FI860847A - Foerfarande foer framstaellning av aktiva 3-aryl-oxiazetidinkarboxamider. - Google Patents

Foerfarande foer framstaellning av aktiva 3-aryl-oxiazetidinkarboxamider. Download PDF

Info

Publication number
FI860847A
FI860847A FI860847A FI860847A FI860847A FI 860847 A FI860847 A FI 860847A FI 860847 A FI860847 A FI 860847A FI 860847 A FI860847 A FI 860847A FI 860847 A FI860847 A FI 860847A
Authority
FI
Finland
Prior art keywords
oxiazetidinkarboxamider
aryl
active
frequency fragmentation
fragmentation
Prior art date
Application number
FI860847A
Other languages
English (en)
Other versions
FI860847A0 (fi
FI87559B (fi
FI87559C (fi
Inventor
Jr Chandler Roy Taylor
Jr Albert Duncan Cale
David Norseen Johnson
Jr Harold Fisher Stauffer
Original Assignee
Robins Co Inc A H
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Robins Co Inc A H filed Critical Robins Co Inc A H
Publication of FI860847A0 publication Critical patent/FI860847A0/fi
Publication of FI860847A publication Critical patent/FI860847A/fi
Publication of FI87559B publication Critical patent/FI87559B/fi
Application granted granted Critical
Publication of FI87559C publication Critical patent/FI87559C/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4151,2-Diazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D205/00Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/04Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D249/00Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/081,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
FI860847A 1985-02-28 1986-02-27 Foerfarande foer framstaellning av aktiva 3-fenyloxiazetidinkarboxamider FI87559C (fi)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US70662185A 1985-02-28 1985-02-28
US70663285A 1985-02-28 1985-02-28
US70663285 1985-02-28
US70662185 1985-02-28

Publications (4)

Publication Number Publication Date
FI860847A0 FI860847A0 (fi) 1986-02-27
FI860847A true FI860847A (fi) 1986-08-29
FI87559B FI87559B (fi) 1992-10-15
FI87559C FI87559C (fi) 1993-01-25

Family

ID=27107712

Family Applications (1)

Application Number Title Priority Date Filing Date
FI860847A FI87559C (fi) 1985-02-28 1986-02-27 Foerfarande foer framstaellning av aktiva 3-fenyloxiazetidinkarboxamider

Country Status (7)

Country Link
EP (1) EP0194112B1 (fi)
CY (1) CY1724A (fi)
DE (1) DE3671369D1 (fi)
FI (1) FI87559C (fi)
HK (1) HK83893A (fi)
IE (1) IE58943B1 (fi)
SG (1) SG50893G (fi)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5095014A (en) * 1990-12-07 1992-03-10 A. H. Robins Company, Incorporated 3-(2-chloro-4-(trifluoromethyl)phenoxy)-1-azetidine carboxamides having anticonvulsant activity
US5183903A (en) * 1991-11-26 1993-02-02 A. H. Robins Company, Incorporated Urea fusion process for the synthesis of 3-phenoxy-1-azetidinecarboxamides
US6403574B1 (en) 1998-01-23 2002-06-11 Vernalis Research Limited Azetidinecarboxamide derivatives for treating CNS disorders
DE69902142T2 (de) * 1998-01-23 2003-01-09 Vernalis Research Ltd., Winnersh Azetidincarboxamidderivate zur behandlung von zns-erkrankungen
GB9801501D0 (en) * 1998-01-23 1998-03-18 Cerebrus Ltd Chemical compounds - II
GB9917386D0 (en) * 1999-07-23 1999-09-22 Cerebrus Ltd Chemical compounds-II
GB9917385D0 (en) * 1999-07-23 1999-09-22 Cerebrus Ltd Chemical compounds-I
WO2011058766A1 (en) * 2009-11-16 2011-05-19 Raqualia Pharma Inc. Aryl carboxamide derivatives as ttx-s blockers
JOP20190072A1 (ar) 2016-10-13 2019-04-07 Glaxosmithkline Ip Dev Ltd مشتقات 1، 3 سيكلوبوتان ثنائي الاستبدال أو آزيتيدين كمثبطات للإنزيم المخلق للبروستاجلاندين d المكون للدم

