FI56843B - FOERFARANDE FOER FRAMSTAELLNING AV ANTIBAKTERIELLA 7- (ALPHA-AMINO-β-HYDROXYPHENYLACETAMIDO) -3-HETEROCYCLIC THIOMETHYLPHALOSPORINER - Google Patents

FOERFARANDE FOER FRAMSTAELLNING AV ANTIBAKTERIELLA 7- (ALPHA-AMINO-β-HYDROXYPHENYLACETAMIDO) -3-HETEROCYCLIC THIOMETHYLPHALOSPORINER

Info

Publication number
FI56843B
FI56843B FI1610/73A FI161073A FI56843B FI 56843 B FI56843 B FI 56843B FI 1610/73 A FI1610/73 A FI 1610/73A FI 161073 A FI161073 A FI 161073A FI 56843 B FI56843 B FI 56843B
Authority
FI
Finland
Prior art keywords
thiomethylphalosporiner
antibakteriella
hydroxyphenylacetamido
heterocyclic
alpha
Prior art date
Application number
FI1610/73A
Other languages
Finnish (fi)
Other versions
FI56843C (en
Inventor
George Lawrence Dunn
John Russel Eugene Hoover
Original Assignee
Smith Kline French Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US262903A external-priority patent/US3867380A/en
Priority claimed from US00289499A external-priority patent/US3855213A/en
Application filed by Smith Kline French Lab filed Critical Smith Kline French Lab
Application granted granted Critical
Publication of FI56843B publication Critical patent/FI56843B/en
Publication of FI56843C publication Critical patent/FI56843C/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D501/00Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/207-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • C07D501/247-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
    • C07D501/36Methylene radicals, substituted by sulfur atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/542Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/545Compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins, cefaclor, or cephalexine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D249/00Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/041,2,3-Triazoles; Hydrogenated 1,2,3-triazoles
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
FI1610/73A 1972-06-14 1973-05-17 FRAMSTARABILATION OF ANTIBACTERIA 7- (ALPHA-AMINO-β-HYDROXYPHENYLACETAMIDO) -3-HETEROCYCLIC THIOMETHYLPHALOSPORINER FI56843C (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US262903A US3867380A (en) 1971-02-18 1972-06-14 3-Heterocyclic thiomethylcephalosporins
US26290372 1972-06-14
US28949972 1972-09-15
US00289499A US3855213A (en) 1971-02-18 1972-09-15 3-heterocyclic thiomethyl-cephalosporins

Publications (2)

Publication Number Publication Date
FI56843B true FI56843B (en) 1979-12-31
FI56843C FI56843C (en) 1980-04-10

Family

ID=26949532

Family Applications (1)

Application Number Title Priority Date Filing Date
FI1610/73A FI56843C (en) 1972-06-14 1973-05-17 FRAMSTARABILATION OF ANTIBACTERIA 7- (ALPHA-AMINO-β-HYDROXYPHENYLACETAMIDO) -3-HETEROCYCLIC THIOMETHYLPHALOSPORINER

Country Status (20)

Country Link
JP (2) JPS5518716B2 (en)
AR (1) AR197237A1 (en)
AT (1) AT324560B (en)
AU (1) AU464107B2 (en)
CA (2) CA1076560A (en)
CH (2) CH586709A5 (en)
DD (1) DD105238A5 (en)
DE (1) DE2316867C2 (en)
DK (1) DK142913B (en)
ES (2) ES412207A1 (en)
FI (1) FI56843C (en)
FR (2) FR2187298B1 (en)
GB (2) GB1363833A (en)
HU (1) HU168689B (en)
IE (2) IE37409B1 (en)
IL (1) IL42126A (en)
NL (2) NL7302817A (en)
PH (1) PH9941A (en)
PL (1) PL91074B1 (en)
SE (2) SE416472B (en)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR780000197B1 (en) * 1972-12-26 1978-05-26 Bristol Myers Co Method for preparing antibacterial agent
NL7401361A (en) * 1973-01-31 1974-08-02
GB1476981A (en) * 1974-06-05 1977-06-16 Bristol Myers Co Substituted penicillanic acids
CA1074784A (en) * 1974-09-06 1980-04-01 Sumitomo Chemical Company N-ACYLAMINO-.alpha.-ARYLACETAMIDO CEPHALOSPORINS
JPS5346995A (en) * 1976-10-12 1978-04-27 Sangyo Kagaku Kenkyu Kyokai Antibacterial agents
NL162387C (en) * 1977-09-06 1980-05-16 Gist Brocades Nv PROCESS FOR PREPARING 6- (D-ALPHA-AMINO-P- HYDROXYPHENYLACETAMIDO) PENICILLANIC ACID.
JPS6010226U (en) * 1983-06-30 1985-01-24 松下電工株式会社 lift device
JPS6182606A (en) * 1984-09-29 1986-04-26 東芝ライテック株式会社 Lift

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA698494B (en) * 1969-02-26 1971-07-28 Lilly Co Eli Sulfur-containing cephalosporing antibiotics
US3641021A (en) * 1969-04-18 1972-02-08 Lilly Co Eli 3 7-(ring-substituted) cephalosporin compounds

