ES415482A1 - A method of preparation of a c-amidino compound. (Machine-translation by Google Translate, not legally binding) - Google Patents

A method of preparation of a c-amidino compound. (Machine-translation by Google Translate, not legally binding)

Info

Publication number
ES415482A1
ES415482A1 ES415482A ES415482A ES415482A1 ES 415482 A1 ES415482 A1 ES 415482A1 ES 415482 A ES415482 A ES 415482A ES 415482 A ES415482 A ES 415482A ES 415482 A1 ES415482 A1 ES 415482A1
Authority
ES
Spain
Prior art keywords
formula
lower alkyl
translation
machine
legally binding
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES415482A
Other languages
Spanish (es)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Merck and Co Inc
Original Assignee
Merck and Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck and Co Inc filed Critical Merck and Co Inc
Publication of ES415482A1 publication Critical patent/ES415482A1/en
Expired legal-status Critical Current

Links

Landscapes

  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)

Abstract

A method of preparing a C-amidino compound of the formula: **(See formula)** where the radical (see formula) is found in positions 5 or 6, and the symbols X, R1, R2, R3 and R4 have the following meanings: X represents oxygen or sulfur, R1 represents a five-membered monocyclic heteroaromatic ring containing from 1 to 3 heteroatoms selected from the group consisting of oxygen, sulfur and nitrogen, R3 represents hydrogen or lower alkyl and R4 represents hydrogen, lower alkyl, lower alkoxy, lower alkyl thio, cycloalkyl, aryl, aryloxy, arylthio, aralkyl, heteroaryl, heteroayloxy, heteroarylthio, mono (lower) alkyl, dialkyl (lower) amino or cycloalkylamino, R6 is lower alkyl and R15 and R16 are members selected from the group consisting of hydrogen and lower alkyl, the method of which is to react an iminoester hydrochloride of the formula: **(See formula)** where R1, R3, R4 and X are as defined above with a compound of the formula: **(See formula)** where R15 and R16 are those previously described. (Machine-translation by Google Translate, not legally binding)
ES415482A 1970-03-05 1973-06-02 A method of preparation of a c-amidino compound. (Machine-translation by Google Translate, not legally binding) Expired ES415482A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US1695770A 1970-03-05 1970-03-05

Publications (1)

Publication Number Publication Date
ES415482A1 true ES415482A1 (en) 1976-11-16

Family

ID=21779932

Family Applications (5)

Application Number Title Priority Date Filing Date
ES388211A Expired ES388211A1 (en) 1970-03-05 1971-02-12 A procedure for the preparation of substituted benzymidazoles. (Machine-translation by Google Translate, not legally binding)
ES415483A Expired ES415483A1 (en) 1970-03-05 1973-06-02 A procedure for the preparation of substituted benzymidazoles. (Machine-translation by Google Translate, not legally binding)
ES415481A Expired ES415481A1 (en) 1970-03-05 1973-06-02 A procedure for the preparation of substituted benzymidazoles. (Machine-translation by Google Translate, not legally binding)
ES415482A Expired ES415482A1 (en) 1970-03-05 1973-06-02 A method of preparation of a c-amidino compound. (Machine-translation by Google Translate, not legally binding)
ES415480A Expired ES415480A1 (en) 1970-03-05 1973-06-02 A method of preparation of an N-amidino compound. (Machine-translation by Google Translate, not legally binding)

Family Applications Before (3)

Application Number Title Priority Date Filing Date
ES388211A Expired ES388211A1 (en) 1970-03-05 1971-02-12 A procedure for the preparation of substituted benzymidazoles. (Machine-translation by Google Translate, not legally binding)
ES415483A Expired ES415483A1 (en) 1970-03-05 1973-06-02 A procedure for the preparation of substituted benzymidazoles. (Machine-translation by Google Translate, not legally binding)
ES415481A Expired ES415481A1 (en) 1970-03-05 1973-06-02 A procedure for the preparation of substituted benzymidazoles. (Machine-translation by Google Translate, not legally binding)

Family Applications After (1)

Application Number Title Priority Date Filing Date
ES415480A Expired ES415480A1 (en) 1970-03-05 1973-06-02 A method of preparation of an N-amidino compound. (Machine-translation by Google Translate, not legally binding)

Country Status (10)

Country Link
AR (3) AR199178A1 (en)
CS (1) CS180571B2 (en)
ES (5) ES388211A1 (en)
IE (2) IE34938B1 (en)
IL (1) IL36101A (en)
NO (1) NO131932C (en)
SU (1) SU472504A3 (en)
YU (1) YU34895B (en)
ZA (1) ZA7164B (en)
ZM (1) ZM2571A1 (en)

Also Published As

Publication number Publication date
CS180571B2 (en) 1978-01-31
IE34939L (en) 1971-09-05
IL36101A0 (en) 1971-04-28
NO131932C (en) 1975-08-27
ZA7164B (en) 1972-08-30
SU472504A3 (en) 1975-05-30
ES415480A1 (en) 1976-02-16
AR199177A1 (en) 1974-08-14
ES415481A1 (en) 1976-02-16
IE34938L (en) 1971-09-05
YU34895B (en) 1980-04-30
ES415483A1 (en) 1976-02-16
IE34939B1 (en) 1975-10-01
ES388211A1 (en) 1974-02-16
AR199178A1 (en) 1974-08-14
NO131932B (en) 1975-05-20
YU51571A (en) 1979-10-31
ZM2571A1 (en) 1972-10-23
IE34938B1 (en) 1975-10-01
IL36101A (en) 1976-02-29
AR199179A1 (en) 1974-08-14

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