ES482075A1 - Procedimiento para la preparacion de carbonilaminofenoxilicosustituidos con biciclo -3.1.0-hexilo. - Google Patents
Procedimiento para la preparacion de carbonilaminofenoxilicosustituidos con biciclo -3.1.0-hexilo.Info
- Publication number
- ES482075A1 ES482075A1 ES482075A ES482075A ES482075A1 ES 482075 A1 ES482075 A1 ES 482075A1 ES 482075 A ES482075 A ES 482075A ES 482075 A ES482075 A ES 482075A ES 482075 A1 ES482075 A1 ES 482075A1
- Authority
- ES
- Spain
- Prior art keywords
- compounds
- carbonylaminophenoxy
- bicyclo
- hexyl
- compositions containing
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D303/00—Compounds containing three-membered rings having one oxygen atom as the only ring hetero atom
- C07D303/02—Compounds containing oxirane rings
- C07D303/12—Compounds containing oxirane rings with hydrocarbon radicals, substituted by singly or doubly bound oxygen atoms
- C07D303/18—Compounds containing oxirane rings with hydrocarbon radicals, substituted by singly or doubly bound oxygen atoms by etherified hydroxyl radicals
- C07D303/20—Ethers with hydroxy compounds containing no oxirane rings
- C07D303/22—Ethers with hydroxy compounds containing no oxirane rings with monohydroxy compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/06—Antiglaucoma agents or miotics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/06—Antiarrhythmics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C53/00—Saturated compounds having only one carboxyl group bound to an acyclic carbon atom or hydrogen
- C07C53/132—Saturated compounds having only one carboxyl group bound to an acyclic carbon atom or hydrogen containing rings
- C07C53/136—Saturated compounds having only one carboxyl group bound to an acyclic carbon atom or hydrogen containing rings containing condensed ring systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
- C07D263/04—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
- C07D263/06—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with hydrocarbon radicals, substituted by oxygen atoms, attached to ring carbon atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Ophthalmology & Optometry (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Procedimiento para la preparación de carbonilaminofenoxílicos sustituidos con biciclo [3.1.0]HEXILO. Este invento se refiere a un procedimiento para la preparación de 1-alcohilamino-3-(4- [endobiciclo[3.1.0]hex-6-il)alcohilureido]-1-fenoxi)-2- propanol y a sus sales farmacéuticamente aceptables; de 1- alcohilamino-3-(4-[endobiciclo[3.1.0]hex-6- il)alcohilcarbonilamino]-1-fenoxi)-2-propanol y a sus sales farmacéuticamente aceptables. Este invento se refiere además a un procedimiento para la preparación de 5-(4/[endobiciclo[3.1.0]hex-6- il)alcohilureido]-metil-3-alcohil-oxazolidinas opcionalmente sustituidas en posición 2 y a sus sales farmacéuticamente aceptables; de 5-(4-/[endobiciclo[3.1.0]nex-6- il)alcohilcarbnilamino]-1-fenoxi)-metil-3-alcohil-oxazolidinas opcionalmente sustituidas en posición 2 y a sus sales farmacéuticamente aceptables.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US05/921,371 US4177280A (en) | 1978-07-03 | 1978-07-03 | Bicyclo[3.1.0]hexyl-substituted carbonylaminophenoxy cardiovascular agents |
Publications (1)
Publication Number | Publication Date |
---|---|
ES482075A1 true ES482075A1 (es) | 1980-03-01 |
Family
ID=25445332
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES482075A Expired ES482075A1 (es) | 1978-07-03 | 1979-06-29 | Procedimiento para la preparacion de carbonilaminofenoxilicosustituidos con biciclo -3.1.0-hexilo. |
Country Status (13)
Country | Link |
---|---|
US (1) | US4177280A (es) |
EP (1) | EP0007710A1 (es) |
JP (1) | JPS559074A (es) |
AU (1) | AU4852379A (es) |
CA (1) | CA1105054A (es) |
DD (1) | DD148215A5 (es) |
DK (1) | DK276479A (es) |
ES (1) | ES482075A1 (es) |
IL (1) | IL57705A0 (es) |
NZ (1) | NZ190880A (es) |
PL (1) | PL116994B1 (es) |
SU (1) | SU854271A3 (es) |
ZA (1) | ZA793292B (es) |