Also Published As

Publication number Publication date
GB1358027A (en) 1974-06-26
FR2187299A1 (en) 1974-01-18
IE37499B1 (en) 1977-08-03
CA1076560A (en) 1980-04-29
DE2316866B2 (en) 1976-10-07
PL91074B1 (en) 1977-02-28
JPS4931689A (en) 1974-03-22
IL42126A0 (en) 1973-06-29
CH589093A5 (en) 1977-06-30
JPS5518716B2 (en) 1980-05-21
ES412207A1 (en) 1976-01-01
CH586709A5 (en) 1977-04-15
AU464107B2 (en) 1975-08-14
IL42126A (en) 1975-12-31
IE37409L (en) 1973-12-14
SE404190B (en) 1978-09-25
PH9941A (en) 1976-06-14
IE37409B1 (en) 1977-07-20
HU168689B (en) 1976-06-28
DE2316867C2 (en) 1982-05-19
DK142913C (en) 1981-09-28
FI56843C (en) 1980-04-10
JPS5953274B2 (en) 1984-12-24
JPS4954393A (en) 1974-05-27
NL7305206A (en) 1973-12-18
AT324560B (en) 1975-09-10
NL7302817A (en) 1973-12-18
FR2187298B1 (en) 1976-12-03
FR2187298A1 (en) 1974-01-18
DD105238A5 (en) 1974-04-12
SE416472B (en) 1981-01-05
DE2316866A1 (en) 1974-01-03
ES413501A1 (en) 1976-07-16
DE2316867A1 (en) 1974-01-03
AU5234573A (en) 1974-08-22
IE37499L (en) 1973-12-14
AR197237A1 (en) 1974-03-22
DK142913B (en) 1981-02-23
GB1363833A (en) 1974-08-21
FR2187299B1 (en) 1976-12-03
CA999293A (en) 1976-11-02

Similar Documents

Publication Publication Date Title
FI55045B (en) FOERFARANDE FOER FRAMSTAELLNING AV SMOERJOLJA
FI54609C (en) FOERFARANDE FOER SEPARERING AV MONOSACKARIDER FRAON EN STAERKELSEKONVERSIONSSIRAP
FI54867B (en) FOERFARANDE FOER GJUTNING AV SEGJAERNSTYCKEN
FI55286B (en) FOERFARANDE FOER FRAMSTAELLNING AV KOETTSURROGAT
FI54564C (en) ANORDING FOER SOENDERDELNING AV AVFALLSMATERIAL
FI53844C (en) FOERFARANDE FOER TILLVERKNING AV EN NAOLAD AENDLOES MASKINFILT
FI55326C (en) FOERFARANDE FOER FRAMSTAELLNING AV SKUMKERAMIK
FI54072B (en) CENTRIFUGHJUL FOER CENTRIFUGERING AV SLAMNINGAR
FI54469C (en) FOERFARANDE FOER KOMPOSTERING AV AVLOPPSSLAM
FI53620C (en) BRAENNUGN SPECIELLT FOER BRAENNING AV AVFALL
FI54344C (en) FOERFARANDE FOER REGLERING AV ALKALISK MASSAFRAMSTAELLNING
FI54332B (en) FLUFALDIG ELEKTROLYSCELL FOER FRAMSTAELLNING AV ALKALIHYDROXIDER
FI56843B (en) FOERFARANDE FOER FRAMSTAELLNING AV ANTIBAKTERIELLA 7- (ALPHA-AMINO-β-HYDROXYPHENYLACETAMIDO) -3-HETEROCYCLIC THIOMETHYLPHALOSPORINER
FI53997C (en) ANORDNING FOER BEHANDLING AV FIBERHALTIGA SUSPENSIONER
FI54118C (en) FOERFARANDE FOER FRAMSTAELLNING AV LYSERGINSYRAAMIDER
FI53773B (en) FOERFARANDE FOER FOERLAENGNING AV FAERSKFOERVARINGSTIDEN FOER FAERSKT KOETT
FI53935C (en) FOER FRAMSTAELLNING AV EN FOERPACKNING AV EXPANDERRAT PLASTMATERIAL
FI53471C (en) FOERFARANDE FOER BEHANDLING AV AVFALLSPAPPER
FI54816B (en) FOERFARANDE FOER FOERKRYMPNING AV EN TRIKAOVARA
FI54442B (en) ANORDNING FOER STUMSVETSNING AV CYLINDRISKA TERMOPLASTROER
FI54933C (en) FOERFARANDE FOER AVSKALNING AV GALVANISKT YTFAELLD METALLPLAOT FRAON KATODISK BASPLAOT
FI53857C (en) FOERFARANDE FOER YTLIMNING AV PAPPER
FI55328C (en) FOERFARANDE FOER FRAMSTAELLNING AV TERAPEUTISKT ANVAENDBARA ALICYKLISKA FENOXIKARBOXYLSYRADERIVAT
FI54399C (en) FOERFARINGSSAETT FOER FRAMSTAELLNING AV ROERSKAOLAR
FI54240B (en) FOERFARANDE FOER FRAMSTAELLNING AV EN SPIRALRUTSCH