ES2087813B1 - NON-AROMATIC HETEROCICLES CONTAINING SUBSTITUTED NITROGEN BENCILAMINE. - Google Patents
NON-AROMATIC HETEROCICLES CONTAINING SUBSTITUTED NITROGEN BENCILAMINE.Info
- Publication number
- ES2087813B1 ES2087813B1 ES9301771A ES9301771A ES2087813B1 ES 2087813 B1 ES2087813 B1 ES 2087813B1 ES 9301771 A ES9301771 A ES 9301771A ES 9301771 A ES9301771 A ES 9301771A ES 2087813 B1 ES2087813 B1 ES 2087813B1
- Authority
- ES
- Spain
- Prior art keywords
- bencilamine
- substituted nitrogen
- aromatic
- containing substituted
- heterocicles
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
Links
Abstract
LA PRESENTE INVENCION SE REFIERE A NUEVOS HETEROCICLOS NO-AROMATICOS QUE CONTIENEN NITROGENO BENCILAMINO SUSTITUIDOS Y, ESPECIFICAMENTE, A COMPUESTOS DE LA FORMULA *FIG* EN LA QUE W, R1, R2, R3 Y A SON COMO SE DEFINEN EN LA MEMORIA DESCRIPTIVA, Y A INTERMEDIOS EMPLEADOS EN LA SINTESIS DE TALES COMPUESTOS. LOS NUEVOS COMPUESTOS DE LA FORMULA I SON UTILES EN EL TRATAMIENTO DE TRASTORNOS INFLAMATORIOS Y DEL SISTEMA NERVIOSA CENTRAL, ASI COMO DE OTROS TRASTORNOS.THE PRESENT INVENTION REFERS TO NEW NON-AROMATIC HETERO CYCLES CONTAINING SUBSTITUTED NITROGEN BENCILAMINE AND, SPECIFICALLY, TO COMPOUNDS OF THE * FIG * FORMULA IN WHICH W, R1, R2, R3 ARE ALREADY AS DEFINED IN THE DESCRIPTIVE MEMORY. EMPLOYEES IN THE SYNTHESIS OF SUCH COMPOUNDS. THE NEW COMPOUNDS OF FORMULA I ARE USEFUL IN THE TREATMENT OF INFLAMMATORY DISORDERS AND THE CENTRAL NERVOUS SYSTEM, AS WELL AS OTHER DISORDERS.
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
ES9301771A ES2087813B1 (en) | 1993-08-09 | 1993-08-09 | NON-AROMATIC HETEROCICLES CONTAINING SUBSTITUTED NITROGEN BENCILAMINE. |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
ES9301771A ES2087813B1 (en) | 1993-08-09 | 1993-08-09 | NON-AROMATIC HETEROCICLES CONTAINING SUBSTITUTED NITROGEN BENCILAMINE. |
Publications (2)
Publication Number | Publication Date |
---|---|
ES2087813A1 ES2087813A1 (en) | 1996-07-16 |
ES2087813B1 true ES2087813B1 (en) | 1997-02-01 |
Family
ID=8282814
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES9301771A Expired - Fee Related ES2087813B1 (en) | 1993-08-09 | 1993-08-09 | NON-AROMATIC HETEROCICLES CONTAINING SUBSTITUTED NITROGEN BENCILAMINE. |
Country Status (1)
Country | Link |
---|---|
ES (1) | ES2087813B1 (en) |
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN111770914A (en) * | 2018-07-26 | 2020-10-13 | 凯瑞康宁生物工程(武汉)有限公司 | Compounds as neurokinin-1 receptor antagonists and uses thereof |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO1995007908A1 (en) * | 1993-09-17 | 1995-03-23 | Pfizer Inc. | Heteroarylamino and heteroarylsulfonamido substituted 3-benzylaminomethyl piperidines and related compounds |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5721255A (en) * | 1992-08-19 | 1998-02-24 | Pfizer Inc. | Substituted benzylamino nitrogen containing non-aromatic heterocycles |
-
1993
- 1993-08-09 ES ES9301771A patent/ES2087813B1/en not_active Expired - Fee Related
Cited By (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN111770914A (en) * | 2018-07-26 | 2020-10-13 | 凯瑞康宁生物工程(武汉)有限公司 | Compounds as neurokinin-1 receptor antagonists and uses thereof |
CN111770914B (en) * | 2018-07-26 | 2023-06-20 | 凯瑞康宁生物工程(武汉)有限公司 | Compounds as neurokinin-1 receptor antagonists and uses thereof |
Also Published As
Publication number | Publication date |
---|---|
ES2087813A1 (en) | 1996-07-16 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
EC2A | Search report published |
Effective date: 19960716 |
|
FD1A | Patent lapsed |
Effective date: 20050810 |