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4226861A (en) * 1978-04-18 1980-10-07 A. H. Robins Company, Inc. N-Lower-alkyl 3-phenoxy-1-azetidinecarboxamides
IL68699A (en) * 1982-08-19 1986-08-31 Robins Co Inc A H 3-phenoxy-1-azetidine-carboxamides,their preparation and pharmaceutical compositions containing them
US4505907A (en) * 1982-09-02 1985-03-19 A. H. Robins Company, Inc. N-Formyl and N-hydroxymethyl-3-phenoxy-1-azetidinecarboxamides

Also Published As

Publication number Publication date
FI860847A0 (fi) 1986-02-27
IE58943B1 (en) 1993-12-01
HK83893A (en) 1993-08-20
FI87559B (fi) 1992-10-15
FI87559C (fi) 1993-01-25
IE860522L (en) 1986-08-28
CY1724A (en) 1994-05-06
DE3671369D1 (de) 1990-06-28
SG50893G (en) 1993-07-09
EP0194112A1 (en) 1986-09-10
EP0194112B1 (en) 1990-05-23

Similar Documents

Publication Publication Date Title
NO862797L (no) Fremstilling av alumoxaner.
DE3673176D1 (de) Doppelfrequenzantennensystem.
FI872367A0 (fi) Foerfarande foer framstaellning av vattenhaltiga n-metylmorfolin n-oxidloesningar.
NO167119C (no) Avstandsdupleksert antenne av firestraalers typen.
FI860847A0 (fi) Foerfarande foer framstaellning av aktiva 3-aryl-oxiazetidinkarboxamider.
DE3683660D1 (de) Herstellung von halogenierten benzolen.
FI882265A (fi) Foerfarande foer bestaemning av fruktosamin.
KR860012498U (ko) 고주파 발진기
FI853938A0 (fi) Anordning foer profilmaetning av raelshjul.
DK405887D0 (da) Vaevplasminogenaktivatorholdig kombination
FI851068L (fi) Foerfarande foer framstaellning av 2- oxindol-1-karboxamider och deras mellanprodukter.
FI860598A (fi) Foerfarande foer framstaellning av arylglycidyletrar och 3-substituerade 1-alkylamino-2-propanoler.
NO863434L (no) Fremgangsmaate for fremstilling av metylendioksyfenantren- og stilbenderivater.
FI852976L (fi) Foerfarande foer framstaellning av angiotensin-ii-analoger, vilka aer susbtituerade i 1-,5- och 8-positionen.
DE3587341D1 (de) Epoxidation von propylen.
FI863883A0 (fi) Anordning foer tillslutning av flaskhals.
FI862965A0 (fi) Foerfarande foer framstaellning av kef-3-em-4-karboxylsyraderivat.
FI874471A0 (fi) Foerfarande foer framstaellning av azetidinoner.
FI904082A0 (fi) Foerfarande foer framstaellning av n-heterocyklyl-4-piperidinaminer.
FI920227A0 (fi) Foerfarande foer framstaellning av 4-demetoxi-4-aminoantracykliner.
FI864790A (fi) Foerfarande foer framstaellning av 5-klor- och 5-brom-2-hydroxinikotinsyror.
NO874967L (no) Panservegg av sÿkalt aktivt panser.
FI850412A0 (fi) Foerfarande foer framstaellning av 4-keto -9-metylfenazin.
NO872970L (no) Reduksjon av marin biogroing.
NO880377L (no) Q-omvekslet laserresonator av enhetlig konstruksjon.

Legal Events

Date Code Title Description
MM Patent lapsed
MM Patent lapsed

Owner name: A.H. ROBINS COMPANY, INCORPORATED