EP3386944A4 - Verfahren zur herstellung von lisdexamphetamin - Google Patents
Verfahren zur herstellung von lisdexamphetamin Download PDFInfo
- Publication number
- EP3386944A4 EP3386944A4 EP16872573.7A EP16872573A EP3386944A4 EP 3386944 A4 EP3386944 A4 EP 3386944A4 EP 16872573 A EP16872573 A EP 16872573A EP 3386944 A4 EP3386944 A4 EP 3386944A4
- Authority
- EP
- European Patent Office
- Prior art keywords
- lisdexamphetamine
- preparation
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
Links
- VOBHXZCDAVEXEY-JSGCOSHPSA-N lisdexamfetamine Chemical compound NCCCC[C@H](N)C(=O)N[C@@H](C)CC1=CC=CC=C1 VOBHXZCDAVEXEY-JSGCOSHPSA-N 0.000 title 1
- 229960001451 lisdexamfetamine Drugs 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C231/00—Preparation of carboxylic acid amides
- C07C231/14—Preparation of carboxylic acid amides by formation of carboxamide groups together with reactions not involving the carboxamide groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D203/00—Heterocyclic compounds containing three-membered rings with one nitrogen atom as the only ring hetero atom
- C07D203/04—Heterocyclic compounds containing three-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
- C07D203/06—Heterocyclic compounds containing three-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
- C07D203/16—Heterocyclic compounds containing three-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with acylated ring nitrogen atoms
- C07D203/18—Heterocyclic compounds containing three-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with acylated ring nitrogen atoms by carboxylic acids, or by sulfur or nitrogen analogues thereof
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IN4670MU2015 | 2015-12-11 | ||
| PCT/IN2016/050441 WO2017098533A2 (en) | 2015-12-11 | 2016-12-12 | Process for preparation of lisdexamphetamine |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| EP3386944A2 EP3386944A2 (de) | 2018-10-17 |
| EP3386944A4 true EP3386944A4 (de) | 2019-08-28 |
Family
ID=59012856
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| EP16872573.7A Withdrawn EP3386944A4 (de) | 2015-12-11 | 2016-12-12 | Verfahren zur herstellung von lisdexamphetamin |
Country Status (4)
| Country | Link |
|---|---|
| EP (1) | EP3386944A4 (de) |
| BR (1) | BR112018011437A2 (de) |
| CA (1) | CA3006537A1 (de) |
| WO (1) | WO2017098533A2 (de) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20220151986A1 (en) | 2020-11-18 | 2022-05-19 | Mind Medicine, Inc. | Mdma prodrugs to assist psychotherapy |
| EP4122914B1 (de) | 2021-07-22 | 2023-08-16 | SCI Pharmtech Inc | Verbindung und verfahren zur herstellung von lisdexamfetamin |
| US11608312B1 (en) | 2021-07-22 | 2023-03-21 | Sci Pharmtech Inc. | Compound and method for preparation of lisdexamfetamine |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2540678C (en) * | 2003-09-30 | 2011-02-22 | New River Pharmaceuticals Inc. | Pharmaceutical compositions for prevention of overdose or abuse |
| WO2010042120A1 (en) * | 2008-10-09 | 2010-04-15 | Archimica, Inc. | Process for the synthesis of amphetamine derivatives |
| US8614346B2 (en) * | 2009-06-19 | 2013-12-24 | Cambrex Charles City, Inc. | Methods and compositions for preparation of amphetamine conjugates and salts thereof |
| US8779191B2 (en) * | 2010-12-20 | 2014-07-15 | Cambrex Charles City, Inc. | Methods and compositions for preparing lisdexamfetamine and salts thereof |
| WO2013011526A1 (en) * | 2011-07-20 | 2013-01-24 | Ind-Swift Laboratories Limited | Process for preparation of lisdexamphetamine and salts thereof |
| WO2015130660A1 (en) * | 2014-02-25 | 2015-09-03 | Chemapotheca, Llc | Synthesis of racemic amphetamine derivatives by cuprate addition reaction with aziridine phosphoramidate compounds |
-
2016
- 2016-12-12 EP EP16872573.7A patent/EP3386944A4/de not_active Withdrawn
- 2016-12-12 CA CA3006537A patent/CA3006537A1/en not_active Abandoned
- 2016-12-12 WO PCT/IN2016/050441 patent/WO2017098533A2/en active Application Filing
- 2016-12-12 BR BR112018011437A patent/BR112018011437A2/pt not_active Application Discontinuation
Non-Patent Citations (1)
| Title |
|---|
| No further relevant documents disclosed * |
Also Published As
| Publication number | Publication date |
|---|---|
| CA3006537A1 (en) | 2017-06-15 |
| BR112018011437A2 (pt) | 2018-11-27 |
| WO2017098533A2 (en) | 2017-06-15 |
| EP3386944A2 (de) | 2018-10-17 |
| WO2017098533A3 (en) | 2017-08-10 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| STAA | Information on the status of an ep patent application or granted ep patent |
Free format text: STATUS: THE INTERNATIONAL PUBLICATION HAS BEEN MADE |
|
| PUAI | Public reference made under article 153(3) epc to a published international application that has entered the european phase |
Free format text: ORIGINAL CODE: 0009012 |
|
| STAA | Information on the status of an ep patent application or granted ep patent |
Free format text: STATUS: REQUEST FOR EXAMINATION WAS MADE |
|
| 17P | Request for examination filed |
Effective date: 20180626 |
|
| AK | Designated contracting states |
Kind code of ref document: A2 Designated state(s): AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR |
|
| AX | Request for extension of the european patent |
Extension state: BA ME |
|
| DAV | Request for validation of the european patent (deleted) | ||
| DAX | Request for extension of the european patent (deleted) | ||
| A4 | Supplementary search report drawn up and despatched |
Effective date: 20190725 |
|
| RIC1 | Information provided on ipc code assigned before grant |
Ipc: C07C 231/14 20060101ALI20190719BHEP Ipc: C07D 203/18 20060101AFI20190719BHEP Ipc: C07C 237/06 20060101ALI20190719BHEP |
|
| STAA | Information on the status of an ep patent application or granted ep patent |
Free format text: STATUS: THE APPLICATION IS DEEMED TO BE WITHDRAWN |
|
| 18D | Application deemed to be withdrawn |
Effective date: 20200225 |