ECSP982568A - FARNESIL PROTEIN TRANSFERASE INHIBITORS - Google Patents

FARNESIL PROTEIN TRANSFERASE INHIBITORS

Info

Publication number
ECSP982568A
ECSP982568A ECSP982568A ECSP982568A EC SP982568 A ECSP982568 A EC SP982568A EC SP982568 A ECSP982568 A EC SP982568A EC SP982568 A ECSP982568 A EC SP982568A
Authority
EC
Ecuador
Prior art keywords
protein transferase
transferase inhibitors
farnesil
compounds
useful
Prior art date
Application number
Other languages
Spanish (es)
Inventor
Rajeev S Bhide
John T Hunt
Katerina Leftheris
Charles Z Ding
Soong-Hoon Kim
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Priority to ECSP982568 priority Critical patent/ECSP982568A/en
Publication of ECSP982568A publication Critical patent/ECSP982568A/en

Links

Abstract

Se describen derivados de quinolina y benzazepina que inhibe la farnesil-proteína transferasa (ftasa) y la farnesilación de la proteína oncogénica Ras. De esta manera los compuestos son útiles como agentes anticáncer. Los compuestos también son útiles en el tratamiento de enfermedades diferentes del cáncer.Quinoline and benzazepine derivatives that inhibit farnesyl protein transferase (phthase) and farnesylation of the oncogenic protein Ras are described. In this way the compounds are useful as anticancer agents. The compounds are also useful in the treatment of diseases other than cancer.

ECSP982568 1998-06-30 1998-06-30 FARNESIL PROTEIN TRANSFERASE INHIBITORS ECSP982568A (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
ECSP982568 ECSP982568A (en) 1998-06-30 1998-06-30 FARNESIL PROTEIN TRANSFERASE INHIBITORS

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
ECSP982568 ECSP982568A (en) 1998-06-30 1998-06-30 FARNESIL PROTEIN TRANSFERASE INHIBITORS

Publications (1)

Publication Number Publication Date
ECSP982568A true ECSP982568A (en) 1999-01-26

Family

ID=42043488

Family Applications (1)

Application Number Title Priority Date Filing Date
ECSP982568 ECSP982568A (en) 1998-06-30 1998-06-30 FARNESIL PROTEIN TRANSFERASE INHIBITORS

Country Status (1)

Country Link
EC (1) ECSP982568A (en)

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