ES8507488A1 - Procedimiento para la preparacion de derivados de n-aminoetil-3-fenil-4-cianopirrol - Google Patents
Procedimiento para la preparacion de derivados de n-aminoetil-3-fenil-4-cianopirrolInfo
- Publication number
- ES8507488A1 ES8507488A1 ES534540A ES534540A ES8507488A1 ES 8507488 A1 ES8507488 A1 ES 8507488A1 ES 534540 A ES534540 A ES 534540A ES 534540 A ES534540 A ES 534540A ES 8507488 A1 ES8507488 A1 ES 8507488A1
- Authority
- ES
- Spain
- Prior art keywords
- c6alkyl
- phenyl
- image
- independently hydrogen
- c6alkoxy
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- DYQJLSDORWRZSG-UHFFFAOYSA-N 1-(aminomethyl)-4-phenylpyrrole-3-carbonitrile Chemical class NCN1C=C(C#N)C(C=2C=CC=CC=2)=C1 DYQJLSDORWRZSG-UHFFFAOYSA-N 0.000 title abstract 2
- 230000003641 microbiacidal effect Effects 0.000 title abstract 2
- 229940124561 microbicide Drugs 0.000 title 1
- 125000004169 (C1-C6) alkyl group Chemical group 0.000 abstract 6
- 229910052739 hydrogen Inorganic materials 0.000 abstract 6
- 150000002431 hydrogen Chemical group 0.000 abstract 6
- 239000001257 hydrogen Substances 0.000 abstract 6
- 125000004454 (C1-C6) alkoxycarbonyl group Chemical group 0.000 abstract 4
- 150000001875 compounds Chemical class 0.000 abstract 3
- 229910052736 halogen Inorganic materials 0.000 abstract 3
- 150000002367 halogens Chemical group 0.000 abstract 3
- 125000000171 (C1-C6) haloalkyl group Chemical group 0.000 abstract 2
- 125000001797 benzyl group Chemical group [H]C1=C([H])C([H])=C(C([H])=C1[H])C([H])([H])* 0.000 abstract 2
- 239000000203 mixture Substances 0.000 abstract 2
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 2
- NINIDFKCEFEMDL-UHFFFAOYSA-N Sulfur Chemical group [S] NINIDFKCEFEMDL-UHFFFAOYSA-N 0.000 abstract 1
- 125000003118 aryl group Chemical group 0.000 abstract 1
- QVGXLLKOCUKJST-UHFFFAOYSA-N atomic oxygen Chemical group [O] QVGXLLKOCUKJST-UHFFFAOYSA-N 0.000 abstract 1
- 125000002915 carbonyl group Chemical group [*:2]C([*:1])=O 0.000 abstract 1
- 125000004093 cyano group Chemical group *C#N 0.000 abstract 1
- 125000002485 formyl group Chemical group [H]C(*)=O 0.000 abstract 1
- 125000000956 methoxy group Chemical group [H]C([H])([H])O* 0.000 abstract 1
- 125000002816 methylsulfanyl group Chemical group [H]C([H])([H])S[*] 0.000 abstract 1
- 244000005700 microbiome Species 0.000 abstract 1
- 229910052760 oxygen Inorganic materials 0.000 abstract 1
- 239000001301 oxygen Substances 0.000 abstract 1
- 230000003032 phytopathogenic effect Effects 0.000 abstract 1
- 229910052717 sulfur Inorganic materials 0.000 abstract 1
- 239000011593 sulfur Chemical group 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
- C07D207/34—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pyrrole Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Plural Heterocyclic Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
