FI45044C - Menetelmä antibioottisesti aktiivisen 3-substituoidun rifamysiini SV:n johdannaisten valmistamiseksi. - Google Patents

Menetelmä antibioottisesti aktiivisen 3-substituoidun rifamysiini SV:n johdannaisten valmistamiseksi.

Info

Publication number
FI45044C
FI45044C FI651805A FI180565A FI45044C FI 45044 C FI45044 C FI 45044C FI 651805 A FI651805 A FI 651805A FI 180565 A FI180565 A FI 180565A FI 45044 C FI45044 C FI 45044C
Authority
FI
Finland
Prior art keywords
preparation
active derivatives
antibiotically active
rifamycin
substituted
Prior art date
Application number
FI651805A
Other languages
English (en)
Finnish (fi)
Swedish (sv)
Other versions
FI45044B (US20090163788A1-20090625-C00002.png
Inventor
Maggi Nicola
Sensi Piero
Original Assignee
Lepetit Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB30327/64A external-priority patent/GB1109631A/en
Application filed by Lepetit Spa filed Critical Lepetit Spa
Publication of FI45044B publication Critical patent/FI45044B/fi
Application granted granted Critical
Publication of FI45044C publication Critical patent/FI45044C/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D498/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/08Bridged systems
    • AHUMAN NECESSITIES
    • A47FURNITURE; DOMESTIC ARTICLES OR APPLIANCES; COFFEE MILLS; SPICE MILLS; SUCTION CLEANERS IN GENERAL
    • A47FSPECIAL FURNITURE, FITTINGS, OR ACCESSORIES FOR SHOPS, STOREHOUSES, BARS, RESTAURANTS OR THE LIKE; PAYING COUNTERS
    • A47F5/00Show stands, hangers, or shelves characterised by their constructional features
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • GPHYSICS
    • G09EDUCATION; CRYPTOGRAPHY; DISPLAY; ADVERTISING; SEALS
    • G09FDISPLAYING; ADVERTISING; SIGNS; LABELS OR NAME-PLATES; SEALS
    • G09F5/00Means for displaying samples

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Physics & Mathematics (AREA)
  • General Physics & Mathematics (AREA)
  • Engineering & Computer Science (AREA)
  • Theoretical Computer Science (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
FI651805A 1964-07-31 1965-07-27 Menetelmä antibioottisesti aktiivisen 3-substituoidun rifamysiini SV:n johdannaisten valmistamiseksi. FI45044C (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB30327/64A GB1109631A (en) 1964-07-31 1964-07-31 Derivatives of rifamycin sv
FR63914A FR5518M (US20090163788A1-20090625-C00002.png) 1964-07-31 1966-06-02

Publications (2)

Publication Number Publication Date
FI45044B FI45044B (US20090163788A1-20090625-C00002.png) 1971-11-30
FI45044C true FI45044C (fi) 1972-03-10

Family

ID=26171063

Family Applications (1)

Application Number Title Priority Date Filing Date
FI651805A FI45044C (fi) 1964-07-31 1965-07-27 Menetelmä antibioottisesti aktiivisen 3-substituoidun rifamysiini SV:n johdannaisten valmistamiseksi.

Country Status (13)

Country Link
US (1) US3342810A (US20090163788A1-20090625-C00002.png)
BE (1) BE667697A (US20090163788A1-20090625-C00002.png)
BR (1) BR6571577D0 (US20090163788A1-20090625-C00002.png)
CH (1) CH458353A (US20090163788A1-20090625-C00002.png)
DE (1) DE1595883A1 (US20090163788A1-20090625-C00002.png)
DK (1) DK115993B (US20090163788A1-20090625-C00002.png)
FI (1) FI45044C (US20090163788A1-20090625-C00002.png)
FR (2) FR5518M (US20090163788A1-20090625-C00002.png)
IL (1) IL23930A (US20090163788A1-20090625-C00002.png)
NL (1) NL6509961A (US20090163788A1-20090625-C00002.png)
NO (1) NO118375B (US20090163788A1-20090625-C00002.png)
SE (3) SE329850B (US20090163788A1-20090625-C00002.png)
YU (2) YU32700B (US20090163788A1-20090625-C00002.png)

