ECSP22003596A - NMDA RECEPTOR MODULATORS - Google Patents
NMDA RECEPTOR MODULATORSInfo
- Publication number
- ECSP22003596A ECSP22003596A ECSENADI20223596A ECDI202203596A ECSP22003596A EC SP22003596 A ECSP22003596 A EC SP22003596A EC SENADI20223596 A ECSENADI20223596 A EC SENADI20223596A EC DI202203596 A ECDI202203596 A EC DI202203596A EC SP22003596 A ECSP22003596 A EC SP22003596A
- Authority
- EC
- Ecuador
- Prior art keywords
- nmda receptor
- receptor modulators
- compounds
- depression
- disorders
- Prior art date
Links
Classifications
-
- B—PERFORMING OPERATIONS; TRANSPORTING
- B62—LAND VEHICLES FOR TRAVELLING OTHERWISE THAN ON RAILS
- B62D—MOTOR VEHICLES; TRAILERS
- B62D15/00—Steering not otherwise provided for
- B62D15/02—Steering position indicators ; Steering position determination; Steering aids
- B62D15/027—Parking aids, e.g. instruction means
- B62D15/0285—Parking performed automatically
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
- A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- B—PERFORMING OPERATIONS; TRANSPORTING
- B60—VEHICLES IN GENERAL
- B60W—CONJOINT CONTROL OF VEHICLE SUB-UNITS OF DIFFERENT TYPE OR DIFFERENT FUNCTION; CONTROL SYSTEMS SPECIALLY ADAPTED FOR HYBRID VEHICLES; ROAD VEHICLE DRIVE CONTROL SYSTEMS FOR PURPOSES NOT RELATED TO THE CONTROL OF A PARTICULAR SUB-UNIT
- B60W30/00—Purposes of road vehicle drive control systems not related to the control of a particular sub-unit, e.g. of systems using conjoint control of vehicle sub-units, or advanced driver assistance systems for ensuring comfort, stability and safety or drive control systems for propelling or retarding the vehicle
- B60W30/06—Automatic manoeuvring for parking
-
- B—PERFORMING OPERATIONS; TRANSPORTING
- B60—VEHICLES IN GENERAL
- B60W—CONJOINT CONTROL OF VEHICLE SUB-UNITS OF DIFFERENT TYPE OR DIFFERENT FUNCTION; CONTROL SYSTEMS SPECIALLY ADAPTED FOR HYBRID VEHICLES; ROAD VEHICLE DRIVE CONTROL SYSTEMS FOR PURPOSES NOT RELATED TO THE CONTROL OF A PARTICULAR SUB-UNIT
- B60W60/00—Drive control systems specially adapted for autonomous road vehicles
- B60W60/001—Planning or execution of driving tasks
-
- B—PERFORMING OPERATIONS; TRANSPORTING
- B60—VEHICLES IN GENERAL
- B60W—CONJOINT CONTROL OF VEHICLE SUB-UNITS OF DIFFERENT TYPE OR DIFFERENT FUNCTION; CONTROL SYSTEMS SPECIALLY ADAPTED FOR HYBRID VEHICLES; ROAD VEHICLE DRIVE CONTROL SYSTEMS FOR PURPOSES NOT RELATED TO THE CONTROL OF A PARTICULAR SUB-UNIT
- B60W2510/00—Input parameters relating to a particular sub-units
- B60W2510/20—Steering systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/07—Optical isomers
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Biomedical Technology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pain & Pain Management (AREA)
- General Chemical & Material Sciences (AREA)
- Psychiatry (AREA)
- Transportation (AREA)
- Mechanical Engineering (AREA)
- Automation & Control Theory (AREA)
- Epidemiology (AREA)
- Combustion & Propulsion (AREA)
- Human Computer Interaction (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
La presente invención se refiere a nuevos moduladores del receptor de NMDA. Aspectos separados de las invenciones se refieren a composiciones farmacéuticas que comprenden dichos compuestos y a usos de los compuestos para tratar trastornos neurológicos o trastornos neuropsiquiátricos tales como la depresión.The present invention relates to new NMDA receptor modulators. Separate aspects of the inventions relate to pharmaceutical compositions comprising said compounds and to uses of the compounds for treating neurological disorders or neuropsychiatric disorders such as depression.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DKPA201900821 | 2019-07-03 |
