EP0480693A3 - Avermectin degradation products and derivatives - Google Patents

Avermectin degradation products and derivatives Download PDF

Info

Publication number
EP0480693A3
EP0480693A3 EP19910309252 EP91309252A EP0480693A3 EP 0480693 A3 EP0480693 A3 EP 0480693A3 EP 19910309252 EP19910309252 EP 19910309252 EP 91309252 A EP91309252 A EP 91309252A EP 0480693 A3 EP0480693 A3 EP 0480693A3
Authority
EP
European Patent Office
Prior art keywords
avermectin
derivatives
degradation products
degradation
products
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
EP19910309252
Other versions
EP0480693A2 (en
Inventor
Thomas L. Shih
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Merck and Co Inc
Original Assignee
Merck and Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck and Co Inc filed Critical Merck and Co Inc
Publication of EP0480693A2 publication Critical patent/EP0480693A2/en
Publication of EP0480693A3 publication Critical patent/EP0480693A3/en
Withdrawn legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/01—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Public Health (AREA)
  • Biochemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Saccharide Compounds (AREA)
EP19910309252 1990-10-11 1991-10-09 Avermectin degradation products and derivatives Withdrawn EP0480693A3 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US59587290A 1990-10-11 1990-10-11
US595872 1990-10-11

Publications (2)

Publication Number Publication Date
EP0480693A2 EP0480693A2 (en) 1992-04-15
EP0480693A3 true EP0480693A3 (en) 1992-06-17

Family

ID=24385037

Family Applications (1)

Application Number Title Priority Date Filing Date
EP19910309252 Withdrawn EP0480693A3 (en) 1990-10-11 1991-10-09 Avermectin degradation products and derivatives

Country Status (5)

Country Link
EP (1) EP0480693A3 (en)
JP (1) JPH05202057A (en)
AU (1) AU8574691A (en)
CA (1) CA2052860A1 (en)
ZA (1) ZA918072B (en)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6010490A (en) * 1992-12-18 2000-01-04 The Procter & Gamble Company Absorbent article having an upstanding transverse partition
GB9300883D0 (en) * 1993-01-18 1993-03-10 Pfizer Ltd Antiparasitic agents
US5981500A (en) * 1994-01-12 1999-11-09 Pfizer Inc. Antiparasitic agents related to the milbemycins and avermectins
JPWO2002012261A1 (en) 2000-08-09 2004-01-15 社団法人北里研究所 Evermectin derivative
CA2418975C (en) * 2000-08-09 2012-01-17 Satoshi Omura Avermectin derivatives
CN103421065B (en) * 2013-07-03 2016-05-18 大庆志飞生物化工有限公司 One class Novel Abamectin derivative and preparation method thereof
CN104402954A (en) * 2014-11-28 2015-03-11 大庆志飞生物化工有限公司 Methylaminoavermectin monosaccharide compound and preparing method and application thereof
CN104447920A (en) * 2014-11-28 2015-03-25 大庆志飞生物化工有限公司 Avermectin chloride as well as preparation method and application thereof
CN113030296B (en) * 2021-02-09 2023-03-21 上海市食品药品检验研究院 Method for screening abamectin and emamectin benzoate degradation products in honeysuckle and planting soil thereof

Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0194125A2 (en) * 1985-03-04 1986-09-10 Merck & Co. Inc. Avermectin bioconversion products
EP0215654A2 (en) * 1985-09-13 1987-03-25 American Cyanamid Company Macrolide antibiotics and their preparation
EP0264576A1 (en) * 1986-09-12 1988-04-27 American Cyanamid Company Delta 23-LL-F28249 compounds

Patent Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0194125A2 (en) * 1985-03-04 1986-09-10 Merck & Co. Inc. Avermectin bioconversion products
EP0215654A2 (en) * 1985-09-13 1987-03-25 American Cyanamid Company Macrolide antibiotics and their preparation
EP0264576A1 (en) * 1986-09-12 1988-04-27 American Cyanamid Company Delta 23-LL-F28249 compounds

Also Published As

Publication number Publication date
EP0480693A2 (en) 1992-04-15
AU8574691A (en) 1992-04-16
ZA918072B (en) 1992-08-26
JPH05202057A (en) 1993-08-10
CA2052860A1 (en) 1992-04-12

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