EP1603881A4 - Substituierte thiophene mit antibakterieller wirksamkeit - Google Patents

Substituierte thiophene mit antibakterieller wirksamkeit

Info

Publication number
EP1603881A4
EP1603881A4 EP04715720A EP04715720A EP1603881A4 EP 1603881 A4 EP1603881 A4 EP 1603881A4 EP 04715720 A EP04715720 A EP 04715720A EP 04715720 A EP04715720 A EP 04715720A EP 1603881 A4 EP1603881 A4 EP 1603881A4
Authority
EP
European Patent Office
Prior art keywords
antibacterial activity
substituted thiophenes
thiophenes
substituted
antibacterial
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
EP04715720A
Other languages
English (en)
French (fr)
Other versions
EP1603881A2 (de
Inventor
John Berge
Richard Jarvest
Catherine S V Frydrych
Joseph Guiles
Jian Qiu
Theodore M Tarasow
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Crestone Inc
Original Assignee
Replidyne Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GBGB0304809.7A external-priority patent/GB0304809D0/en
Application filed by Replidyne Inc filed Critical Replidyne Inc
Publication of EP1603881A2 publication Critical patent/EP1603881A2/de
Publication of EP1603881A4 publication Critical patent/EP1603881A4/de
Withdrawn legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
EP04715720A 2003-03-03 2004-02-27 Substituierte thiophene mit antibakterieller wirksamkeit Withdrawn EP1603881A4 (de)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
GBGB0304809.7A GB0304809D0 (en) 2003-03-03 2003-03-03 Novel compounds
GB0304809 2003-03-03
US52722903P 2003-12-05 2003-12-05
US527229P 2003-12-05
PCT/US2004/005930 WO2004078119A2 (en) 2003-03-03 2004-02-27 Substituted thiophenes with antibacterial activity

Publications (2)

Publication Number Publication Date
EP1603881A2 EP1603881A2 (de) 2005-12-14
EP1603881A4 true EP1603881A4 (de) 2010-07-07

Family

ID=32964063

Family Applications (1)

Application Number Title Priority Date Filing Date
EP04715720A Withdrawn EP1603881A4 (de) 2003-03-03 2004-02-27 Substituierte thiophene mit antibakterieller wirksamkeit

Country Status (5)

Country Link
EP (1) EP1603881A4 (de)
JP (1) JP2006519261A (de)
AU (2) AU2004218481A1 (de)
CA (1) CA2517523A1 (de)
WO (1) WO2004078119A2 (de)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1619947A4 (de) * 2003-05-01 2006-05-31 Replidyne Inc Antibakterielle verfahren und zusammensetzungen
US7973050B2 (en) 2006-09-26 2011-07-05 Crestone, Inc. Enantiomeric compounds with antibacterial activity
WO2008039642A2 (en) 2006-09-26 2008-04-03 Replidyne, Inc. Methods and compounds for treatment of clostridium based infection
US8697720B2 (en) 2006-09-26 2014-04-15 Crestone, Inc. Substituted phenylether-thienopyridone compounds with antibacterial activity
US7994192B2 (en) 2006-09-26 2011-08-09 Crestone, Inc. Substituted thienopyridone compounds with antibacterial activity

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2004052288A2 (en) * 2002-12-06 2004-06-24 Replidyne, Inc. 2-nh-heteroarylimidazoles with antibacterial activity
WO2005009336A2 (en) * 2003-05-01 2005-02-03 Replidyne, Inc. Antibacterial methods and compositions

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL138906A0 (en) * 1998-04-29 2001-11-25 Smithkline Beecham Plc Quinolones used as mrs inhibitors and bactericides
AU5213300A (en) * 1999-05-19 2000-12-12 Smithkline Beecham Plc 2-nh-pyridones and pyrimidones as mrs inhibitors
GB9911594D0 (en) * 1999-05-19 1999-07-21 Smithkline Beecham Plc Novel compounds

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2004052288A2 (en) * 2002-12-06 2004-06-24 Replidyne, Inc. 2-nh-heteroarylimidazoles with antibacterial activity
WO2005009336A2 (en) * 2003-05-01 2005-02-03 Replidyne, Inc. Antibacterial methods and compositions

Non-Patent Citations (2)

* Cited by examiner, † Cited by third party
Title
DATABASE CA [online] CHEMICAL ABSTRACTS SERVICE, COLUMBUS, OHIO, US; 2004, BERGE, JOHN ET AL: "Preparation of 2-aminoheteroarylimidazoles with antibacterial activity", XP002582745, retrieved from STN Database accession no. 2004:513484 *
See also references of WO2004078119A2 *

Also Published As

Publication number Publication date
EP1603881A2 (de) 2005-12-14
AU2011201854A1 (en) 2011-05-19
WO2004078119A2 (en) 2004-09-16
WO2004078119A3 (en) 2004-12-29
JP2006519261A (ja) 2006-08-24
AU2004218481A1 (en) 2004-09-16
CA2517523A1 (en) 2004-09-16

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Legal Events

Date Code Title Description
PUAI Public reference made under article 153(3) epc to a published international application that has entered the european phase

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17P Request for examination filed

Effective date: 20050928

AK Designated contracting states

Kind code of ref document: A2

Designated state(s): AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IT LI LU MC NL PT RO SE SI SK TR

AX Request for extension of the european patent

Extension state: AL LT LV MK

DAX Request for extension of the european patent (deleted)
RIC1 Information provided on ipc code assigned before grant

Ipc: C07D 409/12 20060101ALI20100521BHEP

Ipc: A61K 31/505 20060101ALI20100521BHEP

Ipc: A61K 31/415 20060101ALI20100521BHEP

Ipc: A61K 31/47 20060101ALI20100521BHEP

Ipc: C07D 495/04 20060101ALI20100521BHEP

Ipc: C07D 235/22 20060101ALI20100521BHEP

Ipc: C07D 215/233 20060101AFI20050118BHEP

A4 Supplementary search report drawn up and despatched

Effective date: 20100608

RAP1 Party data changed (applicant data changed or rights of an application transferred)

Owner name: QIU, JIAN

Owner name: CRESTONE, INC.

RAP1 Party data changed (applicant data changed or rights of an application transferred)

Owner name: CRESTONE, INC.

17Q First examination report despatched

Effective date: 20110803

GRAP Despatch of communication of intention to grant a patent

Free format text: ORIGINAL CODE: EPIDOSNIGR1

RIC1 Information provided on ipc code assigned before grant

Ipc: A61P 31/04 20060101ALI20130626BHEP

Ipc: C07D 409/12 20060101ALI20130626BHEP

Ipc: A61K 31/505 20060101ALI20130626BHEP

Ipc: C07D 215/233 20060101AFI20130626BHEP

Ipc: A61K 31/415 20060101ALI20130626BHEP

Ipc: C07D 495/04 20060101ALI20130626BHEP

Ipc: A61K 31/47 20060101ALI20130626BHEP

Ipc: C07D 235/22 20060101ALI20130626BHEP

INTG Intention to grant announced

Effective date: 20130709

RIN1 Information on inventor provided before grant (corrected)

Inventor name: FRYDRYCH, CATHERINE, S. V.

Inventor name: JARVEST, RICHARD

Inventor name: BERGE, JOHN

Inventor name: TARASOW, THEODORE, M.

Inventor name: GUILES, JOSEPH

Inventor name: QIU, JIAN

STAA Information on the status of an ep patent application or granted ep patent

Free format text: STATUS: THE APPLICATION IS DEEMED TO BE WITHDRAWN

18D Application deemed to be withdrawn

Effective date: 20131120