FI882443A - SUBSTITUERADE VINYLKEFALOSPORINER, FOERFARANDE FOER DERAS FRAMSTAELLNING OCH DERAS ANVAENDNING SOM LAEKEMEDEL. - Google Patents

SUBSTITUERADE VINYLKEFALOSPORINER, FOERFARANDE FOER DERAS FRAMSTAELLNING OCH DERAS ANVAENDNING SOM LAEKEMEDEL. Download PDF

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Publication number
FI882443A
FI882443A FI882443A FI882443A FI882443A FI 882443 A FI882443 A FI 882443A FI 882443 A FI882443 A FI 882443A FI 882443 A FI882443 A FI 882443A FI 882443 A FI882443 A FI 882443A
Authority
FI
Finland
Prior art keywords
deras
vinylkefalosporiner
substituerade
foerfarande foer
framstaellning och
Prior art date
Application number
FI882443A
Other languages
Finnish (fi)
Other versions
FI882443A0 (en
Inventor
Gunter Schmidt
Karl Georg Metzger
Hans-Joachim Zeiler
Rainer Endermann
Ingo Haller
Original Assignee
Bayer Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Ag filed Critical Bayer Ag
Publication of FI882443A0 publication Critical patent/FI882443A0/en
Publication of FI882443A publication Critical patent/FI882443A/en

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D501/00Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/207-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • AHUMAN NECESSITIES
    • A23FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
    • A23KFODDER
    • A23K20/00Accessory food factors for animal feeding-stuffs
    • A23K20/10Organic substances
    • A23K20/195Antibiotics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D501/00Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/207-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • C07D501/227-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with radicals containing only hydrogen and carbon atoms, attached in position 3
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D501/00Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/207-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • C07D501/247-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Polymers & Plastics (AREA)
  • Oncology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Food Science & Technology (AREA)
  • Zoology (AREA)
  • Communicable Diseases (AREA)
  • Animal Husbandry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
FI882443A 1987-05-26 1988-05-24 SUBSTITUERADE VINYLKEFALOSPORINER, FOERFARANDE FOER DERAS FRAMSTAELLNING OCH DERAS ANVAENDNING SOM LAEKEMEDEL. FI882443A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE3717664 1987-05-26
DE19873734004 DE3734004A1 (en) 1987-05-26 1987-10-08 SUBSTITUTED VINYLCEPHALOSPORINE, METHOD FOR THE PRODUCTION THEREOF AND THEIR USE AS A MEDICINAL PRODUCT

Publications (2)

Publication Number Publication Date
FI882443A0 FI882443A0 (en) 1988-05-24
FI882443A true FI882443A (en) 1988-11-27

Family

ID=25856024

Family Applications (1)

Application Number Title Priority Date Filing Date
FI882443A FI882443A (en) 1987-05-26 1988-05-24 SUBSTITUERADE VINYLKEFALOSPORINER, FOERFARANDE FOER DERAS FRAMSTAELLNING OCH DERAS ANVAENDNING SOM LAEKEMEDEL.

Country Status (14)

Country Link
EP (1) EP0292808B1 (en)
JP (1) JPH0645627B2 (en)
KR (1) KR880013950A (en)
CN (1) CN88103202A (en)
AU (1) AU1630188A (en)
CA (1) CA1340154C (en)
DE (2) DE3734004A1 (en)
DK (1) DK284688A (en)
ES (1) ES2062997T3 (en)
FI (1) FI882443A (en)
HU (1) HU205937B (en)
IL (1) IL86478A (en)
NO (1) NO170020C (en)
PT (1) PT87564B (en)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3734005A1 (en) * 1987-05-26 1988-12-15 Bayer Ag SUBSTITUTED VINYLCEPHALOSPORINS, THE METHOD OF MANUFACTURING THEIR PRODUCTS AND THEIR USE AS A MEDICINAL PRODUCT
DE3933934A1 (en) * 1989-10-03 1991-04-11 Bayer Ag METHOD FOR PRODUCING 7-AMINO-3 - ((Z) -1-PROPEN-1-YL) -3-CEPHEM-4-CARBONIC ACID
DK0503453T3 (en) 1991-03-08 2001-07-16 Biochemie Gmbh Process for preparing cephalosporins and intermediates in this process
US6248881B1 (en) 1991-03-08 2001-06-19 Biochemie Gmbh Intermediates and process for the production of 3-vinyl cephalosporins
KR930007261B1 (en) * 1991-04-19 1993-08-04 한국과학기술연구원 Cephem-4-carboxylic acid derivatives
JP3224279B2 (en) * 1992-07-27 2001-10-29 大塚化学株式会社 Method for producing cefm compound
KR20000002217A (en) * 1998-06-18 2000-01-15 김종인 Novel cephalosporin antibiotics and manufacturing method of it
EP2209474A4 (en) 2007-10-09 2013-07-24 Sopharmia Inc Broad spectrum beta-lactamase inhibitors
US9975905B2 (en) 2013-03-12 2018-05-22 Gladius Pharmaceuticals Corporation Derivatized 3-styryl-cephalosporins

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3769277A (en) * 1970-01-23 1973-10-30 Glaxo Lab Ltd Preparation of delta3-4 carboxy cephalosporins having a 3-vinyl or substituted 3-vinyl group
US4255423A (en) * 1977-07-27 1981-03-10 Merck & Co., Inc. Cephalosporin compounds
US4390693A (en) * 1977-07-27 1983-06-28 Merck & Co., Inc. Cephalosporin compounds
US4520022A (en) * 1983-01-28 1985-05-28 Bristol-Myers Company Substituted vinyl cephalosporins
GB8406231D0 (en) * 1984-03-09 1984-04-11 Fujisawa Pharmaceutical Co Cephem compounds
DE3508258A1 (en) * 1985-03-08 1986-09-18 Bayer Ag, 5090 Leverkusen SS LACTAMANTIBIOTICS, METHOD FOR THE PRODUCTION AND THEIR USE AS AND IN MEDICINAL PRODUCTS
JPS63126023A (en) * 1986-11-14 1988-05-30 Fujitsu Ltd Display device
DE3734005A1 (en) * 1987-05-26 1988-12-15 Bayer Ag SUBSTITUTED VINYLCEPHALOSPORINS, THE METHOD OF MANUFACTURING THEIR PRODUCTS AND THEIR USE AS A MEDICINAL PRODUCT

Also Published As

Publication number Publication date
FI882443A0 (en) 1988-05-24
DK284688D0 (en) 1988-05-25
CA1340154C (en) 1998-12-01
ES2062997T3 (en) 1995-01-01
DE3888018D1 (en) 1994-04-07
DE3734004A1 (en) 1988-12-15
EP0292808A3 (en) 1990-09-19
HUT47940A (en) 1989-04-28
PT87564A (en) 1989-05-31
JPH0645627B2 (en) 1994-06-15
HU205937B (en) 1992-07-28
EP0292808A2 (en) 1988-11-30
CN88103202A (en) 1988-12-21
AU1630188A (en) 1988-12-01
EP0292808B1 (en) 1994-03-02
NO882112L (en) 1988-11-28
KR880013950A (en) 1988-12-22
IL86478A (en) 1993-02-21
NO882112D0 (en) 1988-05-13
NO170020C (en) 1992-09-02
PT87564B (en) 1992-09-30
IL86478A0 (en) 1988-11-15
NO170020B (en) 1992-05-25
JPS63307885A (en) 1988-12-15
DK284688A (en) 1988-11-27

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