ES2120885B1 - NEW TIENOPIRIMIDONAS WITH ANTIFUNGAL ACTIVITY. - Google Patents

NEW TIENOPIRIMIDONAS WITH ANTIFUNGAL ACTIVITY.

Info

Publication number
ES2120885B1
ES2120885B1 ES9600646A ES9600646A ES2120885B1 ES 2120885 B1 ES2120885 B1 ES 2120885B1 ES 9600646 A ES9600646 A ES 9600646A ES 9600646 A ES9600646 A ES 9600646A ES 2120885 B1 ES2120885 B1 ES 2120885B1
Authority
ES
Spain
Prior art keywords
tienopirimidonas
new
antifungal activity
halogen
compounds
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
ES9600646A
Other languages
Spanish (es)
Other versions
ES2120885A1 (en
Inventor
Javier Bartroli
Manuel Anguita
Enric Turmo
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Noucor Health SA
Original Assignee
J Uriach y Cia SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority to ES9600646A priority Critical patent/ES2120885B1/en
Application filed by J Uriach y Cia SA filed Critical J Uriach y Cia SA
Priority to AU68703/96A priority patent/AU6870396A/en
Priority to JP50725497A priority patent/JP4049207B2/en
Priority to DK96929201T priority patent/DK0783501T3/en
Priority to PCT/EP1996/003420 priority patent/WO1997005130A1/en
Priority to DE69611512T priority patent/DE69611512T2/en
Priority to CA002201477A priority patent/CA2201477C/en
Priority to KR1019970701515A priority patent/KR100423590B1/en
Priority to PT96929201T priority patent/PT783501E/en
Priority to ES96929201T priority patent/ES2153975T3/en
Priority to MX9702382A priority patent/MX9702382A/en
Priority to BR9606547A priority patent/BR9606547A/en
Priority to EP96929201A priority patent/EP0783501B9/en
Priority to AT96929201T priority patent/ATE198593T1/en
Priority to US08/809,967 priority patent/US5807854A/en
Priority to NO19971470A priority patent/NO312898B1/en
Publication of ES2120885A1 publication Critical patent/ES2120885A1/en
Application granted granted Critical
Publication of ES2120885B1 publication Critical patent/ES2120885B1/en
Priority to GR20010400466T priority patent/GR3035621T3/en
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Abstract

COMPUESTOS DE FORMULA I, Y SUS SALES Y SOLVATOS, EN DONDE AR ES UN GRUPO FENILO OPCIONALMENTE SUSTITUIDO POR UNO O MAS GRUPOS HALOGENO Y/O TRIFLUOROMETILO; R1 ES UN GRUPO C1-C4 ALQUILO; R2 ES HIDROGENO O UN GRUPO C1-C4 ALQUILO; O BIEN R1 JUNTO CON R2 FORMAN UNA CADENA C2-C4 POLIMETILENO; R3 REPRESENTA CIANO, HALOGENO, C1-C4 HALOALQUILO O C1-C4 HALOALCOXI; Y R4 REPRESENTA HIDROGENO O C1-C4 ALQUILO. DICHOS COMPUESTOS SON UTILES COMO ANTIFUNGICOS. SE DESCRIBE TAMBIEN PROCEDIMIENTOS PARA SU OBTENCION Y COMPOSICIONES FARMACEUTICAS QUE LOS CONTIENEN.COMPOUNDS OF FORMULA I, AND ITS SALTS AND SOLVATES, WHERE AR IS A PHENYLUS GROUP OPTIONALLY REPLACED BY ONE OR MORE HALOGEN AND / OR TRIFLUOROMETILE GROUPS; R1 IS A GROUP C1-C4 ALKYL; R2 IS HYDROGEN OR A C1-C4 ALKYL GROUP; OR R1 TOGETHER WITH R2 FORM A CHAIN C2-C4 POLYMETHYLENE; R3 REPRESENTS CYAN, HALOGEN, C1-C4 HALOALKYL OR C1-C4 HALOALCOXI; AND R4 REPRESENTS HYDROGEN OR C1-C4 RENT. SUCH COMPOUNDS ARE USEFUL AS ANTIFUNGALS. IT IS ALSO DESCRIBED PROCEDURES FOR THEIR OBTAINING AND PHARMACEUTICAL COMPOSITIONS THAT CONTAIN THEM.