Families Citing this family (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4402976A (en) * | 1981-04-24 | 1983-09-06 | E. R. Squibb & Sons, Inc. | Method for treating glaucoma with systemic nadolol compositions |
EP0282127B1 (en) * | 1987-03-09 | 1994-02-02 | The Procter & Gamble Company | Beta-aminoethyl-substituted phenyl compounds, and anti-inflammatory or analgesic compositions containing them |
DE60234057D1 (de) | 2001-07-25 | 2009-11-26 | Raptor Pharmaceutical Inc | Zusammensetzungen und verfahren zur modulation des transports durch die blut-hirn-schranke |
CN103259027A (zh) | 2005-04-28 | 2013-08-21 | 普罗透斯数字保健公司 | 药物信息系统 |
EP2063905B1 (en) | 2006-09-18 | 2014-07-30 | Raptor Pharmaceutical Inc | Treatment of liver disorders by administration of receptor-associated protein (rap)-conjugates |
CA2969926C (en) | 2009-02-20 | 2018-05-15 | 2-Bbb Medicines B.V. | Glutathione-based drug delivery system |
EP2427178B1 (en) | 2009-05-06 | 2023-01-04 | Laboratory Skin Care, Inc. | Dermal delivery compositions comprising active agent-calcium phosphate particle complexes and methods of using the same |
US20120077778A1 (en) | 2010-09-29 | 2012-03-29 | Andrea Bourdelais | Ladder-Frame Polyether Conjugates |
JP2020506895A (ja) * | 2017-01-17 | 2020-03-05 | ボード オブ レジェンツ, ザ ユニバーシティ オブ テキサス システムBoard Of Regents, The University Of Texas System | インドールアミン2,3−ジオキシゲナーゼおよび/またはトリプトファンジオキシゲナーゼの阻害剤として有用な化合物 |
WO2020018670A1 (en) | 2018-07-17 | 2020-01-23 | Board Of Regents, The University Of Texas System | Compounds useful as inhibitors of indoleamine 2,3-dioxygenase and/or tryptophan dioxygenase |
Family Cites Families (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB1078852A (en) * | 1964-09-30 | 1967-08-09 | Ici Ltd | Alkanolamine derivatives |
US4038313A (en) * | 1970-01-08 | 1977-07-26 | Ciba-Geigy Corporation | Cycloalkylureido phenoxy propanolamines |
CA1149819A (en) * | 1970-01-08 | 1983-07-12 | Max Wilhelm | Process for the manufacture of new amines |
US4038414A (en) * | 1972-06-08 | 1977-07-26 | Ciba-Geigy Corporation | Amines and processes for their manufacture |
US4035420A (en) * | 1972-07-06 | 1977-07-12 | Aktiebolaget Hassle | Substituted ureido alkylene phenoxy propanolamines |
AT334385B (de) * | 1973-12-20 | 1976-01-10 | Chemie Linz Ag | Verfahren zur herstellung von neuen phenoxypropylaminderivaten und deren salzen |
US4063025A (en) * | 1975-02-05 | 1977-12-13 | Yamanouchi Pharmaceutical Co., Ltd. | 4-Substituted amino-α-aminomethylbenzyl alcohol derivatives |
US4064258A (en) * | 1976-07-19 | 1977-12-20 | Syntex (U.S.A.) Inc. | Thiazole cardiovascular agents |
-
1978
- 1978-07-03 US US05/921,371 patent/US4177280A/en not_active Expired - Lifetime
-
1979
- 1979-06-27 PL PL1979216661A patent/PL116994B1/pl unknown
- 1979-06-29 NZ NZ190880A patent/NZ190880A/xx unknown
- 1979-06-29 AU AU48523/79A patent/AU4852379A/en not_active Abandoned
- 1979-06-29 CA CA331,064A patent/CA1105054A/en not_active Expired
- 1979-06-29 DK DK276479A patent/DK276479A/da not_active Application Discontinuation
- 1979-06-29 EP EP79301262A patent/EP0007710A1/en not_active Withdrawn
- 1979-06-29 ES ES482075A patent/ES482075A1/es not_active Expired
- 1979-06-29 JP JP8153979A patent/JPS559074A/ja active Pending
- 1979-07-02 SU SU792788053A patent/SU854271A3/ru active
- 1979-07-02 IL IL57705A patent/IL57705A0/xx unknown
- 1979-07-03 ZA ZA793292A patent/ZA793292B/xx unknown
- 1979-07-03 DD DD79214074A patent/DD148215A5/de unknown
Also Published As
Publication number | Publication date |
---|---|
JPS559074A (en) | 1980-01-22 |
CA1105054A (en) | 1981-07-14 |
DD148215A5 (de) | 1981-05-13 |
DK276479A (da) | 1980-01-04 |
EP0007710A1 (en) | 1980-02-06 |
AU4852379A (en) | 1980-01-10 |
PL116994B1 (en) | 1981-07-31 |
SU854271A3 (ru) | 1981-08-07 |
ZA793292B (en) | 1981-02-25 |
US4177280A (en) | 1979-12-04 |
NZ190880A (en) | 1981-04-24 |
IL57705A0 (en) | 1979-11-30 |
PL216661A1 (es) | 1980-03-24 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FD1A | Patent lapsed |
Effective date: 19971001 |