-ether derivatives of 2-azetidinone-1-sulfonic acids
US4670553A (en) * 1982-01-04 1987-06-02 E. R. Squibb & Sons, Inc. 2-oxo-1-(aminocarbonylaminosulfonyl-aminocarbonyl)azetidines
CA1272726C (en) * 1982-01-04 1990-08-14 2-oxo-1-(aminocarbonylaminosulfonyl- aminocarbonyl)azetidines
EG18314A (en) * 1985-09-26 1993-02-28 Squibb & Sons Inc Process for preparing of 2-oxo-1((substituted sulfonyl)amino)carbonyl)-azitidines
AU7541487A (en) * 1986-05-23 1987-12-22 Upjohn Company, The N-1 substituted sulfonylaminocarbonyl, c-4 substituted monobactams
US4801705A (en) * 1986-06-23 1989-01-31 E. R. Squibb & Sons, Inc. 2-oxo-1-(((substituted sulfonyl)amino)-carbonyl)azetidines
WO1988006587A1 (en) * 1987-02-27 1988-09-07 The Upjohn Company ANTIBIOTIC beta-LACTAMS CONTAINING A PYRIDONE CARBOXYLIC ACID OR ACID DERIVATIVE

Also Published As

Publication number Publication date
KR890700589A (ko) 1989-04-26
AU1345688A (en) 1988-09-26
AU599766B2 (en) 1990-07-26
CA1317298C (en) 1993-05-04
WO1988006588A1 (en) 1988-09-07
FI894139A (fi) 1989-09-01
EP0281289A1 (en) 1988-09-07
EP0352269A1 (en) 1990-01-31
US4975538A (en) 1990-12-04
JPH02502281A (ja) 1990-07-26

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Legal Events

Date Code Title Description
FA Application withdrawn

Owner name: THE UPJOHN COMPANY