ECSP961919A - INTERMEDIATE PROCEDURES TO PREPARE 3- (1- PIPERAZINYL) - 1,2 BENZOISOTIAZOLE - Google Patents

INTERMEDIATE PROCEDURES TO PREPARE 3- (1- PIPERAZINYL) - 1,2 BENZOISOTIAZOLE

Info

Publication number
ECSP961919A
ECSP961919A ECSP961919A ECSP961919A EC SP961919 A ECSP961919 A EC SP961919A EC SP961919 A ECSP961919 A EC SP961919A EC SP961919 A ECSP961919 A EC SP961919A
Authority
EC
Ecuador
Prior art keywords
piperazinyl
benzoisotiazole
prepare
intermediate procedures
benzoisothiazole
Prior art date
Application number
Other languages
Spanish (es)
Inventor
Darrell E Fox
John Francis Lambert
Terry G Sinay Jr
Stanley W Walinsky
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Priority to ECSP961919 priority Critical patent/ECSP961919A/en
Publication of ECSP961919A publication Critical patent/ECSP961919A/en

Links

Landscapes

  • Thiazole And Isothizaole Compounds (AREA)

Abstract

La presente invención se refiere a procedimientos para la preparación de 3-(1-piperazinil) -1,2- benzoisotiazol o sus sales farmacéuticamente aceptables y a nuevos intermedios usados en el procedimiento. El 3-(1-piperazinil)-1,2-benzoisotiazol es un intermedio calve útil para la preparación de ziprasidona.The present invention relates to processes for the preparation of 3- (1-piperazinyl) -1,2-benzoisothiazole or its pharmaceutically acceptable salts and to new intermediates used in the process. 3- (1-piperazinyl) -1,2-benzoisothiazole is a useful key intermediate for the preparation of ziprasidone.

ECSP961919 1996-11-01 1996-11-01 INTERMEDIATE PROCEDURES TO PREPARE 3- (1- PIPERAZINYL) - 1,2 BENZOISOTIAZOLE ECSP961919A (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
ECSP961919 ECSP961919A (en) 1996-11-01 1996-11-01 INTERMEDIATE PROCEDURES TO PREPARE 3- (1- PIPERAZINYL) - 1,2 BENZOISOTIAZOLE

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
ECSP961919 ECSP961919A (en) 1996-11-01 1996-11-01 INTERMEDIATE PROCEDURES TO PREPARE 3- (1- PIPERAZINYL) - 1,2 BENZOISOTIAZOLE

Publications (1)

Publication Number Publication Date
ECSP961919A true ECSP961919A (en) 1997-10-17

Family

ID=42042645

Family Applications (1)

Application Number Title Priority Date Filing Date
ECSP961919 ECSP961919A (en) 1996-11-01 1996-11-01 INTERMEDIATE PROCEDURES TO PREPARE 3- (1- PIPERAZINYL) - 1,2 BENZOISOTIAZOLE

Country Status (1)

Country Link
EC (1) ECSP961919A (en)

Similar Documents

Publication Publication Date Title
ATE346039T1 (en) SULFONAMIDO-SUBSTITUTED BRIDGED BICYCLOALKYL DERIVATIVES
DK154287D0 (en) SUBSTITUTED OXADIAZOL DERIVATIVES, PROCEDURES FOR THE PRODUCTION THEREOF AND INTERMEDIATES FOR USE BY THE PROCEDURE AND MEDICINAL CONTAINING THE OXADIAZOLES
LU91083I2 (en) Bortezomib or one of the pharmaceutically acceptable esters, optionally in the form of a pharmaceutically acceptable salt-Velcade.
AR008853A1 (en) NEW PHARMACEUTICALLY ACTIVE COMPOUNDS, THEIR USE IN THE MANUFACTURE OF MEDICINES, TREATMENT METHOD, PHARMACEUTICAL COMPOSITION, INTERMEDIATE COMPOUNDS AND PROCESS FOR THE MANUFACTURE OF SUCH COMPOUNDS
CO4940465A1 (en) SALT MESYLATE TRIHYDRATE 5- (2- (4- (1,2-BENZOISOTIAZOL-3- IL) -1-PIPERAZINIL) ETIL) -6-CHLORINE-1,3-DIHYDRO-2H-INDOL-2-ONA
MY134129A (en) Polymorphs of an epothilone analog
ES2097908T3 (en) NEW BENZOPYRANONES, PROCEDURE FOR THEIR PREPARATION AND USE.
PT766668E (en) PROCESSES FOR THE PREPARATION OF ANTIBODIES AND HYDRATE OF ANTIHISTAMINIC DERIVATIVES OF PIPERIDINE AND POLYMORPHES AND PSEUDOMORPHES OF THESE
DK0776324T3 (en) Endothelin antagonists
SV2003000633A (en) NEW TIADIAZOLS AND OXADIAZOLS AND THEIR USE AS INHIBITORS OF PHOSPHODIESTERASA-7
NO941884L (en) 1,3-substituted cycloalkenes and cycloalkanes as central nervous system agents
DK0675717T3 (en) Use of 2-amino-6-n-propylamino-4,5,6,7-tetrahydrobenzothiazole (pramipexole) as a drug with antidepressant effect
DK0841851T3 (en) Fungicidal mixtures
EE03953B1 (en) Use of 2-Phenyl-1,2-benzisoselenazole-3 (2H) -one in the preparation of a pharmaceutical preparation for the treatment of Alzheimer's disease
AR004279A1 (en) PROCEDURES FOR PREPARING 3- (1-PIPERAZINYL) -1,2-BENZOISOTIAZOLE
PT790236E (en) 5- (2- (4- (1,2-BENZISOYZAZOL-3-YL) -1-PYRAZAZYL) -ETHYL-6-CHLORO-1,3-DIHYDRO-2H-INDOL-2-ONA
ECSP961919A (en) INTERMEDIATE PROCEDURES TO PREPARE 3- (1- PIPERAZINYL) - 1,2 BENZOISOTIAZOLE
BR0016941A (en) Aminomethyl-phenyl-cyclohexanone derivatives
FI92199B (en) A process for the preparation of new therapeutically useful chromium derivatives
ATE189894T1 (en) NAPHTHAMIDE DERIVATIVES OF 3-BETA-AMINO AZABICYCLOOCTAN OR NONANE AS ANTIPSYCHOTIC DRUGS
DK599686D0 (en) TRICYCLIC PYRIDON DERIVATIVES, THEIR PREPARATION AND USE OF THE PREPARATION, AND THE USE OF THE PRESENT APPLICABLE MATERIALS
DE69430074T2 (en) ANALGETIC 4-ARYLISOINDOLS
ES2190499T3 (en) USE OF BRADIQUININE ANTAGONISTS FOR THE PREPARATION OF MEDICINES FOR THE TREATMENT AND PREVENTION OF ALZHEIMER'S DISEASE.
BR9810031A (en) Pyrrolidine carboxylic acid derivatives as endothelin antagonists
AR001772A1 (en) Process for preparing (5-hydroxypyrazole-4-yl) carbonyl-thiochroman, y1-oxide or 1,1-dioxide compounds and intermediates for application in said process and processes to obtain said intermediates