ES499610A0 - Un procedimiento de preparacion de una sal cuaternaria de un ester de eritromicina.a. - Google Patents

Un procedimiento de preparacion de una sal cuaternaria de un ester de eritromicina.a.

Info

Publication number
ES499610A0
ES499610A0 ES499610A ES499610A ES499610A0 ES 499610 A0 ES499610 A0 ES 499610A0 ES 499610 A ES499610 A ES 499610A ES 499610 A ES499610 A ES 499610A ES 499610 A0 ES499610 A0 ES 499610A0
Authority
ES
Spain
Prior art keywords
erythromycin
ester
procedure
preparation
quaternary salt
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
ES499610A
Other languages
English (en)
Other versions
ES8207192A1 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Abbott Laboratories
Original Assignee
Abbott Laboratories
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Abbott Laboratories filed Critical Abbott Laboratories
Publication of ES8207192A1 publication Critical patent/ES8207192A1/es
Publication of ES499610A0 publication Critical patent/ES499610A0/es
Granted legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
ES499610A 1980-02-20 1981-02-19 Un procedimiento de preparacion de una sal cuaternaria de un ester de eritromicina.a. Granted ES499610A0 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/122,948 US4264765A (en) 1980-02-20 1980-02-20 Salts of erythromycin A esters

Publications (2)

Publication Number Publication Date
ES8207192A1 ES8207192A1 (es) 1982-09-01
ES499610A0 true ES499610A0 (es) 1982-09-01

Family

ID=22405837

Family Applications (1)

Application Number Title Priority Date Filing Date
ES499610A Granted ES499610A0 (es) 1980-02-20 1981-02-19 Un procedimiento de preparacion de una sal cuaternaria de un ester de eritromicina.a.

Country Status (8)

Country Link
US (1) US4264765A (es)
EP (1) EP0034700A1 (es)
JP (1) JPS56118098A (es)
AU (1) AU6600981A (es)
CA (1) CA1144543A (es)
ES (1) ES499610A0 (es)
GR (1) GR73848B (es)
PH (1) PH16035A (es)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2519988B1 (fr) * 1982-01-20 1985-06-14 Refarmed Sa Derives thioliques de l'erythromycine a activite therapeutique, procede de preparation et produits pharmaceutiques dans lesquels ils apparaissent
FR2502627A1 (fr) * 1981-02-02 1982-10-01 Refarmed Sa Derives thioliques de l'erythromycine a activite therapeutique, procede de preparation et produits pharmaceutiques dans lesquels ils apparaissent
IT1163108B (it) * 1983-02-16 1987-04-08 Corvi Camillo Spa Sale di eritromicina dell'acido benzoico-o-carboniltiazolidina,procedimento per la sua preparazione e composizioni farmaceutiche che lo contengono
IT1173550B (it) * 1984-04-02 1987-06-24 Corvi Camillo Spa Sale di eritromicina con attivita'mucosecretolitica e fluidificante, processo per la sua preparazione e sue composizioni farmaceutiche
US4670549A (en) * 1985-03-18 1987-06-02 Taisho Pharmaceutical Co., Ltd. Method for selective methylation of erythromycin a derivatives
AU593006B2 (en) * 1985-08-31 1990-02-01 Kenkyusho, Kitasato Erythromycin derivative and process for preparing the same
US5723447A (en) * 1996-07-02 1998-03-03 Rhone Merieux, Inc. Water miscible erythromycin solutions
EP1051181B1 (en) * 1997-12-31 2004-03-17 The University Of Kansas Water soluble prodrugs of tertiary amine containing drugs and methods of making thereof
WO2011084846A1 (en) * 2010-01-07 2011-07-14 Alkermes, Inc. Quaternary ammonium salt prodrugs

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2857312A (en) * 1953-09-25 1958-10-21 Lilly Co Eli Esters of erythromycin and carbomycin
US2881163A (en) * 1953-11-16 1959-04-07 Abbott Lab Process of preparing salts
US3558594A (en) * 1968-09-04 1971-01-26 Abbott Lab Erythromycin aliphatic sulfate
PL122884B1 (en) * 1978-07-19 1982-08-31 Politechnika Gdanska Method of manufacture of quaternary trimethylammonium salts of inorganic derivatives of polyene macrolides

Also Published As

Publication number Publication date
GR73848B (es) 1984-05-07
AU6600981A (en) 1981-08-27
CA1144543A (en) 1983-04-12
US4264765A (en) 1981-04-28
PH16035A (en) 1983-06-02
ES8207192A1 (es) 1982-09-01
JPS56118098A (en) 1981-09-16
EP0034700A1 (en) 1981-09-02

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