Families Citing this family (48)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH536851A (de) * 1966-10-25 1973-05-15 Ciba Geigy Ag Verfahren zur Herstellung neuer antibiotisch wirksamer Verbindungen der Rifamycinreihen
GB1165179A (en) * 1966-10-25 1969-09-24 Lepetit Spa Derivatives of Rifamycin SV
GB1159267A (en) * 1966-11-03 1969-07-23 Lepetit Spa Rifamycin Derivatives
US3542762A (en) * 1967-06-07 1970-11-24 Lepetit Spa Process for rifamycins
FR2059967A1 (US20090163788A1-20090625-C00002.png) * 1969-08-06 1971-06-11 Lepetit Spa
US3933800A (en) * 1971-06-07 1976-01-20 Gruppo Lepetit S.P.A. New 3-formylrifamycin SV derivatives
IL39305A (en) * 1971-06-07 1975-08-31 Lepetit Spa O-substituted oximes of 3-formylrifamycin sv
GB1336399A (en) * 1971-06-24 1973-11-07 Lepetit Spa 3-formylrifamycin sv derivatives
US4005076A (en) * 1971-06-24 1977-01-25 Gruppo Lepetit S.P.A. Hydrazones of 3-formylrifamycin SV
BE794100A (fr) * 1972-02-23 1973-05-16 Lepetit Spa Derives 3-hydrazonomethyles de rifamycine et leur preparation
AR205434A1 (es) * 1972-03-27 1976-05-07 Lepetit Spa Proceso para la preparacion de 3-acilhidrazonometil rifamicinas sv
AR207762A1 (es) * 1973-07-25 1976-10-29 Archifar Ind Chim Trentino Procedimiento para la preparacion de 3-((4-metil-1-piperazin-1-il)-imino)-metil-rifamicina sv o rifampicina
GB1486118A (en) * 1975-03-05 1977-09-21 Lepetit Spa Rifamycin derivatives
GB1478563A (en) * 1975-03-05 1977-07-06 Lepetit Spa Rifamycin derivatives
IT1056271B (it) * 1975-05-20 1982-01-30 Archifar Ind Chim Trentino Prodotti derivati dalle amine aromatiche
US4179439A (en) * 1977-07-01 1979-12-18 Intreprinderea De Antibiotice Iasi Rifamycins and method for their preparation
US4150023A (en) * 1977-07-01 1979-04-17 Intreprinderea De Antibiotice Iasi Hydrosoluble rifamycins and process for their preparation
GB1594134A (en) * 1977-11-25 1981-07-30 Holco Investment Inc Rifamycins
IT1090772B (it) * 1977-12-20 1985-06-26 Alfa Farmaceutici Spa Derivati della rifamicina e procedimento per la loro preparazione
IT1090771B (it) * 1977-12-20 1985-06-26 Alfa Farmaceutici Spa Derivati delle 3 carbossirifamicines ed sv e procedimento per la loro preparazione
GB1591697A (en) * 1978-03-09 1981-06-24 Archifar Lab Chim Farm Process for producing 3-amino-rifamycins s and sv
US4220657A (en) * 1978-08-11 1980-09-02 Johnson Lewis A Method for treatment of human eye disease
US4292327A (en) * 1978-08-11 1981-09-29 Johnson Lewis A Method for treatment of human eye disease
AU536524B2 (en) * 1979-06-28 1984-05-10 Gruppo Lepetit S.P.A. Water soluble hydrozones of 3-formylifamyan
US4447432A (en) * 1981-11-17 1984-05-08 Farmitalia Carlo Erba S.P.A. Azino rifamycins
GB8308166D0 (en) * 1983-03-24 1983-05-05 Erba Farmitalia Preparation of azinomethyl-rifamycins
IT1201963B (it) * 1983-03-24 1989-02-02 Prodotti Antibiotici Spa Derivati delle rifamicine e procedimento per la loro preparazione
GB8318072D0 (en) * 1983-07-04 1983-08-03 Lepetit Spa Water-soluble rifampicin derivatives
MC1617A1 (fr) * 1983-09-01 1985-07-18 Ciba Geigy Ag Nouvelles hydrazones polycycliques,procede pour leur preparation
