EP1237851A4 - SELS D'ACIDE CARBOXYLIQUE i Cis /i -4-CYANO-4- 3-(CYCLOPENTYLOXY)-4-METHOXYPHENYL]CYCLOHEXANE-1 - Google Patents
SELS D'ACIDE CARBOXYLIQUE i Cis /i -4-CYANO-4- 3-(CYCLOPENTYLOXY)-4-METHOXYPHENYL]CYCLOHEXANE-1Info
- Publication number
- EP1237851A4 EP1237851A4 EP00989266A EP00989266A EP1237851A4 EP 1237851 A4 EP1237851 A4 EP 1237851A4 EP 00989266 A EP00989266 A EP 00989266A EP 00989266 A EP00989266 A EP 00989266A EP 1237851 A4 EP1237851 A4 EP 1237851A4
- Authority
- EP
- European Patent Office
- Prior art keywords
- cyclopentyloxy
- methoxyphenyl
- cis
- cyclohexane
- cyano
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C215/00—Compounds containing amino and hydroxy groups bound to the same carbon skeleton
- C07C215/02—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton
- C07C215/04—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being saturated
- C07C215/06—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being saturated and acyclic
- C07C215/10—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being saturated and acyclic with one amino group and at least two hydroxy groups bound to the carbon skeleton
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C211/00—Compounds containing amino groups bound to a carbon skeleton
- C07C211/01—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to acyclic carbon atoms
- C07C211/02—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton
- C07C211/09—Diamines
- C07C211/10—Diaminoethanes
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C255/00—Carboxylic acid nitriles
- C07C255/45—Carboxylic acid nitriles having cyano groups bound to carbon atoms of rings other than six-membered aromatic rings
- C07C255/46—Carboxylic acid nitriles having cyano groups bound to carbon atoms of rings other than six-membered aromatic rings to carbon atoms of non-condensed rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2601/00—Systems containing only non-condensed rings
- C07C2601/06—Systems containing only non-condensed rings with a five-membered ring
- C07C2601/08—Systems containing only non-condensed rings with a five-membered ring the ring being saturated
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2601/00—Systems containing only non-condensed rings
- C07C2601/12—Systems containing only non-condensed rings with a six-membered ring
- C07C2601/14—The ring being saturated
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Engineering & Computer Science (AREA)
- Pulmonology (AREA)
- Biomedical Technology (AREA)
- Rheumatology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Hospice & Palliative Care (AREA)
- Pain & Pain Management (AREA)
- Immunology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Physical Education & Sports Medicine (AREA)
- Psychiatry (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US17097799P | 1999-12-15 | 1999-12-15 | |
US170977P | 1999-12-15 | ||
PCT/US2000/033966 WO2001043692A2 (fr) | 1999-12-15 | 2000-12-15 | SELS D'ACIDE CARBOXYLIQUE Cis-4-CYANO-4-[3-(CYCLOPENTYLOXY)-4-METHOXYPHENYL]CYCLOHEXANE-1 |
Publications (2)
Publication Number | Publication Date |
---|---|
EP1237851A2 EP1237851A2 (fr) | 2002-09-11 |
EP1237851A4 true EP1237851A4 (fr) | 2004-06-23 |
Family
ID=22622045
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EP00989266A Withdrawn EP1237851A4 (fr) | 1999-12-15 | 2000-12-15 | SELS D'ACIDE CARBOXYLIQUE i Cis /i -4-CYANO-4- 3-(CYCLOPENTYLOXY)-4-METHOXYPHENYL]CYCLOHEXANE-1 |
Country Status (3)
Country | Link |
---|---|
EP (1) | EP1237851A4 (fr) |
JP (1) | JP2003534238A (fr) |
WO (1) | WO2001043692A2 (fr) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AR024076A1 (es) * | 1999-05-25 | 2002-09-04 | Smithkline Beecham Corp | Sales de cis-[4-ciano-4-(3-ciclopentiloxi-4-metoxifenil) ciclohexan-1-carboxilato] |
KR101743783B1 (ko) * | 2008-12-08 | 2017-06-05 | 글락소스미스클라인 엘엘씨 | 신규 화합물 |
Citations (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO1999018793A1 (fr) * | 1997-10-10 | 1999-04-22 | Smithkline Beecham Corporation | Procede de preparation d'acides 4-phenyl-4-cyanocyclohexanoiques substitues |
WO2000071114A1 (fr) * | 1999-05-25 | 2000-11-30 | Smithkline Beecham Corporation | Sels de cis-¢4-cyano-4-(3-cyclopentyloxy-4-methoxyphenyle) cyclohexane-1-carboxylate! |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