Publications (1)
Publication Number | Publication Date |
---|---|
ECSP22003596A true ECSP22003596A (en) | 2022-02-25 |
Family
ID=74065626
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ECSENADI20223596A ECSP22003596A (en) | 2019-07-03 | 2022-01-17 | NMDA RECEPTOR MODULATORS |
Country Status (20)
Country | Link |
---|---|
US (1) | US11466027B2 (en) |
EP (1) | EP3994141A1 (en) |
JP (1) | JP2022539197A (en) |
KR (1) | KR20220029568A (en) |
CN (1) | CN114008054A (en) |
AR (1) | AR119340A1 (en) |
AU (1) | AU2020299992A1 (en) |
BR (1) | BR112021003928A2 (en) |
CA (1) | CA3144304A1 (en) |
CL (1) | CL2021003557A1 (en) |
CO (1) | CO2021017142A2 (en) |
CR (1) | CR20210662A (en) |
EC (1) | ECSP22003596A (en) |
IL (1) | IL289575A (en) |
JO (1) | JOP20210331A1 (en) |
MA (1) | MA56451A (en) |
MX (1) | MX2021015742A (en) |
PE (1) | PE20220137A1 (en) |
TW (1) | TW202116779A (en) |
WO (1) | WO2021001423A1 (en) |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US11358971B2 (en) | 2019-07-03 | 2022-06-14 | H. Lundbeck A/S | Prodrugs of modulators of the NMDA receptor |
Family Cites Families (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5026700A (en) | 1989-05-16 | 1991-06-25 | Merrell Dow Pharmaceuticals | Certain quinolines and thienopyridines as excitatory amino acid antagonists |
US5252581A (en) | 1992-07-20 | 1993-10-12 | Hoechst-Roussel Pharmaceuticals Inc. | Substituted aminothienopyridines, pharmaceutical composition and use |
US6071970A (en) | 1993-02-08 | 2000-06-06 | Nps Pharmaceuticals, Inc. | Compounds active at a novel site on receptor-operated calcium channels useful for treatment of neurological disorders and diseases |
DE69434889D1 (en) | 1994-02-08 | 2007-01-11 | Nps Pharma Inc | Compounds acting on a new site of receptor-dependent calcium channels for the treatment of neurological disorders |
WO1997046511A1 (en) | 1996-06-07 | 1997-12-11 | Nps Pharmaceuticals, Inc. | Coumpounds active at a novel site on receptor-operated calcium channels useful for treatment of neurological disorders and diseases |
WO1998056752A1 (en) | 1997-06-11 | 1998-12-17 | Nps Pharmaceuticals, Inc. | Compounds active at a novel site on receptor-operated calcium channels useful for treatment of neurological disorders and diseases |
CL2003002287A1 (en) | 2002-11-25 | 2005-01-14 | Wyeth Corp | COMPOUNDS DERIVED FROM TIENO [3,2-b] -PIRIDINA-6-CARBONITRILOS AND TIENEO [2,3-b] -PIRIDINA-5-CARBONITRILS, PHARMACEUTICAL COMPOSITION, PROCEDURE OF PREPARATION AND INTERMEDIARY COMPOUNDS, AND THEIR USE IN THE TREATMENT OF CANCER, APOPLEJIA, OSTEOPOROSIS |
GB0401332D0 (en) | 2004-01-21 | 2004-02-25 | Novartis Ag | Organic compounds |
GB0420719D0 (en) | 2004-09-17 | 2004-10-20 | Addex Pharmaceuticals Sa | Novel allosteric modulators |
US9340555B2 (en) | 2009-09-03 | 2016-05-17 | Allergan, Inc. | Compounds as tyrosine kinase modulators |
CA2789474A1 (en) * | 2010-03-04 | 2011-09-09 | Merck Sharp & Dohme Corp. | Inhibitors of catechol o-methyl transferase and their use in the treatment of psychotic disorders |
US11358971B2 (en) | 2019-07-03 | 2022-06-14 | H. Lundbeck A/S | Prodrugs of modulators of the NMDA receptor |
-
2020
- 2020-06-30 US US16/916,769 patent/US11466027B2/en active Active
- 2020-07-01 WO PCT/EP2020/068522 patent/WO2021001423A1/en unknown
- 2020-07-01 BR BR112021003928-7A patent/BR112021003928A2/en not_active Application Discontinuation
- 2020-07-01 CN CN202080045423.9A patent/CN114008054A/en active Pending
- 2020-07-01 JP JP2021577855A patent/JP2022539197A/en active Pending
- 2020-07-01 MX MX2021015742A patent/MX2021015742A/en unknown
