ES2106683A1 - Derivados de 1,3-dioxoperhidropirido (1,2-c) pirimidinas como antagonistas de colecistoquinina. - Google Patents

Derivados de 1,3-dioxoperhidropirido (1,2-c) pirimidinas como antagonistas de colecistoquinina.

Info

Publication number
ES2106683A1
ES2106683A1 ES09501857A ES9501857A ES2106683A1 ES 2106683 A1 ES2106683 A1 ES 2106683A1 ES 09501857 A ES09501857 A ES 09501857A ES 9501857 A ES9501857 A ES 9501857A ES 2106683 A1 ES2106683 A1 ES 2106683A1
Authority
ES
Spain
Prior art keywords
derivatives
dioxoperhydropyrido
pyrimidines
cholecystokinin
antagonists
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
ES09501857A
Other languages
English (en)
Other versions
ES2106683B1 (es
Inventor
Muniz Rosario Gonzalez
Lopez M Teresa Garcia
Monterrey Isabel Gomez
Rosario Herranz
Martinez Mercedes Martin
Carcamo Ana Maria Barber
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Consejo Superior de Investigaciones Cientificas CSIC
Original Assignee
Consejo Superior de Investigaciones Cientificas CSIC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Consejo Superior de Investigaciones Cientificas CSIC filed Critical Consejo Superior de Investigaciones Cientificas CSIC
Priority to ES9501857A priority Critical patent/ES2106683B1/es
Publication of ES2106683A1 publication Critical patent/ES2106683A1/es
Application granted granted Critical
Publication of ES2106683B1 publication Critical patent/ES2106683B1/es
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

DERIVADOS DE 1,3-DIOXOPERHIDROPIRIDO [1,2,-C] PIRIMINAS COMO ANTAGONISTAS DE COLECISTOQUININA. LA PRESENTE INVENCION SE REFIERE A DERIVADOS DE 1,3-DIOXOPERHIDROPIRIDO [1,2,-C] PIRIMINAS, E INTERMEDIOS PARA SU PREPARACION DE FORMULA GENERAL FORMULA DICHOS DERIVADOS SON UTILES COMO ANTAGONISTAS DE COLECISTOQUININA (CCK) Y POR LO TANTO COMO AGENTES ACTIVOS SOBRE EL SISTEMA NERVIOSO CENTRAL Y EL PERIFERICO.
ES9501857A 1995-09-26 1995-09-26 Derivados de 1,3-dioxoperhidropirido (1,2-c) pirimidinas como antagonistas de colecistoquinina. Expired - Fee Related ES2106683B1 (es)

Priority Applications (1)

Application Number Priority Date Filing Date Title
ES9501857A ES2106683B1 (es) 1995-09-26 1995-09-26 Derivados de 1,3-dioxoperhidropirido (1,2-c) pirimidinas como antagonistas de colecistoquinina.

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
ES9501857A ES2106683B1 (es) 1995-09-26 1995-09-26 Derivados de 1,3-dioxoperhidropirido (1,2-c) pirimidinas como antagonistas de colecistoquinina.

Publications (2)

Publication Number Publication Date
ES2106683A1 true ES2106683A1 (es) 1997-11-01
ES2106683B1 ES2106683B1 (es) 1998-07-01

Family

ID=8291662

Family Applications (1)

Application Number Title Priority Date Filing Date
ES9501857A Expired - Fee Related ES2106683B1 (es) 1995-09-26 1995-09-26 Derivados de 1,3-dioxoperhidropirido (1,2-c) pirimidinas como antagonistas de colecistoquinina.

Country Status (1)

Country Link
ES (1) ES2106683B1 (es)

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1992000295A1 (en) * 1990-06-21 1992-01-09 Rhone-Poulenc Rorer International (Holdings) Inc. Tetrahydropyridoindoles as cholecystokinin and gastrin antagonists

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1992000295A1 (en) * 1990-06-21 1992-01-09 Rhone-Poulenc Rorer International (Holdings) Inc. Tetrahydropyridoindoles as cholecystokinin and gastrin antagonists

Non-Patent Citations (2)

* Cited by examiner, † Cited by third party
Title
TETRAHEDRON LETTERS, Vol. 34, n‘ 22, pßginas 3593-3594, 1993. GOMEZ-MONTERREY et al. "Stereospecific synthesis of (2R-3S)-3-amino-2-piperidineacetic acid derivatives for use as conformational constraint in peptides". *
TETRAHEDRON, Vol. 51, n‘ 9, pßginas 2729-2736, 1995. GOMEZ-MONTERREY et al. "Synthesis of 8-amino-3-oxoindolizidine-1-carboxylic acid derivatives as conformationally restricted templates for use in design of peptide mimetics". *

Also Published As

Publication number Publication date
ES2106683B1 (es) 1998-07-01

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