ES2106683A1 - Derivados de 1,3-dioxoperhidropirido (1,2-c) pirimidinas como antagonistas de colecistoquinina. - Google Patents
Derivados de 1,3-dioxoperhidropirido (1,2-c) pirimidinas como antagonistas de colecistoquinina.Info
- Publication number
- ES2106683A1 ES2106683A1 ES09501857A ES9501857A ES2106683A1 ES 2106683 A1 ES2106683 A1 ES 2106683A1 ES 09501857 A ES09501857 A ES 09501857A ES 9501857 A ES9501857 A ES 9501857A ES 2106683 A1 ES2106683 A1 ES 2106683A1
- Authority
- ES
- Spain
- Prior art keywords
- derivatives
- dioxoperhydropyrido
- pyrimidines
- cholecystokinin
- antagonists
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
DERIVADOS DE 1,3-DIOXOPERHIDROPIRIDO [1,2,-C] PIRIMINAS COMO ANTAGONISTAS DE COLECISTOQUININA. LA PRESENTE INVENCION SE REFIERE A DERIVADOS DE 1,3-DIOXOPERHIDROPIRIDO [1,2,-C] PIRIMINAS, E INTERMEDIOS PARA SU PREPARACION DE FORMULA GENERAL FORMULA DICHOS DERIVADOS SON UTILES COMO ANTAGONISTAS DE COLECISTOQUININA (CCK) Y POR LO TANTO COMO AGENTES ACTIVOS SOBRE EL SISTEMA NERVIOSO CENTRAL Y EL PERIFERICO.
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
ES9501857A ES2106683B1 (es) | 1995-09-26 | 1995-09-26 | Derivados de 1,3-dioxoperhidropirido (1,2-c) pirimidinas como antagonistas de colecistoquinina. |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
ES9501857A ES2106683B1 (es) | 1995-09-26 | 1995-09-26 | Derivados de 1,3-dioxoperhidropirido (1,2-c) pirimidinas como antagonistas de colecistoquinina. |
Publications (2)
Publication Number | Publication Date |
---|---|
ES2106683A1 true ES2106683A1 (es) | 1997-11-01 |
ES2106683B1 ES2106683B1 (es) | 1998-07-01 |
Family
ID=8291662
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES9501857A Expired - Fee Related ES2106683B1 (es) | 1995-09-26 | 1995-09-26 | Derivados de 1,3-dioxoperhidropirido (1,2-c) pirimidinas como antagonistas de colecistoquinina. |
Country Status (1)
Country | Link |
---|---|
ES (1) | ES2106683B1 (es) |
Citations (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO1992000295A1 (en) * | 1990-06-21 | 1992-01-09 | Rhone-Poulenc Rorer International (Holdings) Inc. | Tetrahydropyridoindoles as cholecystokinin and gastrin antagonists |
-
1995
- 1995-09-26 ES ES9501857A patent/ES2106683B1/es not_active Expired - Fee Related
Patent Citations (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO1992000295A1 (en) * | 1990-06-21 | 1992-01-09 | Rhone-Poulenc Rorer International (Holdings) Inc. | Tetrahydropyridoindoles as cholecystokinin and gastrin antagonists |
Non-Patent Citations (2)
Title |
---|
TETRAHEDRON LETTERS, Vol. 34, n‘ 22, pßginas 3593-3594, 1993. GOMEZ-MONTERREY et al. "Stereospecific synthesis of (2R-3S)-3-amino-2-piperidineacetic acid derivatives for use as conformational constraint in peptides". * |
TETRAHEDRON, Vol. 51, n‘ 9, pßginas 2729-2736, 1995. GOMEZ-MONTERREY et al. "Synthesis of 8-amino-3-oxoindolizidine-1-carboxylic acid derivatives as conformationally restricted templates for use in design of peptide mimetics". * |
Also Published As
Publication number | Publication date |
---|---|
ES2106683B1 (es) | 1998-07-01 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
DE69705300T2 (de) | Cyclopropylalkansäurederivate | |
ES2164657T3 (es) | Derivados aza-biciclicos puenteados como antagonistas de la sustancia p. | |
AU2337197A (en) | Cinnamic acid derivatives and their use as integrin antagonists | |
AU2962295A (en) | Cannabinoid receptor antagonists | |
MY113806A (en) | Antiparasitic marcfortines and paraherquamides | |
AU2420897A (en) | Meta-substituted phenylene sulphonamide derivatives | |
CA2174494A1 (en) | Benzofurans | |
AU9057191A (en) | N-substituted lactams useful as cholecystokinin antagonists | |
BG103548A (en) | Vitronectine receptor antagonists | |
GR3036813T3 (en) | Novel n-(1-alkyl-5-phenyl-2,3,4,5-tetrahydro-1h-benzo[b][1,4]diazepin-3-yl)-acetamides | |
DE69516128D1 (de) | Mercaptoacetylamid-1,3,4,5-tetrahydrobenzo(c)azepin-3-ein disulfidderivate als enkephalinase und ace inhibitoren | |
EP0833819A4 (en) | N- (2,4-DIOXO-2,3,4,5-TETRAHYDRO-1H-1,5-BENZODIAZEPIN-3-YL) -3-AMIDE | |
DE69330754D1 (de) | 2,5-DIOXO-2,5-DIHYDRO-1H-BENZ[b]AZEPINE ALS NMDA REZEPTOR ANTAGONISTEN | |
GR3034602T3 (en) | Novel n-(2,4-dioxo-2,3,4,5-tetrahydro-1h-1,5-benzodiazepin-3y l)-3-amides | |
CA2219359A1 (en) | Hydantoin derivatives as intermediates for pharmaceutical active compounds | |
CA2066083A1 (en) | Benzodiazepine analogs as cholecystokinin antagonists | |
IT1276167B1 (it) | Imidazo(1,2-alfa)chinossalin-4-ammine attivi come antagonisti adenosinici,procedimento per la loro preparazione e loro composizioni | |
PL316870A1 (en) | Derivatives of 5-heterocyclo 1,5-benzodiazepine | |
AU7681198A (en) | Novel compounds | |
EP0842156A4 (en) | N- (2,4-DIOXO-2,3,4,5-TETRAHYDRO-1H-1,5-BENZODIAZEPIN-3-YL) -3-AMIDE | |
CA2214072A1 (en) | Benzo [b] thiophene compounds, intermediates, processes, compositions, and methods | |
ES2106683A1 (es) | Derivados de 1,3-dioxoperhidropirido (1,2-c) pirimidinas como antagonistas de colecistoquinina. | |
HUP9900883A3 (en) | Amino acid derivatives of substituted quinoxaline 2,3-dione derivatives as glutamate receptor antagonists | |
ITTO930661A1 (it) | Derivati acidi poliamidici ad attivita' antigastrinica, procedimento per la loro preparazione e loro uso farmaceutico. | |
TW371661B (en) | Novel intermediates and their use to prepare N,N'-bridged bisindolylmaleimides |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
EC2A | Search report published |
Date of ref document: 19971101 Kind code of ref document: A1 Effective date: 19971101 |
|
FD1A | Patent lapsed |
Effective date: 20050927 |