ECSP982672A - VITRONECTIN III RECEPTOR ANTAGONISTS - Google Patents
VITRONECTIN III RECEPTOR ANTAGONISTSInfo
- Publication number
- ECSP982672A ECSP982672A ECSP982672A ECSP982672A EC SP982672 A ECSP982672 A EC SP982672A EC SP982672 A ECSP982672 A EC SP982672A EC SP982672 A ECSP982672 A EC SP982672A
- Authority
- EC
- Ecuador
- Prior art keywords
- receptor antagonists
- alkyl
- vitronectin
- iii receptor
- halo
- Prior art date
Links
Abstract
Se describen compuestos de fórmula (I) que son antagonistas de receptores de vitronectina y son útiles en el tratamiento de osteoporosis: (gráfico), en la cual: A es Ch2 u o; R1 es H, halo o alquilo C1-6; R2 es H, alquilo C1-6 p Ch2NR¿¿R¿¿, X es 0 o CH2, Y es (gráfico), G es NR¿¿, SuO; R¿es H, alquilo C1-6, 0 alquilo C1-6, S-alquilo C1-6, Nr¿¿R¿¿ o halo; cada R¿¿es independientemente H alquilo C1-6; y o una sal farmacéuticamente aceptable de los mismos.Compounds of formula (I) are described which are vitronectin receptor antagonists and are useful in the treatment of osteoporosis: (graph), in which: A is Ch2 or o; R1 is H, halo or C1-6 alkyl; R2 is H, C1-6 alkyl p Ch2NR¿¿R¿¿, X is 0 or CH2, Y is (graph), G is NR¿¿, SuO; R¿ is H, C1-6 alkyl, 0 C1-6 alkyl, S-C1-6 alkyl, Nr¿¿R¿¿ or halo; each R¿¿is independently H C1-6alkyl; and or a pharmaceutically acceptable salt thereof.
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
ECSP982672 ECSP982672A (en) | 1998-09-18 | 1998-09-18 | VITRONECTIN III RECEPTOR ANTAGONISTS |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
ECSP982672 ECSP982672A (en) | 1998-09-18 | 1998-09-18 | VITRONECTIN III RECEPTOR ANTAGONISTS |
Publications (1)
Publication Number | Publication Date |
---|---|
ECSP982672A true ECSP982672A (en) | 1999-04-13 |
Family
ID=42043591
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ECSP982672 ECSP982672A (en) | 1998-09-18 | 1998-09-18 | VITRONECTIN III RECEPTOR ANTAGONISTS |
Country Status (1)
Country | Link |
---|---|
EC (1) | ECSP982672A (en) |
-
1998
- 1998-09-18 EC ECSP982672 patent/ECSP982672A/en unknown
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