EP4136056A4 - NON-AQUEOUS TOPICAL FORMULATIONS - Google Patents

NON-AQUEOUS TOPICAL FORMULATIONS Download PDF

Info

Publication number
EP4136056A4
EP4136056A4 EP21788324.8A EP21788324A EP4136056A4 EP 4136056 A4 EP4136056 A4 EP 4136056A4 EP 21788324 A EP21788324 A EP 21788324A EP 4136056 A4 EP4136056 A4 EP 4136056A4
Authority
EP
European Patent Office
Prior art keywords
topical formulations
aqueous topical
aqueous
formulations
topical
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
EP21788324.8A
Other languages
German (de)
French (fr)
Other versions
EP4136056A2 (en
Inventor
Jihoon P. BAEK
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Baek Clinical Inc
Original Assignee
Baek Clinical Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Baek Clinical Inc filed Critical Baek Clinical Inc
Publication of EP4136056A2 publication Critical patent/EP4136056A2/en
Publication of EP4136056A4 publication Critical patent/EP4136056A4/en
Pending legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00—Cosmetics or similar toiletry preparations
    • A61K8/02—Cosmetics or similar toiletry preparations characterised by special physical form
    • A61K8/04—Dispersions; Emulsions
    • A61K8/06—Emulsions
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/365—Lactones
    • A61K31/375—Ascorbic acid, i.e. vitamin C; Salts thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/02—Inorganic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00—Cosmetics or similar toiletry preparations
    • A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/33—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing oxygen
    • A61K8/34—Alcohols
    • A61K8/345—Alcohols containing more than one hydroxy group
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00—Cosmetics or similar toiletry preparations
    • A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/33—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing oxygen
    • A61K8/36—Carboxylic acids; Salts or anhydrides thereof
    • A61K8/365—Hydroxycarboxylic acids; Ketocarboxylic acids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00—Cosmetics or similar toiletry preparations
    • A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/33—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing oxygen
    • A61K8/36—Carboxylic acids; Salts or anhydrides thereof
    • A61K8/368—Carboxylic acids; Salts or anhydrides thereof with carboxyl groups directly bound to carbon atoms of aromatic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00—Cosmetics or similar toiletry preparations
    • A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/40—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing nitrogen
    • A61K8/42—Amides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00—Cosmetics or similar toiletry preparations
    • A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/67—Vitamins
    • A61K8/676—Ascorbic acid, i.e. vitamin C
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00—Cosmetics or similar toiletry preparations
    • A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/72—Cosmetics or similar toiletry preparations characterised by the composition containing organic macromolecular compounds
    • A61K8/84—Cosmetics or similar toiletry preparations characterised by the composition containing organic macromolecular compounds obtained by reactions otherwise than those involving only carbon-carbon unsaturated bonds
    • A61K8/89—Polysiloxanes
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0014—Skin, i.e. galenical aspects of topical compositions
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/10—Dispersions; Emulsions
    • A61K9/107—Emulsions ; Emulsion preconcentrates; Micelles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q19/00—Preparations for care of the skin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q19/00—Preparations for care of the skin
    • A61Q19/08—Anti-ageing preparations
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2800/00—Properties of cosmetic compositions or active ingredients thereof or formulation aids used therein and process related aspects
    • A61K2800/20—Chemical, physico-chemical or functional or structural properties of the composition as a whole
    • A61K2800/30—Characterized by the absence of a particular group of ingredients
    • A61K2800/31—Anhydrous

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Birds (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Emergency Medicine (AREA)
  • Dermatology (AREA)
  • Dispersion Chemistry (AREA)
  • Gerontology & Geriatric Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Inorganic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Cosmetics (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
EP21788324.8A 2020-04-16 2021-04-16 NON-AQUEOUS TOPICAL FORMULATIONS Pending EP4136056A4 (en)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
US202063010888P 2020-04-16 2020-04-16
US202063010878P 2020-04-16 2020-04-16
US202063010884P 2020-04-16 2020-04-16
US202063010881P 2020-04-16 2020-04-16
US202063010889P 2020-04-16 2020-04-16
PCT/US2021/027832 WO2021212077A2 (en) 2020-04-16 2021-04-16 Non-aqueous topical formulations

Publications (2)

Publication Number Publication Date
EP4136056A2 EP4136056A2 (en) 2023-02-22
EP4136056A4 true EP4136056A4 (en) 2024-09-04

Family

ID=78084516

Family Applications (1)

Application Number Title Priority Date Filing Date
EP21788324.8A Pending EP4136056A4 (en) 2020-04-16 2021-04-16 NON-AQUEOUS TOPICAL FORMULATIONS

Country Status (7)