PROCEDIMIENTO PARA LA PREPARACION DE DERIVADOS DE N-AMINOETIL-3-FENIL-4-CIANOPIRROL.COMPRENDE: HACER REACCIONAR UN COMPUESTO DE FORMULA (II) CON UN COMPUESTO DE FORMULA (III), EN UN DISOLVENTE PROTICO A UNA TEMPERATURA DE 0J A 120JC, Y CON FORMALDEHIDO EN PRESENCIA DE UNA BASE O DE UN ACIDO ORGANICO O INORGANICO COMO CATALIZADOR DE LA REACCION, O EN UN DISOLVENTE APROTICO A TEMPERATURAS DE 0J A 120JC Y CON PARAFORMALDEHIDO EN PRESNCIA DE UNA BASE ORGANICA O INORGANICA COMO CATALIZADOR, PARA OBTENER UN COMPUESTO DE FORMULA (I) EN DONDE R1 Y R2 ES H, HALOGENO U OTROS, Z ES UNO DE LOS GRUPOS DE FORMULA (IV), (V) O (VI), EN DONDE R3 Y R4 SON H, ALQUILO DE C 1 A 6 U OTROS, O UNIDOS UN ANILLO AROMATICO YUXTACONDENSADO, R5 Y R6 SON H, ALQUILO DE C 1 A 6 U OTROS, N ES 4-5, X ES 0,5 U OTROS, R7 Y R8 SON H, ALQUILO DE C 1 A 6 U OTROS.SE UTILIZAN PARA COMBATIR A LOS HONGOS FITOPATOGENOS.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CH403183 | 1983-07-22 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| ES8507488A1 true ES8507488A1 (es) | 1985-10-01 |
| ES534540A0 ES534540A0 (es) | 1985-10-01 |
Family
ID=4268512
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES534540A Granted ES534540A0 (es) | 1983-07-22 | 1984-07-21 | Procedimiento para la preparacion de derivados de n-aminoetil-3-fenil-4-cianopirrol |
Country Status (13)
| Country | Link |
|---|---|
| US (1) | US4546099A (es) |
| EP (1) | EP0133247B1 (es) |
| JP (1) | JPS6042366A (es) |
| AT (1) | ATE48596T1 (es) |
| AU (1) | AU576773B2 (es) |
| CA (1) | CA1225990A (es) |
| DE (1) | DE3480703D1 (es) |
| ES (1) | ES534540A0 (es) |
| GR (1) | GR82206B (es) |
| IL (1) | IL72476A (es) |
| NZ (1) | NZ208972A (es) |
| PT (1) | PT78945B (es) |
| ZA (1) | ZA845629B (es) |
Families Citing this family (17)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BG43855A3 (en) * | 1983-06-17 | 1988-08-15 | Ciba- Geigy Ag,Ch | Fungicide means and method for protection from phytopathogenic fungi |
| EP0174910B1 (de) * | 1984-09-12 | 1990-04-04 | Ciba-Geigy Ag | Verfahren zur Herstellung von 4-Phenyl-pyrrol-derivaten |
| US4687861A (en) * | 1984-11-28 | 1987-08-18 | Ciba-Geigy Corporation | Microbicidal compositions |
| US4705800A (en) * | 1985-06-21 | 1987-11-10 | Ciba-Geigy Corporation | Difluorbenzodioxyl cyanopyrrole microbicidal compositions |
| LV5693A3 (lv) * | 1986-03-04 | 1995-02-20 | Ciba Geigy Ag | Panemiens kulturaugu aizsardzibai no fitopatogeniem Fungi imperfecti grupas mikroorganismiem |
| ES2022443B3 (es) * | 1986-03-04 | 1991-12-01 | Ciba-Geigy Ag | Utilizacion fungicida de un derivado de cianopirrol. |
| DE3702852A1 (de) * | 1987-01-31 | 1988-08-11 | Bayer Ag | 1-aminomethyl-3-aryl-4-cyano-pyrrole |
| DE3702853A1 (de) * | 1987-01-31 | 1988-08-11 | Bayer Ag | 1-aminomethyl-3-aryl-4-cyano-pyrrole |
| DE3804128A1 (de) * | 1988-02-11 | 1989-08-24 | Bayer Ag | 1-aminomethyl-3-(2-fluor-3-chlorphenyl)-4-cyano-pyrrol-derivate |
| DE3804127A1 (de) * | 1988-02-11 | 1989-08-24 | Bayer Ag | 1-aminomethyl-3-(2,4-difluor-3-chlorphenyl)-4-cyano-pyrrole |
| US4958030A (en) * | 1988-12-12 | 1990-09-18 | Ciba-Geigy Corporation | Process for the preparation of 3-phenylpyrrole derivatives |
| DE3922104A1 (de) * | 1989-07-05 | 1991-01-17 | Bayer Ag | N-vinyl-3-cyano-4-phenyl-pyrrol-derivate |