ES9600646A 1995-08-02 1996-03-15 NEW TIENOPIRIMIDONAS WITH ANTIFUNGAL ACTIVITY. Expired - Fee Related ES2120885B1 (en)

Priority Applications (17)

Application Number Priority Date Filing Date Title
ES9600646A ES2120885B1 (en) 1996-03-15 1996-03-15 NEW TIENOPIRIMIDONAS WITH ANTIFUNGAL ACTIVITY.
EP96929201A EP0783501B9 (en) 1995-08-02 1996-08-02 pyrimidone derivatives with antifungal activity
DK96929201T DK0783501T3 (en) 1995-08-02 1996-08-02 Pyrimidone derivatives with anti-fungal activity
PCT/EP1996/003420 WO1997005130A1 (en) 1995-08-02 1996-08-02 New pyrimidone derivatives with antifungal activity
DE69611512T DE69611512T2 (en) 1995-08-02 1996-08-02 PYRIMIDONE DERIVATIVES WITH ANTIFUNGAL EFFECT
CA002201477A CA2201477C (en) 1995-08-02 1996-08-02 New pyrimidone derivatives with antifungal activity
KR1019970701515A KR100423590B1 (en) 1995-08-02 1996-08-02 New pyrimidone derivatives with antifungal activity
PT96929201T PT783501E (en) 1995-08-02 1996-08-02 PYRIMIDONE DERIVATIVES WITH ANTIFUNGAL ACTIVITY
AU68703/96A AU6870396A (en) 1995-08-02 1996-08-02 New pyrimidone derivatives with antifungal activity
MX9702382A MX9702382A (en) 1995-08-02 1996-08-02 New pyrimidone derivatives with antifungal activity.
BR9606547A BR9606547A (en) 1995-08-02 1996-08-02 New pyrimidone derivatives with fungicidal activity
JP50725497A JP4049207B2 (en) 1995-08-02 1996-08-02 Novel pyrimidone derivatives with antifungal activity
AT96929201T ATE198593T1 (en) 1995-08-02 1996-08-02 PYRIMIDONE DERIVATIVES WITH ANTI-FUNGAL EFFECT
US08/809,967 US5807854A (en) 1995-08-02 1996-08-02 Pyrimidone derivatives with antifungal activity
ES96929201T ES2153975T3 (en) 1995-08-02 1996-08-02 DERIVATIVES OF PIRIMIDONA WITH ANTIFUNGIC ACTIVITY.
NO19971470A NO312898B1 (en) 1995-08-02 1997-04-01 New pyrimidone derivatives with fungicidal activity
GR20010400466T GR3035621T3 (en) 1995-08-02 2001-03-23 New pyrimidone derivatives with antifungal activity

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
ES9600646A ES2120885B1 (en) 1996-03-15 1996-03-15 NEW TIENOPIRIMIDONAS WITH ANTIFUNGAL ACTIVITY.

Publications (2)

Publication Number Publication Date
ES2120885A1 ES2120885A1 (en) 1998-11-01
ES2120885B1 true ES2120885B1 (en) 1999-06-16

Family

ID=8294213

Family Applications (1)

Application Number Title Priority Date Filing Date
ES9600646A Expired - Fee Related ES2120885B1 (en) 1995-08-02 1996-03-15 NEW TIENOPIRIMIDONAS WITH ANTIFUNGAL ACTIVITY.

Country Status (1)

Country Link
ES (1) ES2120885B1 (en)

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2024336A6 (en) * 1990-10-16 1992-02-16 Uriach & Cia Sa J Process for obtaining new thiazole derivatives
TW218017B (en) * 1992-04-28 1993-12-21 Takeda Pharm Industry Co Ltd

Also Published As

Publication number Publication date
ES2120885A1 (en) 1998-11-01

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