- 2020-07-01 CA CA3144304A patent/CA3144304A1/en active Pending
- 2020-07-01 CR CR20210662A patent/CR20210662A/en unknown
- 2020-07-01 KR KR1020217041215A patent/KR20220029568A/en unknown
- 2020-07-01 MA MA056451A patent/MA56451A/en unknown
- 2020-07-01 TW TW109122237A patent/TW202116779A/en unknown
- 2020-07-01 JO JOP/2021/0331A patent/JOP20210331A1/en unknown
- 2020-07-01 EP EP20740250.4A patent/EP3994141A1/en not_active Withdrawn
- 2020-07-01 PE PE2021002225A patent/PE20220137A1/en unknown
- 2020-07-01 AU AU2020299992A patent/AU2020299992A1/en active Pending
- 2020-07-02 AR ARP200101878A patent/AR119340A1/en unknown
-
2021
- 2021-12-15 CO CONC2021/0017142A patent/CO2021017142A2/en unknown
- 2021-12-29 CL CL2021003557A patent/CL2021003557A1/en unknown
-
2022
- 2022-01-02 IL IL289575A patent/IL289575A/en unknown
- 2022-01-17 EC ECSENADI20223596A patent/ECSP22003596A/en unknown
Also Published As
Publication number | Publication date |
---|---|
BR112021003928A2 (en) | 2021-05-18 |
AU2020299992A1 (en) | 2022-02-24 |
CL2021003557A1 (en) | 2022-08-19 |
CA3144304A1 (en) | 2021-01-07 |
TW202116779A (en) | 2021-05-01 |
US20210002292A1 (en) | 2021-01-07 |
WO2021001423A1 (en) | 2021-01-07 |
PE20220137A1 (en) | 2022-01-27 |
MA56451A (en) | 2022-05-11 |
JOP20210331A1 (en) | 2023-01-30 |
IL289575A (en) | 2022-03-01 |
MX2021015742A (en) | 2022-01-27 |
CO2021017142A2 (en) | 2022-01-17 |
US11466027B2 (en) | 2022-10-11 |
CR20210662A (en) | 2022-03-02 |
EP3994141A1 (en) | 2022-05-11 |
AR119340A1 (en) | 2021-12-09 |
JP2022539197A (en) | 2022-09-07 |
CN114008054A (en) | 2022-02-01 |
KR20220029568A (en) | 2022-03-08 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
SV2016005311A (en) | COMPOUNDS AND COMPOSITIONS AS AGENTS OF THE TOLL TYPE 7 RECEIVER | |
CL2020000422A1 (en) | Compositions of glp-1 and their uses. | |
CL2018003265A1 (en) | Modular of the spiro-lactam n-methyl-d-aspartate receptor and uses thereof. | |
DOP2018000204A (en) | NICOTINIC ACETILCOLINE RECEPTORS ALOSTERIC MODULATORS | |
UY36126A (en) | ? 6,8-DIOXABICICLO COMPOUNDS [3.2.1] OCTANO-2,3-DIOL REPLACED AS ADDRESS AGENTS TO ASGPR ?. | |
DOP2017000117A (en) | 2-AMINO-6- (DIFLUOROMETIL) - 5,5-DIFLUORO-6-PHENYL-3,4,5,6-TETRAHYDROPIRIDINES AS INHIBITORS OF BACE1 | |
CL2015002121A1 (en) | Modular spiro-lactam nmda receptors and their uses. | |
CR20190392A (en) | Aryl hydrocarbon receptor (ahr) modulator compounds | |
DOP2014000230A (en) | AGENTS TO TREAT DISORDERS THAT INVOLVE THE MODULATION OF RIANODINE RECEPTORS | |
CL2022000201A1 (en) | akr1c3-dependent tricyclic inhibitors of kars | |
CO2019012767A2 (en) | Phenyl-2-hydroxy-acetylamino-2-methyl-phenyl compound | |
CR20190393A (en) | Aryl hydrocarbon receptor (ahr) modulator compounds | |
CL2018001210A1 (en) | Novel cryptophycin compounds and conjugated products, their preparation and therapeutic use. | |
CO2021014008A2 (en) | Pharmaceutical Compounds for the Treatment of Complement-Mediated Disorders | |
CL2020001140A1 (en) | Spirocyclic compounds as modulators of the x-farnesoid receptor. | |
CL2021002357A1 (en) | Fused and Related Bicyclic Piperidinyl Compounds as Modulators of the c5a Receptor | |
UY37729A (en) | NEW COMPOUNDS THAT INHIBIT THE ACTIVITY OF Nav1.7 | |
CL2015002545A1 (en) | New phosphodiesterase inhibitor compounds of type 10a. | |
CL2021000930A1 (en) | Novel Pyridazines | |
ECSP22003596A (en) | NMDA RECEPTOR MODULATORS | |
CL2021003534A1 (en) | Prodrugs of nmda receptor modulators. | |
CO2021001174A2 (en) | Ckd8 / 19 inhibitors | |
CR20170195A (en) | ESPIRO-TIAZOLONAS | |
DOP2022000026A (en) | ALCOHOL DERIVATIVES AS KV7 POTASSIUM CHANNEL OPENERS | |
UY38217A (en) | DERIVATIVES OF 1-IMIDAZOTIADIAZOL-2H-PIRROL-5-ONA |