US4681938A (en) * 1984-08-27 1987-07-21 Ciba-Geigy Corporation Novel polycyclic hydrazones of rifamycins, their manufacture, and their pharmaceutical compositions for treating tuberculosis
US4551450A (en) * 1984-08-27 1985-11-05 Ciba-Geigy Corporation Rifamycin hydrazones, pharmaceutical compositions containing them and their use
US4631290A (en) * 1985-08-29 1986-12-23 American Home Products Corporation Method of treating hepatitis
US4743619A (en) * 1985-08-29 1988-05-10 American Home Products Corporation Method of treating hepatitis
WO1987002361A1 (en) * 1985-10-18 1987-04-23 Ciba-Geigy Ag Substituted 4-benzyl-piperazinyl compounds
US4876258A (en) * 1987-08-13 1989-10-24 Ciba-Geigy Corporation Biphenylyl compounds
KR890701591A (ko) * 1987-09-25 1989-12-21 베르너 발데그 4-(트리알킬벤질)-피페라지닐 화합물의 디아실 유도체
GB8816620D0 (en) * 1988-07-13 1988-08-17 Lepetit Spa Rifapentine hydrohalides
US6143740A (en) * 1996-11-19 2000-11-07 Georgetown University Heregulin antagonists and methods for their use
AU2002360416A1 (en) * 2001-11-21 2003-06-10 Activbiotics, Inc. Targeted therapeutics and uses thereof
US7820652B2 (en) * 2003-09-24 2010-10-26 Activbiotics Pharma, Llc Regimen for the administration of rifamycin-class antibiotics
BRPI0614758A2 (pt) 2005-08-11 2011-04-12 Targanta Therapeutics Inc rifamicinas fosfonadas e usos destas para a prevenção e tratamento de infecções na articulação e osso
WO2008008480A2 (en) * 2006-07-12 2008-01-17 Cumbre Pharmaceuticals Inc. Nitroheteroaryl-containing rifamycin derivatives
WO2009137380A1 (en) * 2008-05-05 2009-11-12 Janssen Pharmaceutica Nv 3-hydrazone piperazinyl rifamycin derivatives useful as antimicrobial agents
WO2010019511A2 (en) 2008-08-13 2010-02-18 Targanta Therapeutics Corp. Phosphonated rifamycins and uses thereof for the prevention and treatment of bone and joint infections
EP3400944B1 (en) 2010-11-08 2020-07-15 Albireo AB Ibat inhibitors for the treatment of liver diseases
US20170202850A1 (en) 2014-07-21 2017-07-20 Hiroaki Serizawa Ophthalmic compositions of rifamycins and uses thereof
US11702443B2 (en) * 2016-10-04 2023-07-18 Pop Test Oncology Llc Therapeutic agents and methods
WO2018067520A2 (en) 2016-10-04 2018-04-12 Pop Test Oncology Llc Therapeutic agents and methods:

Also Published As

Publication number Publication date
SE329895B (US20090163788A1-20090625-C00002.png) 1970-10-26
YU1168A (en) 1973-08-31
YU31937B (en) 1974-02-28
NL6509961A (US20090163788A1-20090625-C00002.png) 1966-02-01
YU1268A (en) 1974-12-31
BE667697A (US20090163788A1-20090625-C00002.png) 1965-11-16
FI45044B (US20090163788A1-20090625-C00002.png) 1971-11-30
SE329850B (US20090163788A1-20090625-C00002.png) 1970-10-26
FR5518M (US20090163788A1-20090625-C00002.png) 1967-11-06
US3342810A (en) 1967-09-19
CH458353A (fr) 1968-06-30
FR208F (US20090163788A1-20090625-C00002.png)
DK115993B (da) 1969-12-01
YU32700B (en) 1975-06-30
BR6571577D0 (pt) 1973-08-14
IL23930A (en) 1969-04-30
NO118375B (US20090163788A1-20090625-C00002.png) 1969-12-22
SE329851B (US20090163788A1-20090625-C00002.png) 1970-10-26
DE1595883A1 (de) 1970-02-12

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