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Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur
(AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds
(AREA)
Abstract
Se refiere a una serie de derivados tetracíclicos, a procesos para su preparación, a composiciones farmacéuticas que los contienen y a su uso como agentes terapéuticos. En particular la invención se refiere a derivados tetraciclicos los cuales son inhibidores potentes y selectivos, adecuados para el tratamiento de desórdenes cardiovasculares.It refers to a series of tetracyclic derivatives, to processes for their preparation, to pharmaceutical compositions containing them and to their use as therapeutic agents. In particular the invention relates to tetracyclic derivatives which are potent and selective inhibitors, suitable for the treatment of cardiovascular disorders.
ECSP9513671995-01-171995-01-17
TETRACICLIC DERIVATIVES PROCESSES FOR ITS PREPARATION AND USE
ECSP951367A
(en)
DERIVATIVES OF FITTED HETERO-PENTACICLO-FENILO, PHARMACEUTICAL COMPOSITION THAT UNDERSTANDS AND USES TO PREPARE A USEFUL MEDICINAL PRODUCT FOR THE TREATMENT OF A CONDITION MEDIATED BY P38
TETRACICLIC DERIVATIVES, THEIR USE IN THE PREPARATION OF A MEDICINAL PRODUCT, A TREATMENT METHOD, A PHARMACEUTICAL COMPOSITION AND PROCESSES FOR THE PREPARATION OF A PHARMACEUTICAL COMPOSITION AND TO PREPARE THE COMPOUNDS.
ADAMANTAN DERIVATIVES, PROCEDURES FOR THE PREPARATION, PHARMACEUTICAL COMPOSITION, PROCEDURE FOR THE PREPARATION OF PHARMACEUTICAL COMPOSITION, AND THE USE OF SUCH DERIVATIVES FOR THE MANUFACTURE OF MEDICINES
DERIVATIVES OF TER.-BUTIL- (7-METHYL-IMIDAZO [1,2, a] PIRIDIN-3-IL) -AMINA, PROCEDURE FOR THEIR PREPARATION, DRUGS THAT CONTAIN THEM, THEIR USE FOR THE PREPARATION OF A MEDICATION FOR THE INHIBITION OF NON-SYNTHEASE AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
DERIVATIVES OF BENZOCONDENSED HETEROARILAMIDE OF USEFUL TIENOPIRIDINS AS THERAPEUTIC AGENTS, PHARMACEUTICAL COMPOSITIONS THAT INCLUDE THE SAME AND METHOD FOR USE
ANALOG COMPOUNDS OF (1R, CIS) -4- (6-AMINO-9H-PURIN-9-IL) -2-CYCLOPENTENE-1-METHANOL, PROCESS FOR PREPARATION, USE IN THE TREATMENT OF VIRAL INFECTIONS, AND PACKING THAT CONTAINS THEM
DERIVATIVES OF PIPERAZINE, PROCEDURES TO PREPARE THEM, THE PHARMACEUTICAL COMPOSITIONS THAT CONTAIN THEM, THEIR USE AS A MEDICINAL PRODUCT AND THE METHOD FOR TREATING DISEASES MEDIATED BY TACHININ.