| DE3942225A1 (de) * | 1989-12-21 | 1991-06-27 | Bayer Ag | N-substituierte 3-cyano-4-phenyl-pyrrole |
| DE4004035A1 (de) * | 1989-12-23 | 1991-06-27 | Bayer Ag | Substituierte 1-aminomethyl-3-aryl-4-cyano-pyrrole |
| US5130328A (en) * | 1991-09-06 | 1992-07-14 | American Cyanamid Company | N-alkanoylaminomethyl and N-aroylaminomethyl pyrrole insecticidal and acaricidal agents |
| HU230609B1 (hu) * | 2000-01-19 | 2017-03-28 | Cadila Healthcare Ltd. | Hipolipidémiás és hipokoleszterinémiás hatású szubsztituált pirrolszármazékok, azokat tartalmazó gyógyszerkészítmények, eljárás előállításukra, köztitermékek és alkalmazásuk |
| US8822694B2 (en) * | 2009-02-25 | 2014-09-02 | Takeda Pharmaceutical Company Limited | Process for producing pyrrole compound |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3629220A (en) * | 1969-06-09 | 1971-12-21 | Pennwalt Corp | Homopolymerization of vinyl chloride with acyl sulfonyl peroxide initiator |
| IL56243A (en) * | 1978-01-31 | 1982-07-30 | Nippon Soda Co | Phenylpyrrole derivatives,their production and their use as fungicides |
| JPS5511524A (en) * | 1978-07-10 | 1980-01-26 | Nippon Soda Co Ltd | Cyanopyrrole derivative, its preparation and agricultural and horticultural fungicide |
| US4369277A (en) * | 1980-06-27 | 1983-01-18 | Ciba-Geigy Corporation | Pyrrole-stabilized chlorine-containing thermoplastics |
| BG43855A3 (en) * | 1983-06-17 | 1988-08-15 | Ciba- Geigy Ag,Ch | Fungicide means and method for protection from phytopathogenic fungi |
-
1984
- 1984-07-18 US US06/632,168 patent/US4546099A/en not_active Expired - Lifetime
- 1984-07-19 PT PT78945A patent/PT78945B/pt not_active IP Right Cessation
- 1984-07-19 AT AT84108547T patent/ATE48596T1/de active
- 1984-07-19 DE DE8484108547T patent/DE3480703D1/de not_active Expired - Lifetime
- 1984-07-19 EP EP84108547A patent/EP0133247B1/de not_active Expired
- 1984-07-20 GR GR75397A patent/GR82206B/el unknown
- 1984-07-20 CA CA000459318A patent/CA1225990A/en not_active Expired
- 1984-07-20 AU AU30900/84A patent/AU576773B2/en not_active Ceased
- 1984-07-20 NZ NZ208972A patent/NZ208972A/en unknown
- 1984-07-20 ZA ZA845629A patent/ZA845629B/xx unknown
- 1984-07-20 IL IL72476A patent/IL72476A/xx not_active IP Right Cessation
- 1984-07-21 ES ES534540A patent/ES534540A0/es active Granted
- 1984-07-23 JP JP59152755A patent/JPS6042366A/ja active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| ES534540A0 (es) | 1985-10-01 |
| ATE48596T1 (de) | 1989-12-15 |
| EP0133247A3 (en) | 1985-04-03 |
| IL72476A (en) | 1988-04-29 |
| NZ208972A (en) | 1987-11-27 |
| ZA845629B (en) | 1985-03-27 |
| AU576773B2 (en) | 1988-09-08 |
| IL72476A0 (en) | 1984-11-30 |
| GR82206B (es) | 1984-12-13 |
| DE3480703D1 (de) | 1990-01-18 |
| EP0133247B1 (de) | 1989-12-13 |
| PT78945A (en) | 1984-08-01 |
| EP0133247A2 (de) | 1985-02-20 |
| PT78945B (en) | 1986-10-21 |
| JPS6042366A (ja) | 1985-03-06 |
| AU3090084A (en) | 1985-01-24 |
| CA1225990A (en) | 1987-08-25 |
| US4546099A (en) | 1985-10-08 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PC1A | Transfer granted | ||
| FD1A | Patent lapsed |
Effective date: 20000301 |