ES8106292A1 - Nn*33mercaptoo22alkyll11oxopropyl**2*33 dihydroo1hhindolee22carboxylic acid and its derivative - Google Patents

Nn*33mercaptoo22alkyll11oxopropyl**2*33 dihydroo1hhindolee22carboxylic acid and its derivative

Info

Publication number
ES8106292A1
ES8106292A1 ES494201A ES494201A ES8106292A1 ES 8106292 A1 ES8106292 A1 ES 8106292A1 ES 494201 A ES494201 A ES 494201A ES 494201 A ES494201 A ES 494201A ES 8106292 A1 ES8106292 A1 ES 8106292A1
Authority
ES
Spain
Prior art keywords
formula
compound
hydrogen
lower alkyl
derivative
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES494201A
Other languages
Spanish (es)
Other versions
ES494201A0 (en
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Wyeth LLC
Original Assignee
American Home Products Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by American Home Products Corp filed Critical American Home Products Corp
Publication of ES494201A0 publication Critical patent/ES494201A0/en
Publication of ES8106292A1 publication Critical patent/ES8106292A1/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
    • C07D209/42—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)

Abstract

PROCEDURE FOR THE OBTAINING OF ACIDS N- (3-MERCAPTO-2-ALQUIL-1-OXOPROPIL) -2,3-DIHIDRO-1H-INDOL-2-CARBOXILICOS AND ITS DERIVATIVES, OF FORMULA (I), IN WHICH "N "VALE 0 O 1; R1, R3, R4, R5, X E Y MAY BE SEVERAL TYPES OF RADICALS, AND R2 IS HYDROGEN OR LOWER ALKYL; OR THE DISULFIDE OF THIS COMPOUND IN WHICH R4 IS SH O -S-, LINKED TO ACICLIC CARBON TO FORM A THYOLCETONE, OR ITS PHARMACOLOGICALLY COMPATIBLE SALTS. IT IS BASED ON THE RELATION OF A COMPOUND OF FORMULA (II); R14 IS R5 OR A PROTECTIVE GROUP OF CARBOXYLIC ACID, AND W1 IS BROMINE, IODINE, CHLORINE OR TOSYLOXYL; OR A COMPOUND OF FORMULA (III), R15 IS HYDROGEN OR LOWER ALKYL, WITH A THIOACIDE OR A THYOL OF FORMULA * FORMULA *. IF R4 IS A THIOACYL DERIVATIVE, THE RESULTING PRODUCT MAY SUBMIT TO HYDROLYSIS OR AMONOLYSIS, AND SUBSEQUENT CONDESATION OR CYCLING. *FORMULA* (Machine-translation by Google Translate, not legally binding)
ES494201A 1979-08-13 1980-08-12 Nn*33mercaptoo22alkyll11oxopropyl**2*33 dihydroo1hhindolee22carboxylic acid and its derivative Expired ES8106292A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US6581779A 1979-08-13 1979-08-13

Publications (2)

Publication Number Publication Date
ES494201A0 ES494201A0 (en) 1981-08-01
ES8106292A1 true ES8106292A1 (en) 1981-08-01

Family

ID=22065303

Family Applications (1)

Application Number Title Priority Date Filing Date
ES494201A Expired ES8106292A1 (en) 1979-08-13 1980-08-12 Nn*33mercaptoo22alkyll11oxopropyl**2*33 dihydroo1hhindolee22carboxylic acid and its derivative

Country Status (11)

Country Link
JP (1) JPS5636453A (en)
KR (2) KR890001194B1 (en)
AR (2) AR229394A1 (en)
DK (1) DK158347C (en)
ES (1) ES8106292A1 (en)
FI (1) FI802530A (en)
IL (1) IL60799A (en)
MX (1) MX160132A (en)
PH (2) PH18389A (en)
PT (1) PT71694B (en)
ZA (1) ZA804946B (en)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4287203A (en) * 1980-04-23 1981-09-01 Usv Pharmaceutical Corporation Antihypertensive 1,4-thiazepine-ones, 1,4-thiazonine-ones, and method of use thereof

Also Published As

Publication number Publication date
DK158347C (en) 1990-10-08
PT71694B (en) 1981-06-17
MX160132A (en) 1989-12-06
ES494201A0 (en) 1981-08-01
PH18414A (en) 1985-06-24
DK158347B (en) 1990-05-07
PH18389A (en) 1985-06-21
FI802530A (en) 1981-02-14
JPS5636453A (en) 1981-04-09
IL60799A (en) 1985-12-31
AR229394A1 (en) 1983-08-15
DK348280A (en) 1981-02-14
KR890001194B1 (en) 1989-04-27
PT71694A (en) 1980-09-01
ZA804946B (en) 1982-03-31
IL60799A0 (en) 1980-10-26
AR227348A1 (en) 1982-10-15
KR850001548B1 (en) 1985-10-17
KR830003421A (en) 1983-06-20

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