FI55334C - Foerfarande foer framstaellning av som mellanprodukter vid framstaellning av triazolobensodiazepiner anvaenda 2-alkoxi-5-fenyl-3h-1,4-bensodiazepinderivat - Google Patents

Foerfarande foer framstaellning av som mellanprodukter vid framstaellning av triazolobensodiazepiner anvaenda 2-alkoxi-5-fenyl-3h-1,4-bensodiazepinderivat

Info

Publication number
FI55334C
FI55334C FI896/71A FI89671A FI55334C FI 55334 C FI55334 C FI 55334C FI 896/71 A FI896/71 A FI 896/71A FI 89671 A FI89671 A FI 89671A FI 55334 C FI55334 C FI 55334C
Authority
FI
Finland
Prior art keywords
triazolobensodiazepiner
benzodiazepinderivat
anvaenda
framstation
alcoxy
Prior art date
Application number
FI896/71A
Other languages
English (en)
Finnish (fi)
Other versions
FI55334B (fi
Inventor
Hiroyuki Tawada
Hideaki Natsugari
Kanji Meguro
Yutaka Kuwada
Original Assignee
Takeda Chemical Industries Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from JP2580570A external-priority patent/JPS5010316B1/ja
Priority claimed from JP2580470A external-priority patent/JPS4811112B1/ja
Priority claimed from JP3495070A external-priority patent/JPS5011920B1/ja
Priority claimed from JP4663770A external-priority patent/JPS4924060B1/ja
Application filed by Takeda Chemical Industries Ltd filed Critical Takeda Chemical Industries Ltd
Priority to FI752812A priority Critical patent/FI57938C/fi
Application granted granted Critical
Publication of FI55334B publication Critical patent/FI55334B/fi
Publication of FI55334C publication Critical patent/FI55334C/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D243/00Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/141,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/161,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • C07D243/181,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
    • C07D243/20Nitrogen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
FI896/71A 1970-03-27 1971-03-29 Foerfarande foer framstaellning av som mellanprodukter vid framstaellning av triazolobensodiazepiner anvaenda 2-alkoxi-5-fenyl-3h-1,4-bensodiazepinderivat FI55334C (fi)

Priority Applications (1)

Application Number Priority Date Filing Date Title
FI752812A FI57938C (fi) 1970-03-27 1975-10-09 Foerfarande foer framstaellning av 2-hydrazino-5-fenyl-3h-1;4-benzodiazepinderivat

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
JP2580570A JPS5010316B1 (es) 1970-03-27 1970-03-27
JP2580470A JPS4811112B1 (es) 1970-03-27 1970-03-27
JP3495070A JPS5011920B1 (es) 1970-04-23 1970-04-23
JP4663770A JPS4924060B1 (es) 1970-05-28 1970-05-28

Publications (2)

Publication Number Publication Date
FI55334B FI55334B (fi) 1979-03-30
FI55334C true FI55334C (fi) 1979-07-10

Family

ID=27458380

Family Applications (1)

Application Number Title Priority Date Filing Date
FI896/71A FI55334C (fi) 1970-03-27 1971-03-29 Foerfarande foer framstaellning av som mellanprodukter vid framstaellning av triazolobensodiazepiner anvaenda 2-alkoxi-5-fenyl-3h-1,4-bensodiazepinderivat

Country Status (14)

Country Link
US (1) US4102881A (es)
BE (1) BE764913A (es)
CA (2) CA922317A (es)
CH (1) CH559188A5 (es)
DE (1) DE2114441A1 (es)
DK (1) DK131374B (es)
FI (1) FI55334C (es)
FR (1) FR2085748B1 (es)
GB (1) GB1353486A (es)
NL (1) NL7104132A (es)
NO (1) NO132800C (es)
PH (1) PH9214A (es)
SE (1) SE400968B (es)
YU (1) YU34997B (es)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3709898A (en) * 1971-02-09 1973-01-09 Upjohn Co Process for the production of triazolobenzodiazepines and intermediates
US3681343A (en) * 1971-05-11 1972-08-01 Upjohn Co 6-phenyl-s-triazolo{8 4,3-a{9 {8 1,4{9 {0 benzodiazepines
US4755508A (en) * 1984-06-26 1988-07-05 Merck & Co., Inc. Benzodiazepine analogs and use as antogonists of gastrin and cholecystokinin
US5939414A (en) * 1996-10-31 1999-08-17 Merck & Co., Inc. Benzodiazepine hydrazide derivatives as inhibitors of HIV integrase
EP0949926A4 (en) * 1996-10-31 2001-01-17 Merck & Co Inc BENZODIAZEPINE HYDROCIDE DERIVATIVES AS HIV INTERASE INHIBITORS

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3462418A (en) * 1963-10-29 1969-08-19 Hoffmann La Roche Preparation of 1,4-benzodiazepin-2-one-4-oxide from 2-lower alkoxy-1,4-benzodiazepine-4-oxide
DK120901B (da) * 1965-09-17 1971-08-02 Rexolin Chem Fremgangsmåde til fremstilling af 7-chlor-1,3-dihydro-1-methyl-5-phenyl-2H-1,4-benzodiazepin-2-on.
US3987052A (en) * 1969-03-17 1976-10-19 The Upjohn Company 6-Phenyl-4H-s-triazolo[4,3-a][1,4]benzodiazepines
NO128154B (es) * 1969-07-30 1973-10-08 Grindstedvaerket As
BE755139A (fr) * 1969-08-21 1971-02-22 Upjohn Co Derives de benzodiazepinones, leurs intermediaires, et leur preparatio
FR2022598A1 (en) * 1969-11-04 1970-07-31 Pakeda Chemical Ind Sedative chloro-phenyl-triazolobenzodiazepines

Also Published As

Publication number Publication date
DK131374B (da) 1975-07-07
PH9214A (en) 1975-07-10
DK131374C (es) 1975-12-01
DE2114441A1 (de) 1971-10-14
YU73771A (en) 1979-12-31
FR2085748B1 (es) 1974-08-02
NO132800B (es) 1975-09-29
BE764913A (fr) 1971-08-16
US4102881A (en) 1978-07-25
FI55334B (fi) 1979-03-30
SE400968B (sv) 1978-04-17
CA936864A (en) 1973-11-13
CA922317A (en) 1973-03-06
NO132800C (es) 1976-01-07
GB1353486A (en) 1974-05-15
FR2085748A1 (es) 1971-12-31
YU34997B (en) 1980-06-30
NL7104132A (es) 1971-09-29
CH559188A5 (es) 1975-02-28

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