Country Link
EP (1) EP4136056A4 (en)
JP (1) JP2023522328A (en)
KR (1) KR20230005221A (en)
CN (1) CN115697903A (en)
BR (1) BR112022020994A2 (en)
TW (1) TW202203912A (en)
WO (1) WO2021212077A2 (en)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2021212073A1 (en) 2020-04-16 2021-10-21 Baek Clinical Inc. High-potency vitamin c and sugar alcohol topical formulations
WO2022141384A1 (en) * 2020-12-31 2022-07-07 L'oreal Composition for caring for kertatin materials
WO2023069639A1 (en) * 2021-10-20 2023-04-27 Baek Clinical Inc. Anhydrous urea emulsions with a retinoid agent
JP2024542652A (en) * 2021-11-30 2024-11-15 ロレアル Kits and methods for treating the skin
CN115887289B (en) * 2022-10-27 2024-03-08 广州百孚润化工有限公司 Moisturizing composition, cosmetic containing moisturizing composition and preparation method of moisturizing composition
KR102671775B1 (en) * 2023-08-30 2024-06-03 한국콜마주식회사 Cosmetic composition with excellent potency retention of active components and formulation stability and a method for manufacturing the cosmetic composition
CN117530874B (en) * 2023-11-15 2025-04-15 无锡知妍生物科技有限公司 A water-soluble azelaic acid system and preparation method thereof
FR3157147A1 (en) * 2023-12-20 2025-06-27 L'oreal Cosmetic composition comprising a polar oil, an alkanol, a polyol, azelaic acid, and a low water content.
FR3157146A1 (en) 2023-12-20 2025-06-27 L'oreal Cosmetic composition comprising an oil, an alkanol, a polyol, azelaic acid, and a low water content.
WO2025132572A1 (en) 2023-12-20 2025-06-26 L'oreal Cosmetic composition comprising an oil, an alkanol, a polyol, azelaic acid and a low content of water

Citations (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH05229927A (en) * 1992-02-21 1993-09-07 Kao Corp Skin-whitening cosmetic
WO1996039119A1 (en) * 1995-06-06 1996-12-12 Neutrogena Corporation Topical vehicles containing solubilized and stabilized azelaic acid
US6361783B2 (en) * 1997-06-27 2002-03-26 Reulon Consumer Products Corporation Compositions containing stabilized ascorbic acid and related methods
WO2005070380A1 (en) * 2004-01-13 2005-08-04 Skinceuticals, Inc. Stabilized ascorbic acid compositions and methods therefor
US20070172436A1 (en) * 2006-01-23 2007-07-26 Jerry Zhang Nonaqueous ascorbic acid compositions and methods for preparing same
US10149808B2 (en) * 2016-03-31 2018-12-11 L'oreal Cosmetic compositions and methods for providing full spectrum photo protection

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6020367A (en) * 1997-12-02 2000-02-01 Avon Products, Inc. Supersaturated ascorbic acid solutions
US8568749B2 (en) * 2009-04-02 2013-10-29 Sesvalia Usa, Llc Systems and methods for skin rejuvenation
JP6776355B2 (en) * 2015-12-29 2020-10-28 ロレアル Stable antioxidant composition
ES2972007T3 (en) * 2016-10-31 2024-06-10 Sytheon Ltd Compositions and methods to improve skin
EP3713583B1 (en) * 2017-11-21 2025-01-22 Topix Pharmaceuticals, Inc. Methods and compositions for treatment of skin
WO2020081868A1 (en) * 2018-10-18 2020-04-23 Baek Clinical Inc. High-potency vitamin c topical formulations

Patent Citations (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH05229927A (en) * 1992-02-21 1993-09-07 Kao Corp Skin-whitening cosmetic
WO1996039119A1 (en) * 1995-06-06 1996-12-12 Neutrogena Corporation Topical vehicles containing solubilized and stabilized azelaic acid
US6361783B2 (en) * 1997-06-27 2002-03-26 Reulon Consumer Products Corporation Compositions containing stabilized ascorbic acid and related methods
WO2005070380A1 (en) * 2004-01-13 2005-08-04 Skinceuticals, Inc. Stabilized ascorbic acid compositions and methods therefor
US20070172436A1 (en) * 2006-01-23 2007-07-26 Jerry Zhang Nonaqueous ascorbic acid compositions and methods for preparing same
US10149808B2 (en) * 2016-03-31 2018-12-11 L'oreal Cosmetic compositions and methods for providing full spectrum photo protection

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
ANONYMOUS: "24hr moisturizing anti-fatigue concentrate", GNPD, MINTEL, 31 March 2010 (2010-03-31), XP002762818 *

Also Published As

Publication number Publication date
EP4136056A2 (en) 2023-02-22
KR20230005221A (en) 2023-01-09
WO2021212077A3 (en) 2022-06-16
JP2023522328A (en) 2023-05-30
BR112022020994A2 (en) 2022-12-06
CN115697903A (en) 2023-02-03
TW202203912A (en) 2022-02-01
WO2021212077A2 (en) 2021-10-21

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