ES2062921A1 - 3-(indol-2-carboxiamido)quinuclidinas. - Google Patents

3-(indol-2-carboxiamido)quinuclidinas.

Info

Publication number
ES2062921A1
ES2062921A1 ES09202252A ES9202252A ES2062921A1 ES 2062921 A1 ES2062921 A1 ES 2062921A1 ES 09202252 A ES09202252 A ES 09202252A ES 9202252 A ES9202252 A ES 9202252A ES 2062921 A1 ES2062921 A1 ES 2062921A1
Authority
ES
Spain
Prior art keywords
quinuclidines
carboxyamido
indol
ind
arylsulphonyloxy
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
ES09202252A
Other languages
English (en)
Other versions
ES2062921B1 (es
Inventor
Henning Boettcher
Cristoph Seyfried
Gerd Bartoszyk
Klaus-Otto Minck
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Merck Patent GmbH
Original Assignee
Merck Patent GmbH
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Patent GmbH filed Critical Merck Patent GmbH
Priority to ES9202252A priority Critical patent/ES2062921B1/es
Publication of ES2062921A1 publication Critical patent/ES2062921A1/es
Application granted granted Critical
Publication of ES2062921B1 publication Critical patent/ES2062921B1/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

3-(INDOL-2-CARBOXIAMIDO)QUINUCLIDINAS DE LA FORMULA I IND-CO-NHR: I, EN LAS QUE IND ES UN GRUPO 2-INDOLILO QUE ESTA INSUBSTITUIDO O DE MONO A TRISUBSTITUIDO POR ALQUILO, ALCOXI, ALCOXICARBONILO Y/O ALQUILTIO CON EN CADA CASO 1-5 ATOMOS DE C, ARALQUILOXI DE 7-11 C, ACILOXI DE 1-5 C, AROILOXI DE 6-10 C, TRIFLUOROMETILO, CIANO, FLUOR, CLORO, HIDROXILO, ALQUILSULFONILOXI DE 1-4 C, ARILSULFONILOXI DE 6-10 C, CARBOXILO Y/OMETILENDIOXI Y R ES 3-QUINUCLIDINILO Y SUS SALES FISIOLOGICAMENTE ACEPTABLES QUE MUESTRAN UN EFECTO ANTAGONISTA HACIA LA SEROTONINA Y PUEDEN USARSE COMO PSICOFARMACOS.
ES9202252A 1992-11-06 1992-11-06 3-(indol-2-carboxiamido)quinuclidinas. Expired - Lifetime ES2062921B1 (es)

Priority Applications (1)

Application Number Priority Date Filing Date Title
ES9202252A ES2062921B1 (es) 1992-11-06 1992-11-06 3-(indol-2-carboxiamido)quinuclidinas.

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
ES9202252A ES2062921B1 (es) 1992-11-06 1992-11-06 3-(indol-2-carboxiamido)quinuclidinas.

Publications (2)

Publication Number Publication Date
ES2062921A1 true ES2062921A1 (es) 1994-12-16
ES2062921B1 ES2062921B1 (es) 1995-06-16

Family

ID=8278717

Family Applications (1)

Application Number Title Priority Date Filing Date
ES9202252A Expired - Lifetime ES2062921B1 (es) 1992-11-06 1992-11-06 3-(indol-2-carboxiamido)quinuclidinas.

Country Status (1)

Country Link
ES (1) ES2062921B1 (es)

Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0289170A2 (en) * 1987-04-25 1988-11-02 Beecham Group Plc Azabicyclic compounds, process for their preparation and pharmaceutical compositions containing them
EP0328200A1 (en) * 1988-02-12 1989-08-16 Merck Sharp & Dohme Ltd. Five-membered ring systems with bonded azacyclic ring substituents
GB2231264A (en) * 1986-07-30 1990-11-14 Sandoz Ltd Therapeutic use of serotonin antagonists

Patent Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2231264A (en) * 1986-07-30 1990-11-14 Sandoz Ltd Therapeutic use of serotonin antagonists
EP0289170A2 (en) * 1987-04-25 1988-11-02 Beecham Group Plc Azabicyclic compounds, process for their preparation and pharmaceutical compositions containing them
EP0328200A1 (en) * 1988-02-12 1989-08-16 Merck Sharp & Dohme Ltd. Five-membered ring systems with bonded azacyclic ring substituents

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
JOURNAL OF MEDICINAL CHEMISTRY, Vol. 34, n‘ 1, Enero 1991, American Chemical Society, Washington, US; C.S. SWAIN et al.: "Novel 5-HT3 antagonists. Indole oxadiazoles"; pßg. 140-146. *

Also Published As

Publication number Publication date
ES2062921B1 (es) 1995-06-16

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Legal Events

Date Code Title Description
FA2A Application withdrawn

Effective date: 19960115