ECSP992879A - PIRAZOLOPIRIMIDINAS AND PIRAZOLOTRIAZINAS - Google Patents
PIRAZOLOPIRIMIDINAS AND PIRAZOLOTRIAZINASInfo
- Publication number
- ECSP992879A ECSP992879A ECSP992879A ECSP992879A EC SP992879 A ECSP992879 A EC SP992879A EC SP992879 A ECSP992879 A EC SP992879A EC SP992879 A ECSP992879 A EC SP992879A
- Authority
- EC
- Ecuador
- Prior art keywords
- disease
- disorders
- depressions
- pirazolotriazinas
- pirazolopirimidinas
- Prior art date
Links
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
La presente invención se refiere a pirazolopirimidinas y pirazolotriazinas de la fórmula general (gráfico), y sus sales farmacéuticamente aceptables. Sorprendentemente, estos compuestos tienen una afinidad selectiva para los receptores de la 5HT-6. Son convenientemente adecuados para el tratamiento y prevención de trastornos nerviosos centrales tales como por ejemplo, psicosis, esquizofrenia, depresiones maniaticas, depresiones, trastornos neurológicos, trastornos de la memoria, enfermedad de Parkinson, esclerosis lateral amiotrófica, enfermedad de Alzheimer y corea de Huntington.The present invention relates to pyrazolopyrimidines and pyrazolotriazines of the general formula (graph), and their pharmaceutically acceptable salts. Surprisingly, these compounds have a selective affinity for 5HT-6 receptors. They are conveniently suitable for the treatment and prevention of central nervous disorders such as, for example, psychosis, schizophrenia, manic depressions, depressions, neurological disorders, memory disorders, Parkinson's disease, amyotrophic lateral sclerosis, Alzheimer's disease and Huntington's chorea.
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
ECSP992879 ECSP992879A (en) | 1999-03-09 | 1999-03-09 | PIRAZOLOPIRIMIDINAS AND PIRAZOLOTRIAZINAS |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
ECSP992879 ECSP992879A (en) | 1999-03-09 | 1999-03-09 | PIRAZOLOPIRIMIDINAS AND PIRAZOLOTRIAZINAS |
Publications (1)
Publication Number | Publication Date |
---|---|
ECSP992879A true ECSP992879A (en) | 2000-11-24 |
Family
ID=42043867
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ECSP992879 ECSP992879A (en) | 1999-03-09 | 1999-03-09 | PIRAZOLOPIRIMIDINAS AND PIRAZOLOTRIAZINAS |
Country Status (1)
Country | Link |
---|---|
EC (1) | ECSP992879A (en) |
-
1999
- 1999-03-09 EC ECSP992879 patent/ECSP992879A/en unknown
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