ES2124162A1 - Un nuevo procedimiento para preparar compuestos farmaceuticamente activos. - Google Patents

Un nuevo procedimiento para preparar compuestos farmaceuticamente activos.

Info

Publication number
ES2124162A1
ES2124162A1 ES09600462A ES9600462A ES2124162A1 ES 2124162 A1 ES2124162 A1 ES 2124162A1 ES 09600462 A ES09600462 A ES 09600462A ES 9600462 A ES9600462 A ES 9600462A ES 2124162 A1 ES2124162 A1 ES 2124162A1
Authority
ES
Spain
Prior art keywords
active compounds
pharmaceutically active
new process
preparing pharmaceutically
preparing
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
ES09600462A
Other languages
English (en)
Other versions
ES2124162B1 (es
Inventor
Norman John Lewis
Neal Ward
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
SmithKline Beecham Ltd
Original Assignee
SmithKline Beecham Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GBGB9504060.6A external-priority patent/GB9504060D0/en
Application filed by SmithKline Beecham Ltd filed Critical SmithKline Beecham Ltd
Priority to ES9600462A priority Critical patent/ES2124162B1/es
Publication of ES2124162A1 publication Critical patent/ES2124162A1/es
Application granted granted Critical
Publication of ES2124162B1 publication Critical patent/ES2124162B1/es
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Un nuevo procedimiento para preparar compuestos farmacéuticamente activos, en particular granisetrón, que comprende hacer reaccionar indazol sustituido en la posición 3 con monóxido de carbono y endo-3-amino-9-meti1-9-azabiciclo-[3.3.1]-nonano o una de sus bases de Schiff.
ES9600462A 1995-03-01 1996-02-28 Un nuevo procedimiento para preparar compuestos farmaceuticamente activos. Expired - Fee Related ES2124162B1 (es)

Priority Applications (1)

Application Number Priority Date Filing Date Title
ES9600462A ES2124162B1 (es) 1995-03-01 1996-02-28 Un nuevo procedimiento para preparar compuestos farmaceuticamente activos.

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB9504060.6A GB9504060D0 (en) 1995-03-01 1995-03-01 Novel process
ES9600462A ES2124162B1 (es) 1995-03-01 1996-02-28 Un nuevo procedimiento para preparar compuestos farmaceuticamente activos.

Publications (2)

Publication Number Publication Date
ES2124162A1 true ES2124162A1 (es) 1999-01-16
ES2124162B1 ES2124162B1 (es) 1999-11-16

Family

ID=26154953

Family Applications (1)

Application Number Title Priority Date Filing Date
ES9600462A Expired - Fee Related ES2124162B1 (es) 1995-03-01 1996-02-28 Un nuevo procedimiento para preparar compuestos farmaceuticamente activos.

Country Status (1)

Country Link
ES (1) ES2124162B1 (es)

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2008117282A1 (en) * 2007-03-27 2008-10-02 Chemagis Ltd. Polymorph of granisetron base and production process therefor
WO2008151677A1 (en) 2007-06-13 2008-12-18 Inke, S.A. Polymorphic form of granisetron base, methods for obtaining it and formulation containing it

Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0200444A2 (en) * 1985-04-27 1986-11-05 Beecham Group Plc Azabicyclononyl-indazole-carboxamide having 5-HT antagonist activity
EP0214772A1 (en) * 1985-08-16 1987-03-18 Beecham Group Plc Novel compounds
EP0223385A2 (en) * 1985-10-21 1987-05-27 Beecham Group Plc 8-Azabicyclo[3,2,1]octane and 9-azabicyclo[3,3,1]nonane derivatives
WO1991001316A1 (en) * 1989-07-21 1991-02-07 Beecham Group Plc New 9-azabicyclo[3.3.1]nonane-derivate

Patent Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0200444A2 (en) * 1985-04-27 1986-11-05 Beecham Group Plc Azabicyclononyl-indazole-carboxamide having 5-HT antagonist activity
EP0214772A1 (en) * 1985-08-16 1987-03-18 Beecham Group Plc Novel compounds
EP0223385A2 (en) * 1985-10-21 1987-05-27 Beecham Group Plc 8-Azabicyclo[3,2,1]octane and 9-azabicyclo[3,3,1]nonane derivatives
WO1991001316A1 (en) * 1989-07-21 1991-02-07 Beecham Group Plc New 9-azabicyclo[3.3.1]nonane-derivate

Cited By (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2008117282A1 (en) * 2007-03-27 2008-10-02 Chemagis Ltd. Polymorph of granisetron base and production process therefor
WO2008151677A1 (en) 2007-06-13 2008-12-18 Inke, S.A. Polymorphic form of granisetron base, methods for obtaining it and formulation containing it
EP2164848A1 (en) 2007-06-13 2010-03-24 Inke, S.A. Polymorphic form of granisetron base, methods for obtaining it and formulation containing it
EP2164848B1 (en) * 2007-06-13 2016-02-24 Inke, S.A. Polymorphic form of granisetron base, methods for obtaining it and formulation containing it

Also Published As

Publication number Publication date
ES2124162B1 (es) 1999-11-16

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