ES2087813B1 - NON-AROMATIC HETEROCICLES CONTAINING SUBSTITUTED NITROGEN BENCILAMINE. - Google Patents

NON-AROMATIC HETEROCICLES CONTAINING SUBSTITUTED NITROGEN BENCILAMINE.

Info

Publication number
ES2087813B1
ES2087813B1 ES9301771A ES9301771A ES2087813B1 ES 2087813 B1 ES2087813 B1 ES 2087813B1 ES 9301771 A ES9301771 A ES 9301771A ES 9301771 A ES9301771 A ES 9301771A ES 2087813 B1 ES2087813 B1 ES 2087813B1
Authority
ES
Spain
Prior art keywords
bencilamine
substituted nitrogen
aromatic
containing substituted
heterocicles
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
ES9301771A
Other languages
Spanish (es)
Other versions
ES2087813A1 (en
Inventor
Jr Harry R Howard
Masaya Ikunaka
Fumitaka Ito
Iii John A Lowe
Masami Nakane
Brian T O'neill
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Inc
Original Assignee
Pfizer Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Inc filed Critical Pfizer Inc
Priority to ES9301771A priority Critical patent/ES2087813B1/en
Publication of ES2087813A1 publication Critical patent/ES2087813A1/en
Application granted granted Critical
Publication of ES2087813B1 publication Critical patent/ES2087813B1/en
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Abstract

LA PRESENTE INVENCION SE REFIERE A NUEVOS HETEROCICLOS NO-AROMATICOS QUE CONTIENEN NITROGENO BENCILAMINO SUSTITUIDOS Y, ESPECIFICAMENTE, A COMPUESTOS DE LA FORMULA *FIG* EN LA QUE W, R1, R2, R3 Y A SON COMO SE DEFINEN EN LA MEMORIA DESCRIPTIVA, Y A INTERMEDIOS EMPLEADOS EN LA SINTESIS DE TALES COMPUESTOS. LOS NUEVOS COMPUESTOS DE LA FORMULA I SON UTILES EN EL TRATAMIENTO DE TRASTORNOS INFLAMATORIOS Y DEL SISTEMA NERVIOSA CENTRAL, ASI COMO DE OTROS TRASTORNOS.THE PRESENT INVENTION REFERS TO NEW NON-AROMATIC HETERO CYCLES CONTAINING SUBSTITUTED NITROGEN BENCILAMINE AND, SPECIFICALLY, TO COMPOUNDS OF THE * FIG * FORMULA IN WHICH W, R1, R2, R3 ARE ALREADY AS DEFINED IN THE DESCRIPTIVE MEMORY. EMPLOYEES IN THE SYNTHESIS OF SUCH COMPOUNDS. THE NEW COMPOUNDS OF FORMULA I ARE USEFUL IN THE TREATMENT OF INFLAMMATORY DISORDERS AND THE CENTRAL NERVOUS SYSTEM, AS WELL AS OTHER DISORDERS.

ES9301771A 1993-08-09 1993-08-09 NON-AROMATIC HETEROCICLES CONTAINING SUBSTITUTED NITROGEN BENCILAMINE. Expired - Fee Related ES2087813B1 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
ES9301771A ES2087813B1 (en) 1993-08-09 1993-08-09 NON-AROMATIC HETEROCICLES CONTAINING SUBSTITUTED NITROGEN BENCILAMINE.

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
ES9301771A ES2087813B1 (en) 1993-08-09 1993-08-09 NON-AROMATIC HETEROCICLES CONTAINING SUBSTITUTED NITROGEN BENCILAMINE.

Publications (2)

Publication Number Publication Date
ES2087813A1 ES2087813A1 (en) 1996-07-16
ES2087813B1 true ES2087813B1 (en) 1997-02-01

Family

ID=8282814

Family Applications (1)

Application Number Title Priority Date Filing Date
ES9301771A Expired - Fee Related ES2087813B1 (en) 1993-08-09 1993-08-09 NON-AROMATIC HETEROCICLES CONTAINING SUBSTITUTED NITROGEN BENCILAMINE.

Country Status (1)

Country Link
ES (1) ES2087813B1 (en)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN111770914A (en) * 2018-07-26 2020-10-13 凯瑞康宁生物工程(武汉)有限公司 Compounds as neurokinin-1 receptor antagonists and uses thereof

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1995007908A1 (en) * 1993-09-17 1995-03-23 Pfizer Inc. Heteroarylamino and heteroarylsulfonamido substituted 3-benzylaminomethyl piperidines and related compounds

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5721255A (en) * 1992-08-19 1998-02-24 Pfizer Inc. Substituted benzylamino nitrogen containing non-aromatic heterocycles

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN111770914A (en) * 2018-07-26 2020-10-13 凯瑞康宁生物工程(武汉)有限公司 Compounds as neurokinin-1 receptor antagonists and uses thereof
CN111770914B (en) * 2018-07-26 2023-06-20 凯瑞康宁生物工程(武汉)有限公司 Compounds as neurokinin-1 receptor antagonists and uses thereof

Also Published As

Publication number Publication date
ES2087813A1 (en) 1996-07-16

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Legal Events

Date Code Title Description
EC2A Search report published

Effective date: 19960716

FD1A Patent lapsed

Effective date: 20050810