EP0165900A3 - Lactones, their preparation and their use as herbicides - Google Patents

Lactones, their preparation and their use as herbicides Download PDF

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Publication number
EP0165900A3
EP0165900A3 EP85810255A EP85810255A EP0165900A3 EP 0165900 A3 EP0165900 A3 EP 0165900A3 EP 85810255 A EP85810255 A EP 85810255A EP 85810255 A EP85810255 A EP 85810255A EP 0165900 A3 EP0165900 A3 EP 0165900A3
Authority
EP
European Patent Office
Prior art keywords
meaning
lactones
herbicides
preparation
oxygen
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
EP85810255A
Other languages
German (de)
French (fr)
Other versions
EP0165900A2 (en
Inventor
Urs Dr. Burckhardt
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Novartis AG
Original Assignee
Ciba Geigy AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ciba Geigy AG filed Critical Ciba Geigy AG
Publication of EP0165900A2 publication Critical patent/EP0165900A2/en
Publication of EP0165900A3 publication Critical patent/EP0165900A3/en
Withdrawn legal-status Critical Current

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/01—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics

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  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Wood Science & Technology (AREA)
  • Dentistry (AREA)
  • Plant Pathology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Molecular Biology (AREA)
  • Veterinary Medicine (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Milbemycin-Derivate der formel I mit der Bedeutung eines aliphatischen oder aromatischen restes oder eines Pyridylrings oder heterocyclischen sauer­ stoffhaltigen 5- oder 6-Rings, die allesamt auch über Sauer­ stoff gebunden sein können, für den substituenten R₁ und der Bedeutung von Methyl, Ethyl oder Isopropyl für R₂ dienen als Wirkstoff zur Bekämpfung von Arthropodenarten, wie Schadinsekten oder tierische Ekto- oder endoparasiten, und werden in Form von Mitteln angewandt. Die verbindun­ gen können auch als Zwischenprodukte zur weiteren Deriva­ tisierung von Milbemycinen eingesetzt werden. Milbemycin derivatives of the formula I with the meaning of an aliphatic or aromatic radical or a pyridyl ring or heterocyclic oxygen-containing 5- or 6-rings, all of which can also be bonded via oxygen, for the substituted R₁ and the meaning of methyl, ethyl or isopropyl for R₂ serve as the active ingredient to control arthropod species, such as insect pests or animal ecto- or endoparasites, and are used in the form of agents. The compounds can also be used as intermediates for the further derivatization of milbemycins.

EP85810255A 1984-06-08 1985-06-03 Lactones, their preparation and their use as herbicides Withdrawn EP0165900A3 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH280884 1984-06-08
CH2808/84 1984-06-08

Publications (2)

Publication Number Publication Date
EP0165900A2 EP0165900A2 (en) 1985-12-27
EP0165900A3 true EP0165900A3 (en) 1986-05-28

Family

ID=4242054

Family Applications (1)

Application Number Title Priority Date Filing Date
EP85810255A Withdrawn EP0165900A3 (en) 1984-06-08 1985-06-03 Lactones, their preparation and their use as herbicides

Country Status (8)

Country Link
US (1) US4791134A (en)
EP (1) EP0165900A3 (en)
JP (1) JPH0633274B2 (en)
AU (1) AU584337B2 (en)
CA (1) CA1254886A (en)
DK (1) DK256885A (en)
IL (1) IL75428A (en)
ZA (1) ZA854334B (en)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4582852A (en) * 1983-11-02 1986-04-15 Ciba-Geigy Corporation 14- and 15-hydroxy milbemycin derivatives for controlling plant and animal parasites
US4584314A (en) * 1983-11-25 1986-04-22 Ciba-Geigy Corporation Lactone derivative, process for the preparation thereof, and use thereof in pest control
EP0237482A1 (en) * 1986-03-06 1987-09-16 Ciba-Geigy Ag Derivatives of C(29)-carbonyloxy-milbemycine against parasites in animals and plants
NZ219467A (en) * 1986-03-07 1990-03-27 Ciba Geigy Ag 5-acyloxy 13b-alkyl milbemycins and parasiticidal compositions
US4855317A (en) * 1987-03-06 1989-08-08 Ciba-Geigy Corporation Insecticides and parasiticides
US4871719A (en) * 1987-03-24 1989-10-03 Ciba-Geigy Corporation Composition for controlling parasites in productive livestock
EP0285561A3 (en) * 1987-03-27 1989-10-25 Ciba-Geigy Ag Milbemycin derivatives with a paraciticidal and insecticidal activity
NZ593184A (en) 2008-12-04 2012-11-30 Merial Ltd Dimeric avermectin and milbemycin derivatives
WO2011075592A1 (en) 2009-12-17 2011-06-23 Merial Limited Compositions comprising macrocyclic lactone compounds and spirodioxepinoindoles
DK2785719T3 (en) 2011-12-02 2017-12-04 Merial Inc LONG-EFFECTIVE INJECTABLE MOXIDECTIN FORMULATIONS AND HIS UNKNOWN MOXIDECTIN CRYSTAL FORMS
PE20151726A1 (en) 2013-04-12 2015-11-18 Zoetis Services Llc STABLE VETERINARY FORMULATIONS OF COMBINATION OF MACROCYCLIC LACTONES AND IMIDAZOTHIAZOLES

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3950360A (en) * 1972-06-08 1976-04-13 Sankyo Company Limited Antibiotic substances
JPS5632481A (en) * 1979-08-23 1981-04-01 Sankyo Co Ltd Antibiotic b-41d, its preparation, and acaricide and anthelminthic agent and repellent containing the same as active constituent
JPS60126289A (en) * 1983-11-14 1985-07-05 Sankyo Co Ltd 5-carbonate derivative of milbemycin
US4584314A (en) * 1983-11-25 1986-04-22 Ciba-Geigy Corporation Lactone derivative, process for the preparation thereof, and use thereof in pest control

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
THE JOURNAL OF ANTIBIOTICS, Oktober 1980, Seiten 1120-1127; YO TAKIGUCHI et al.: "Milbemycins, a new family of macrolide antibiotics: fermentation, isolation and physico-chemical properties" *

Also Published As

Publication number Publication date
EP0165900A2 (en) 1985-12-27
IL75428A0 (en) 1985-10-31
US4791134A (en) 1988-12-13
CA1254886A (en) 1989-05-30
AU584337B2 (en) 1989-05-25
DK256885A (en) 1985-12-09
ZA854334B (en) 1986-01-29
IL75428A (en) 1988-04-29
AU4341885A (en) 1985-12-12
JPS611692A (en) 1986-01-07
JPH0633274B2 (en) 1994-05-02
DK256885D0 (en) 1985-06-07

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Legal Events

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PUAI Public reference made under article 153(3) epc to a published international application that has entered the european phase

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Effective date: 19850605

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PUAL Search report despatched

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Designated state(s): AT BE CH DE FR GB IT LI NL SE

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Effective date: 19890119

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18W Application withdrawn

Withdrawal date: 19890316

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Effective date: 19890316

RIN1 Information on inventor provided before grant (corrected)

Inventor name: BURCKHARDT, URS, DR.