UY25338A1 (es) * | 1998-01-07 | 2001-08-27 | Smithkline Beecham Corp | Método para tratar copd |
-
2000
- 2000-12-15 EP EP00989266A patent/EP1237851A4/fr not_active Withdrawn
- 2000-12-15 JP JP2001544633A patent/JP2003534238A/ja not_active Withdrawn
- 2000-12-15 WO PCT/US2000/033966 patent/WO2001043692A2/fr not_active Application Discontinuation
Patent Citations (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO1999018793A1 (fr) * | 1997-10-10 | 1999-04-22 | Smithkline Beecham Corporation | Procede de preparation d'acides 4-phenyl-4-cyanocyclohexanoiques substitues |
WO2000071114A1 (fr) * | 1999-05-25 | 2000-11-30 | Smithkline Beecham Corporation | Sels de cis-¢4-cyano-4-(3-cyclopentyloxy-4-methoxyphenyle) cyclohexane-1-carboxylate! |
Non-Patent Citations (1)
Title |
---|
See also references of WO0143692A3 * |
Also Published As
Publication number | Publication date |
---|---|
JP2003534238A (ja) | 2003-11-18 |
EP1237851A2 (fr) | 2002-09-11 |
WO2001043692A3 (fr) | 2002-03-07 |
WO2001043692A2 (fr) | 2001-06-21 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
PL335027A1 (en) | Derivatives of arylsulphonylamino hydroxamic acid | |
ZA200004725B (en) | Process for the fermentative preparation of D-pantothenic acid using coryneform bacteria. | |
AU2754501A (en) | Treatment of acne using lipoic acid | |
IL147216A0 (en) | Arylsulfonamido-substituted hydroxamic acid derivatives | |
AU5925200A (en) | Control of dc/dc converters having synchronous rectifiers | |
EP1408991A4 (fr) | Aerosol nasal a base de sels de la mer morte | |
HUP0202283A2 (en) | Process for the preparation of basic antibiotic-inorganic acid addition salts and intermediate oxalates | |
EP1237851A4 (fr) | SELS D'ACIDE CARBOXYLIQUE i Cis /i -4-CYANO-4- 3-(CYCLOPENTYLOXY)-4-METHOXYPHENYL]CYCLOHEXANE-1 | |
AU2233001A (en) | Preparation method of methacrylic acid | |
AU2001256324A1 (en) | Process for the preparation of alkaline earth salts of d-pantothenic acid | |
GB9929979D0 (en) | Hydroxamic acid derivatives | |
IL138316A0 (en) | Process for the fermentative preparation of d-pantothenic acid using coryneform bacteria | |
AU2002303210A1 (en) | Pharmacologically active strong acid solutions | |
PL351945A1 (en) | Salts of cis [4-cyano-4-(cyclopentyloxy-4-methoxyphenyl) cyclohexan-1-carboxylan] | |
AU6525700A (en) | Reductive combustion of ammonium salts of sulfuric acid | |
AU7608100A (en) | 1-cyclohexene-1-carboxylic acid and 1-cyclohexene-1-carboxylates as neuraminidase inhibitors | |
AU2967100A (en) | Hypertonic aqueous solutions of polybasic acid salts | |
GB9911071D0 (en) | Hydroxamic and carboxylic acid derivatives | |
EP1250313A4 (fr) | Cis-lithium-cyano-4- 3-(cyclopentyloxy)-4-methoxyphenyl]cyclohexanecarboxylate monohydrate | |
GB9907082D0 (en) | The preparation of carboxylic acid derivatives | |
AU2003224361A1 (en) | Hepatoprotective activity of 2'-p-hydroxybenzoylmussaenosidic acid | |
IL144946A0 (en) | Method of detecting shikimic acid | |
SI1250313T1 (sl) | Monohidrat cis-litij-ciano-4(3-(ciklopentiloksi)-4-metoksifenil) cikloheksankarboksilata | |
AU2001285881A1 (en) | Process for the fermentative preparation of d-pantothenic acid using coryneform bacteria | |
GB9911073D0 (en) | Hydroxamic and carboxylic acid derivatives |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
PUAI | Public reference made under article 153(3) epc to a published international application that has entered the european phase |
Free format text: ORIGINAL CODE: 0009012 |
|
17P | Request for examination filed |
Effective date: 20020625 |
|
AK | Designated contracting states |
Kind code of ref document: A2 Designated state(s): AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE TR |
|
A4 | Supplementary search report drawn up and despatched |
Effective date: 20040507 |
|
RIC1 | Information provided on ipc code assigned before grant |
Ipc: 7C 07C 255/46 B Ipc: 7C 07C 215/10 B Ipc: 7C 07C 211/10 B Ipc: 7C 07C 255/00 A |
|
STAA | Information on the status of an ep patent application or granted ep patent |
Free format text: STATUS: THE APPLICATION IS DEEMED TO BE WITHDRAWN |
|
18D | Application deemed to be withdrawn |
Effective date: 20040722 |
|
RTI1 | Title (correction) |
Free format text: SALTS OF I CIS /I -4-CYANO-4- 3-(CYCLOPENTYLOXY)-4-METHOXYPHENYL CYCLOHEXANE-1-CARBOXYLIC ACID |